IL77506A - Aqueous formulations of piperazino-fluoro-oxo-quinolinecarboxylic acid,analogs thereof and their preparation - Google Patents

Aqueous formulations of piperazino-fluoro-oxo-quinolinecarboxylic acid,analogs thereof and their preparation

Info

Publication number
IL77506A
IL77506A IL77506A IL7750686A IL77506A IL 77506 A IL77506 A IL 77506A IL 77506 A IL77506 A IL 77506A IL 7750686 A IL7750686 A IL 7750686A IL 77506 A IL77506 A IL 77506A
Authority
IL
Israel
Prior art keywords
piperazino
analogs
oxo
fluoro
preparation
Prior art date
Application number
IL77506A
Other languages
English (en)
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=25828371&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IL77506(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of IL77506A publication Critical patent/IL77506A/xx

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/02—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/08—Solutions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Inorganic Chemistry (AREA)
  • Dermatology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Quinoline Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Silicon Polymers (AREA)
  • Noodles (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
IL77506A 1985-01-05 1986-01-02 Aqueous formulations of piperazino-fluoro-oxo-quinolinecarboxylic acid,analogs thereof and their preparation IL77506A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE3500243 1985-01-05
DE19853517709 DE3517709A1 (de) 1985-01-05 1985-05-17 Basische zubereitungen von chinoloncarbonsaeuren

Publications (1)

Publication Number Publication Date
IL77506A true IL77506A (en) 1990-03-19

Family

ID=25828371

Family Applications (1)

Application Number Title Priority Date Filing Date
IL77506A IL77506A (en) 1985-01-05 1986-01-02 Aqueous formulations of piperazino-fluoro-oxo-quinolinecarboxylic acid,analogs thereof and their preparation

Country Status (18)

Country Link
US (1) US4772605A (hu)
EP (1) EP0187315B1 (hu)
KR (1) KR890002240B1 (hu)
CN (2) CN1011572B (hu)
AT (1) ATE62595T1 (hu)
AU (1) AU563777B2 (hu)
CA (1) CA1273578A (hu)
DE (2) DE3517709A1 (hu)
DK (1) DK165666C (hu)
ES (3) ES8802423A1 (hu)
FI (1) FI87425C (hu)
GR (1) GR860008B (hu)
HU (1) HU194735B (hu)
IE (1) IE58450B1 (hu)
IL (1) IL77506A (hu)
NO (1) NO172674C (hu)
PH (1) PH25649A (hu)
PT (1) PT81792B (hu)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3705621C2 (de) * 1986-02-25 1997-01-09 Otsuka Pharma Co Ltd Heterocyclisch substituierte Chinoloncarbonsäurederivate
JPH0696533B2 (ja) * 1987-01-14 1994-11-30 北陸製薬株式会社 キノロンカルボン酸の水性組成物
JPH01175935A (ja) * 1987-12-28 1989-07-12 Kyorin Pharmaceut Co Ltd 凍結乾燥注射剤
JPH0228178A (ja) * 1988-04-23 1990-01-30 Toyama Chem Co Ltd 新規なピリドンカルボン酸誘導体およびその塩並びにそれらの製造法
DE3902079A1 (de) * 1988-04-15 1989-10-26 Bayer Ag I.m. injektionsformen von gyrase-inhibitoren
US5225413A (en) * 1988-09-16 1993-07-06 Bayer-Aktiengesellschaft pH-neutral aqueous solutions of quinolone-carboxylic acids
US4978661A (en) * 1988-09-29 1990-12-18 Innocenzo Caruso Use of 6-halo-4-quinolone compounds and pharmaceutical compositions thereof for the preparation of a medicament for the therapeutical application in rheumatoid arthritis
US5262417A (en) * 1988-12-06 1993-11-16 The Upjohn Company Antibacterial quinolone compounds
FR2655545B1 (fr) * 1989-12-11 1994-06-10 Rhone Poulenc Sante Nouvelle application therapeutique des derives des fluoroquinolones.
US5084276A (en) * 1990-01-05 1992-01-28 Abbott Laboratories Quinolone carboxylic acid compositions with polymeric additive to reduce vein irritation
KR0159540B1 (ko) * 1992-01-21 1998-12-01 김정순 퀴놀론-카복실산의 염 및 그 함유조성물
IT1270836B (it) * 1993-10-27 1997-05-13 Archimica Spa Procedimento per la preparazione di rufloxacina e suoi sali
EP0868183B1 (en) * 1995-12-21 2002-01-30 Pfizer Inc. Injectable quinolone formulations
IN186245B (hu) 1997-09-19 2001-07-14 Ranbaxy Lab Ltd
ID21415A (id) 1997-12-05 1999-06-10 Upjohn Co Senyawa-senyawa antibiotik magnesium quinolon
JP4331944B2 (ja) * 2001-04-17 2009-09-16 大日本住友製薬株式会社 新規アデニン誘導体
US6872723B2 (en) * 2002-01-28 2005-03-29 Wyeth Stabilized difloxacin injectable solution
CN101480384A (zh) * 2002-12-17 2009-07-15 阿伯特有限及两合公司 包含非诺贝酸、其生理可接受的盐或衍生物的制剂
US20080051411A1 (en) * 2002-12-17 2008-02-28 Cink Russell D Salts of Fenofibric Acid and Pharmaceutical Formulations Thereof
US20060073117A1 (en) * 2004-10-01 2006-04-06 Stowers Institute For Medical Research Methods and compositions for controlling hair follicle stem cell fate
DE102004054873A1 (de) 2004-11-12 2006-05-18 Bayer Healthcare Ag Behandlung von Mastitis
DE102006010642A1 (de) * 2006-03-08 2007-09-27 Bayer Healthcare Aktiengesellschaft Arzneimittelformulierungen, enthaltend Fluorchinolone
GB2480276A (en) * 2010-05-11 2011-11-16 Michael Hilary Burke Process for the preparation of an aqueous injectable enrofloxacin antimicrobial formulation
EP3034078A1 (en) 2010-09-27 2016-06-22 Emergent Product Development Gaithersburg Inc. 2-pyridone antimicrobial compositions

