IL76778A - Synthesis of 7-halo-7-deoxylincomycins - Google Patents

Synthesis of 7-halo-7-deoxylincomycins

Info

Publication number
IL76778A
IL76778A IL76778A IL7677885A IL76778A IL 76778 A IL76778 A IL 76778A IL 76778 A IL76778 A IL 76778A IL 7677885 A IL7677885 A IL 7677885A IL 76778 A IL76778 A IL 76778A
Authority
IL
Israel
Prior art keywords
deoxylincomycins
halo
synthesis
analogue
halodeoxylincomycin
Prior art date
Application number
IL76778A
Other languages
English (en)
Other versions
IL76778A0 (en
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of IL76778A0 publication Critical patent/IL76778A0/xx
Publication of IL76778A publication Critical patent/IL76778A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/02—Acyclic radicals, not substituted by cyclic structures
    • C07H15/14—Acyclic radicals, not substituted by cyclic structures attached to a sulfur, selenium or tellurium atom of a saccharide radical
    • C07H15/16—Lincomycin; Derivatives thereof

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Peptides Or Proteins (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Cephalosporin Compounds (AREA)
  • Indole Compounds (AREA)
IL76778A 1984-11-29 1985-10-22 Synthesis of 7-halo-7-deoxylincomycins IL76778A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US67615784A 1984-11-29 1984-11-29

Publications (2)

Publication Number Publication Date
IL76778A0 IL76778A0 (en) 1986-02-28
IL76778A true IL76778A (en) 1991-09-16

Family

ID=24713464

Family Applications (1)

Application Number Title Priority Date Filing Date
IL76778A IL76778A (en) 1984-11-29 1985-10-22 Synthesis of 7-halo-7-deoxylincomycins

Country Status (19)

Country Link
US (1) US4710565A (xx)
EP (1) EP0183505B1 (xx)
JP (1) JPH0649714B2 (xx)
KR (1) KR930003492B1 (xx)
CN (2) CN1004002B (xx)
AT (1) ATE50265T1 (xx)
AU (1) AU574232B2 (xx)
CA (1) CA1238319A (xx)
DE (1) DE3575930D1 (xx)
DK (1) DK165010C (xx)
ES (1) ES8605817A1 (xx)
FI (1) FI78708C (xx)
GR (1) GR852861B (xx)
HU (1) HU199497B (xx)
IL (1) IL76778A (xx)
MX (1) MX162251A (xx)
PT (1) PT81496B (xx)
SU (1) SU1405705A3 (xx)
ZA (1) ZA858117B (xx)

