IL220921B - 8-Fluoro-2-{4-[(methylamino)methyl]phenyl}-5,4,3,1-tetrahydro-h6-azepino[3,4,5-dc]indole-6-one camislate salt - Google Patents

8-Fluoro-2-{4-[(methylamino)methyl]phenyl}-5,4,3,1-tetrahydro-h6-azepino[3,4,5-dc]indole-6-one camislate salt

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Publication number
IL220921B
IL220921B IL220921A IL22092112A IL220921B IL 220921 B IL220921 B IL 220921B IL 220921 A IL220921 A IL 220921A IL 22092112 A IL22092112 A IL 22092112A IL 220921 B IL220921 B IL 220921B
Authority
IL
Israel
Prior art keywords
azepino
indol
methylamino
tetrahydro
fluoro
Prior art date
Application number
IL220921A
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English (en)
Hebrew (he)
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Pfizer
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43859823&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IL220921(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer filed Critical Pfizer
Publication of IL220921B publication Critical patent/IL220921B/en

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    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
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    • C07C309/02Sulfonic acids having sulfo groups bound to acyclic carbon atoms
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    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C57/00Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms
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    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/06Peri-condensed systems
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    • C07B2200/13Crystalline forms, e.g. polymorphs

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
IL220921A 2010-02-12 2012-07-12 8-Fluoro-2-{4-[(methylamino)methyl]phenyl}-5,4,3,1-tetrahydro-h6-azepino[3,4,5-dc]indole-6-one camislate salt IL220921B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US30427710P 2010-02-12 2010-02-12
PCT/IB2011/050571 WO2011098971A1 (en) 2010-02-12 2011-02-10 Salts and polymorphs of 8-fluoro-2-{4-[(methylamino}methyl]phenyl}-1,3,4,5-tetrahydro-6h-azepino[5,4,3-cd]indol-6-one

Publications (1)

Publication Number Publication Date
IL220921B true IL220921B (en) 2020-03-31

Family

ID=43859823

Family Applications (1)

Application Number Title Priority Date Filing Date
IL220921A IL220921B (en) 2010-02-12 2012-07-12 8-Fluoro-2-{4-[(methylamino)methyl]phenyl}-5,4,3,1-tetrahydro-h6-azepino[3,4,5-dc]indole-6-one camislate salt

Country Status (32)

Country Link
US (5) US8754072B2 (hr)
EP (4) EP3597651A1 (hr)
JP (6) JP5745283B2 (hr)
KR (2) KR102108226B1 (hr)
CN (2) CN104876937B (hr)
AR (2) AR080164A1 (hr)
AU (1) AU2011213944B2 (hr)
BR (1) BR112012019050B1 (hr)
CA (2) CA3024216C (hr)
CY (3) CY1118319T1 (hr)
DK (2) DK2534153T4 (hr)
ES (2) ES2753748T3 (hr)
FI (1) FI2534153T4 (hr)
HK (1) HK1176617A1 (hr)
HR (2) HRP20161742T4 (hr)
HU (3) HUE030969T2 (hr)
IL (1) IL220921B (hr)
LT (3) LT2534153T (hr)
LU (1) LUC00093I2 (hr)
MX (1) MX343383B (hr)
NL (1) NL300958I2 (hr)
NO (1) NO2018039I1 (hr)
NZ (1) NZ601445A (hr)
PL (2) PL2534153T3 (hr)
PT (2) PT2534153T (hr)
RS (2) RS55487B2 (hr)
RU (1) RU2570198C2 (hr)
SG (2) SG182533A1 (hr)
SI (2) SI2534153T2 (hr)
SM (1) SMT201600462B (hr)
TW (1) TWI545123B (hr)
WO (1) WO2011098971A1 (hr)

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BR112022000337A2 (pt) 2019-07-10 2022-04-12 Cybrexa 2 Inc Conjugados de peptídeos de citotoxinas como terapêuticos
CN111004244A (zh) * 2019-12-27 2020-04-14 重庆市碚圣医药科技股份有限公司 一种瑞卡帕布樟脑磺酸盐的合成方法
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