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6019910B2 (ja) * 1979-10-11 1985-05-18 大塚製薬株式会社 ベンゾ〔ｉｊ〕キノリジン−２−カルボン酸誘導体及びその製造法
DE2953974C2 (hu) * 1978-04-12 1992-06-25 Otsuka Pharmaceutical Co., Ltd., Tokio/Tokyo, Jp
AR223983A1 (es) * 1978-08-25 1981-10-15 Dainippon Pharmaceutical Co Un procedimiento para-preparar derivados de acido 6-halogeno-4-oxo-7-(1-piperazinil)-1,8-naftiridin-3-carboxilico
JPS5551422A (en) * 1978-10-11 1980-04-15 Takeda Chem Ind Ltd Deodorization
JPS5746986A (en) * 1980-09-02 1982-03-17 Dai Ichi Seiyaku Co Ltd Pyrido(1,2,3-de)(1,4)benzoxazine derivative
DE3142854A1 (de) * 1981-10-29 1983-05-11 Bayer Ag, 5090 Leverkusen 1-cyclopropyl-6-fluor-1,4-dihydro-4-oxo-7-piperazino-chinolin-3-carbonsaeuren, verfahren zu ihrer herstellung sowie diese enthaltende antibakterielle mittel
DE3033157A1 (de) * 1980-09-03 1982-04-01 Bayer Ag, 5090 Leverkusen 7-amino-1-cyclopropyl-4-oxo-1,4-dihydro-naphthyridin-3-carbonsaeuren, verfahren zu ihrer herstellung sowie diese enthaltende antibakterielle mittel
US4404197A (en) * 1981-05-15 1983-09-13 Fox Jr Charles L Antimicrobial compositions containing 1-ethyl-6-fluoro-1,4-dihydro-4-dihydro-4-oxo-7-(1-piperazinyl)-3-quinoline carboxylic acid or metal salts thereof and silver sulfadiazine
HU188181B (en) * 1981-06-11 1986-03-28 Warner-Lambert Co,Us Process for producing salts of naphtiridine and quinoline compounds of antimicrobial activity
DE3225367A1 (de) * 1982-07-07 1984-01-12 Hoechst Ag, 6230 Frankfurt Arzneimittel zur behandlung von infektioes bedingten diarrhoeen
US4551456A (en) * 1983-11-14 1985-11-05 Merck & Co., Inc. Ophthalmic use of norfloxacin and related antibiotics

Also Published As

Publication number Publication date
DE3582575D1 (de) 1991-05-23
AU563777B2 (en) 1987-07-23
CN1011572B (zh) 1991-02-13
PT81792A (en) 1986-02-01
FI87425C (fi) 1993-01-11
EP0187315B1 (de) 1991-04-17
FI860010A (fi) 1986-07-06
HU194735B (en) 1988-03-28
DE3517709A1 (de) 1986-07-10
CA1273578A (en) 1990-09-04
ATE62595T1 (de) 1991-05-15
FI87425B (fi) 1992-09-30
ES557771A0 (es) 1988-04-01
NO172674C (no) 1993-08-25
ES557770A0 (es) 1989-03-16
KR860005635A (ko) 1986-08-11
PT81792B (pt) 1988-05-27
DK2386A (da) 1986-07-06
CN1040143A (zh) 1990-03-07
DK165666B (da) 1993-01-04
EP0187315A2 (de) 1986-07-16
AU5104685A (en) 1986-07-10
IE58450B1 (en) 1993-09-22
KR890002240B1 (ko) 1989-06-26
ES550668A0 (es) 1988-06-01
NO172674B (no) 1993-05-18
HUT40329A (en) 1986-12-28
ES8802150A1 (es) 1988-04-01
EP0187315A3 (en) 1987-08-12
DK2386D0 (da) 1986-01-03
GR860008B (en) 1986-04-25
ES8900196A1 (es) 1989-03-16
NO855094L (no) 1986-07-07
US4772605A (en) 1988-09-20
IE860018L (en) 1986-07-05
ES8802423A1 (es) 1988-06-01
DK165666C (da) 1993-06-01
FI860010A0 (fi) 1986-01-02
CN85109451A (zh) 1986-09-10
PH25649A (en) 1991-08-21

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