IL67530A - 1,1-alkanediol dicarboxylate linked penicillins and pharmaceutical compositions containing them - Google Patents

1,1-alkanediol dicarboxylate linked penicillins and pharmaceutical compositions containing them

Info

Publication number
IL67530A
IL67530A IL67530A IL6753082A IL67530A IL 67530 A IL67530 A IL 67530A IL 67530 A IL67530 A IL 67530A IL 6753082 A IL6753082 A IL 6753082A IL 67530 A IL67530 A IL 67530A
Authority
IL
Israel
Prior art keywords
alkanediol
penicillins
pharmaceutical compositions
compositions containing
dicarboxylate
Prior art date
Application number
IL67530A
Other languages
English (en)
Other versions
IL67530A0 (en
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of IL67530A0 publication Critical patent/IL67530A0/xx
Publication of IL67530A publication Critical patent/IL67530A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D499/28—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with modified 2-carboxyl group
    • C07D499/32—Esters
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Cephalosporin Compounds (AREA)
IL67530A 1981-12-22 1982-12-21 1,1-alkanediol dicarboxylate linked penicillins and pharmaceutical compositions containing them IL67530A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US33402281A 1981-12-22 1981-12-22
US06/429,915 US4457924A (en) 1981-12-22 1982-09-30 1,1-Alkanediol dicarboxylate linked antibacterial agents

Publications (2)

Publication Number Publication Date
IL67530A0 IL67530A0 (en) 1983-05-15
IL67530A true IL67530A (en) 1986-02-28

Family

ID=26989011

Family Applications (1)

Application Number Title Priority Date Filing Date
IL67530A IL67530A (en) 1981-12-22 1982-12-21 1,1-alkanediol dicarboxylate linked penicillins and pharmaceutical compositions containing them

Country Status (25)

Country Link
US (1) US4457924A (es)
EP (1) EP0083484B1 (es)
JP (1) JPH02270881A (es)
KR (1) KR860001370B1 (es)
AU (1) AU537214B2 (es)
BG (4) BG50161A3 (es)
CA (1) CA1213582A (es)
DD (1) DD207379A5 (es)
DE (1) DE3269267D1 (es)
DK (3) DK565482A (es)
ES (3) ES8402310A1 (es)
FI (1) FI80039C (es)
GR (1) GR77066B (es)
GT (1) GT198200058A (es)
HU (1) HU187737B (es)
IE (1) IE54333B1 (es)
IL (1) IL67530A (es)
NO (1) NO824305L (es)
NZ (1) NZ202670A (es)
PH (1) PH18311A (es)
PL (3) PL141306B1 (es)
PT (1) PT76012B (es)
RO (2) RO87709A (es)
SU (1) SU1405704A3 (es)
YU (2) YU43111B (es)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4675186A (en) 1985-04-18 1987-06-23 Pfizer Inc. 6-(1-acyl-1-hydroxymethyl)penicillanic acid derivatives
LU87821A1 (fr) * 1990-10-12 1992-05-25 Cird Galderma Composes bi-aromatiques,et leur utilisation en medecine humaine et veterinaire et en cosmetique
ATE115114T1 (de) * 1991-03-11 1994-12-15 Schweizerhall Saeurefab Verfahren zur herstellung von chlorierten carbonsäureestern.
DK0508943T3 (da) * 1991-03-11 1995-01-30 Schweizerhall Saeurefab Fremgangsmåde til fremstilling af halogenerede carboxylsyreestere
AU2003301426A1 (en) * 2002-10-18 2004-05-04 Meiji Seika Kaisha, Ltd. Malonic acid monoesters and process for producing the same
EP2508504B1 (en) * 2009-12-01 2016-04-13 Sumitomo Chemical Co., Ltd Process for preparation of cycloalkanedicarboxylic acid monoesters
US7973194B1 (en) 2010-03-18 2011-07-05 Eastman Chemical Company High solvating cyclohexane dicarboxylate diesters plasticizers
CN115385934A (zh) * 2022-10-26 2022-11-25 北京纳百生物科技有限公司 一种舒巴坦半抗原及其合成方法和应用

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2985648A (en) * 1958-10-06 1961-05-23 Doyle Frank Peter Alpha-aminobenzylpenicillins
DE1249280B (de) * 1962-11-02 1967-09-07 Beecham GrouD Limited, Brentford Middlesex (Großbritannien) Verfahren zur Herstellung von Hydroxybenzyl y amino-pemciUmen
US3520876A (en) * 1967-11-01 1970-07-21 American Home Prod Process for the preparation of 6-(alpha-aminoacylamino)penicillanic acids
ES436565A1 (es) * 1974-06-05 1977-04-01 Bristol Myers Co Un procedimiento para la preparacion de acidos acetamidope- nicilanicos.
FR2290443A1 (fr) * 1974-11-06 1976-06-04 Aries Robert Nouveaux esters bispenicillaniques
FR2309570A1 (fr) * 1975-04-29 1976-11-26 Aries Robert Derives polymeriques des penicillines et cephalosporines
GB1569421A (en) * 1976-06-11 1980-06-18 Beecham Group Ltd Penicillin compositions
US4234579A (en) * 1977-06-07 1980-11-18 Pfizer Inc. Penicillanic acid 1,1-dioxides as β-lactamase inhibitors
IE49881B1 (en) * 1979-02-13 1986-01-08 Leo Pharm Prod Ltd B-lactam intermediates
US4244951A (en) * 1979-05-16 1981-01-13 Pfizer Inc. Bis-esters of methanediol with penicillins and penicillanic acid 1,1-dioxide
US4309347A (en) * 1979-05-16 1982-01-05 Pfizer Inc. Penicillanoyloxymethyl penicillanate 1,1,1',1'-tetraoxide