Families Citing this family (30)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4568741A (en) * 1984-05-15 1986-02-04 The Upjohn Company Synthesis of 7-halo-7-deoxylincomycins
JP2531876Y2 (ja) * 1988-12-15 1997-04-09 日東工器株式会社 電磁式ダイアフラムポンプ用マグネットホルダ
JP2531877Y2 (ja) * 1988-12-15 1997-04-09 日東工器株式会社 電磁式ダイアフラムポンプ
JP2544782Y2 (ja) * 1988-12-27 1997-08-20 日東工器株式会社 電磁式ダイアフラムポンプ用マグネットホルダ
US6565882B2 (en) 2000-02-24 2003-05-20 Advancis Pharmaceutical Corp Antibiotic composition with inhibitor
US6544555B2 (en) 2000-02-24 2003-04-08 Advancis Pharmaceutical Corp. Antibiotic product, use and formulation thereof
US6541014B2 (en) 2000-10-13 2003-04-01 Advancis Pharmaceutical Corp. Antiviral product, use and formulation thereof
US20020068078A1 (en) 2000-10-13 2002-06-06 Rudnic Edward M. Antifungal product, use and formulation thereof
BR0212214A (pt) * 2001-08-28 2004-10-19 Pharmacia Corp Base livre de clindamicina cristalina
JP2006504673A (ja) * 2002-08-15 2006-02-09 バイクロン ファーマシューティカルズ， インコーポレイテッド 抗菌活性を有するリンコマイシン誘導体
US7199105B2 (en) * 2002-08-15 2007-04-03 Vicuron Pharmaceuticals, Inc. Lincomycin derivatives possessing antibacterial activity
CA2513773C (en) 2003-01-24 2013-03-26 Connetics Australia Pty Ltd Clindamycin phosphate foam
US7199106B2 (en) 2003-06-17 2007-04-03 Vicuron Pharmaceuticals, Inc. Lincomycin derivatives possessing antimicrobial activity
US7256177B2 (en) 2003-06-17 2007-08-14 Vicuron Pharmaceuticals, Inc. Lincomycin derivatives possessing antibacterial activity
EP1648407A4 (en) 2003-07-21 2011-08-31 Middlebrook Pharmaceuticals Inc ANTIBIOTIC PRODUCT, CORRESPONDING USE AND FORMULATION
JP2006528185A (ja) 2003-07-21 2006-12-14 アドバンシス ファーマスーティカル コーポレイション 抗生物質製剤、その使用法及び作成方法
WO2005009365A2 (en) 2003-07-21 2005-02-03 Advancis Pharmaceutical Corporation Antibiotic product, use and formulation thereof
AU2004264939A1 (en) 2003-08-11 2005-02-24 Middlebrook Pharmaceuticals, Inc. Robust pellet
JP2007502294A (ja) 2003-08-12 2007-02-08 アドバンシス ファーマスーティカル コーポレイション 抗生物質製剤、その使用法及び作成方法
CA2535780A1 (en) 2003-08-29 2005-03-17 Advancis Pharmaceuticals Corporation Antibiotic product, use and formulation thereof
AU2004273830B2 (en) 2003-09-15 2011-03-24 Shionogi, Inc. Antibiotic product, use and formulation thereof
US7361743B2 (en) * 2004-02-11 2008-04-22 Pfizer Inc Lincomycin derivatives possessing antibacterial activity
AU2005269981A1 (en) 2004-07-02 2006-02-09 Bonck, John A Tablet for pulsed delivery
US8357394B2 (en) 2005-12-08 2013-01-22 Shionogi Inc. Compositions and methods for improved efficacy of penicillin-type antibiotics
US8778924B2 (en) 2006-12-04 2014-07-15 Shionogi Inc. Modified release amoxicillin products
MX2008010982A (es) * 2006-02-28 2008-10-21 V B Medicare Private Ltd Reactivo novedosos de cloracion y proceso novedoso para la cloracion de azucares que usa cloruro de tionilo.
BRPI0709674A2 (pt) 2006-03-31 2011-12-06 Stiefel Res Australia Pty Ltd gel de suspensão espumante
US8299052B2 (en) 2006-05-05 2012-10-30 Shionogi Inc. Pharmaceutical compositions and methods for improved bacterial eradication
CN101205245B (zh) * 2007-12-06 2011-04-06 河南天方药业股份有限公司 盐酸克林霉素的制备方法
CN102675146A (zh) * 2012-05-22 2012-09-19 山东凯盛新材料股份有限公司 新型固体氯化剂（氯亚甲基）二甲基氯化铵的制备方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3496163A (en) * 1965-02-08 1970-02-17 Upjohn Co 7-halo-7-deoxylincomycins and process for preparing the same
US3435025A (en) * 1966-03-18 1969-03-25 Upjohn Co 7-deoxylincomycin and analogs and isomers thereof and process for making the same
US3580904A (en) * 1969-04-03 1971-05-25 Upjohn Co 7-halo-7-deoxy-lincomycin derivatives
US3574186A (en) * 1969-10-08 1971-04-06 Upjohn Co Process for making 7-chloro-7-deoxylincomycin and related compounds and novel intermediates produced therein
US4568741A (en) * 1984-05-15 1986-02-04 The Upjohn Company Synthesis of 7-halo-7-deoxylincomycins

Also Published As

Publication number Publication date
FI78708C (fi) 1989-09-11
AU574232B2 (en) 1988-06-30
IL76778A0 (en) 1986-02-28
CN85101921A (zh) 1987-01-10
PT81496B (pt) 1987-11-11
EP0183505A3 (en) 1987-06-24
DE3575930D1 (de) 1990-03-15
KR860004077A (ko) 1986-06-16
CN85108244A (zh) 1986-08-20
ES548152A0 (es) 1986-04-01
EP0183505B1 (en) 1990-02-07
US4710565A (en) 1987-12-01
FI78708B (fi) 1989-05-31
GR852861B (xx) 1986-03-28
SU1405705A3 (ru) 1988-06-23
MX162251A (es) 1991-04-17
FI854711A0 (fi) 1985-11-28
AU4883785A (en) 1986-06-05
KR930003492B1 (ko) 1993-05-01
DK165010B (da) 1992-09-28
ES8605817A1 (es) 1986-04-01
PT81496A (en) 1985-12-01
DK542785A (da) 1986-05-30
JPH0649714B2 (ja) 1994-06-29
EP0183505A2 (en) 1986-06-04
HUT40806A (en) 1987-02-27
DK542785D0 (da) 1985-11-22
JPS61137892A (ja) 1986-06-25
CA1238319A (en) 1988-06-21
ATE50265T1 (de) 1990-02-15
DK165010C (da) 1993-02-22
CN1004002B (zh) 1989-04-26
CN1016694B (zh) 1992-05-20
HU199497B (en) 1990-02-28
ZA858117B (en) 1986-06-25
FI854711A (fi) 1986-05-30

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Legal Events

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