Also Published As

Publication number Publication date
ES8503001A1 (es) 1985-02-01
ES8530002A1 (es) 1985-02-01
ES518425A0 (es) 1984-02-01
PL141306B1 (en) 1987-07-31
FI824409L (fi) 1983-06-23
NZ202670A (en) 1985-12-13
GT198200058A (es) 1984-06-09
RO87709B (ro) 1985-10-01
ES8402310A1 (es) 1984-02-01
RO84911A (ro) 1984-08-17
SU1405704A3 (ru) 1988-06-23
NO824305L (no) 1983-06-23
DK69192D0 (da) 1992-05-26
DE3269267D1 (en) 1986-03-27
RO87709A (ro) 1985-10-31
US4457924A (en) 1984-07-03
EP0083484A1 (en) 1983-07-13
YU43992B (en) 1990-02-28
PL248637A1 (en) 1985-02-27
BG48694A3 (en) 1991-04-15
DK69192A (da) 1992-05-26
BG50162A3 (en) 1992-05-15
RO84911B (ro) 1984-09-30
IE54333B1 (en) 1989-08-30
CA1213582A (en) 1986-11-04
AU537214B2 (en) 1984-06-14
BG50161A3 (en) 1992-05-15
PL145927B1 (en) 1988-11-30
PT76012B (en) 1985-12-13
YU43111B (en) 1989-02-28
DK69092A (da) 1992-05-26
EP0083484B1 (en) 1986-02-19
BG50160A3 (en) 1992-05-15
PT76012A (en) 1983-01-01
YU284482A (en) 1985-03-20
FI824409A0 (fi) 1982-12-21
IE823034L (en) 1983-06-22
GR77066B (es) 1984-04-05
ES524894A0 (es) 1985-02-01
YU183084A (en) 1986-10-31
DK69092D0 (da) 1992-05-26
DK565482A (da) 1983-06-23
ES524895A0 (es) 1985-02-01
PL140291B1 (en) 1987-04-30
FI80039C (fi) 1990-04-10
AU9172182A (en) 1983-06-30
DD207379A5 (de) 1984-02-29
HU187737B (en) 1986-02-28
IL67530A0 (en) 1983-05-15
PH18311A (en) 1985-05-29
FI80039B (fi) 1989-12-29
KR860001370B1 (ko) 1986-09-17
KR840002840A (ko) 1984-07-21
JPH02270881A (ja) 1990-11-05
PL239651A1 (en) 1985-01-16

Similar Documents

Publication Publication Date Title
IL65056A0 (en) Imidazodiazepines,their manufacture and pharmaceutical compositions containing them
IL66501A (en) Benzazepine-2-one derivatives,their manufacture and pharmaceutical compositions containing them
DE3265978D1 (en) 1,4-dihydropyridine derivative and pharmaceutical composition containing same
DE3267350D1 (en) 5,6,7-trinor-4,8-inter-m-phenylene pgi derivatives and pharmaceutical compositions containing them
PT74923A (en) Process for preparing substituted 1,2-diaminocyclobutene-3,4-diones and pharmaceutical compositions containing the same
IL65167A (en) N-acyl-polypeptides,their production and pharmaceutical compositions containing them
IL72566A (en) Androst-5-en-17-one and 5alpha-androstan-17-one derivatives and pharmaceutical compositions containing the same
IL64847A0 (en) Hexapyranose compounds,their manufacture and pharmaceutical compositions containing them
IL65076A (en) 3,4-dihydro-5h-2,3-benzo-diazepine derivatives,their preparation and pharmaceutical compositions containing them
NZ201520A (en) Substituted aminopyridazines and pharmaceutical compositions
IL63801A0 (en) 2-amino-3-carbethoxyamino-6-(p-fluorobenzylamino)-pyridine-maleate,its production and pharmaceutical compositions containing it
IL61930A (en) 25-hydroxy-26,26,26,27,27,27-hexafluorocholecalciferol and pharmaceutical compositions containing it
IL63368A0 (en) 4,5-diaryl-alpha-polyfluoroalkyl-1h-imidazole-2-methanamines,their preparation and pharmaceutical compositions containing them
IL72054A0 (en) Beta-lactam derivative,its preparation and pharmaceutical compositions containing it
IL72562A (en) 6,7-dimethoxy-4-piperidino-quinazoline derivatives and pharmaceutical compositions containing them
PH16982A (en) Penicillanoyloxymethyl penicillanate 1,1,1',1'-tetraoxide and its pharmaceutical composition
IL67284A (en) N-substituted-2-pyridylindoles,their manufacture and pharmaceutical compositions containing them
EP0180190A3 (en) 3,4-dihydrobenzopyran compounds and pharmaceutical composition containing the same
IL67530A0 (en) 1,1-alkanediol dicarboxylate linked penicillins and pharmaceutical compositions containing them
DE3265871D1 (en) 3-amino-2-hydroxy-4-phenylbutanoic acid derivatives and pharmaceutical composition containing the same
JPS6468379A (en) Novel compound, its production and pharmaceutical composition containing the same
IL77426A (en) 2,6-dimethyl-8alpha-pivaloyl-amino-9,10-didehydro-ergoline,its production and pharmaceutical compositions containing it
IL67715A (en) 3,3-dialkyl-and 3,3-alkyleneindolene derivatives,their production and pharmaceutical compositions containing them
IL64755A0 (en) Cycloheptene derivatives,their manufacture and pharmaceutical compositions containing them
IL61862A0 (en) 4,5-diaryl- -(polyhaloalkyl)-1h-imidazole-2-methanols,their preparation and pharmaceutical compositions containing them