IL193322A - Derivatives of 4– (3 – benzoylaminophenyl) –7,6 – domethoxy – 2– methylaminoquinazoline - Google Patents

Derivatives of 4– (3 – benzoylaminophenyl) –7,6 – domethoxy – 2– methylaminoquinazoline

Info

Publication number
IL193322A
IL193322A IL193322A IL19332208A IL193322A IL 193322 A IL193322 A IL 193322A IL 193322 A IL193322 A IL 193322A IL 19332208 A IL19332208 A IL 19332208A IL 193322 A IL193322 A IL 193322A
Authority
IL
Israel
Prior art keywords
salt
compound
hydrate
dimethoxy
methylaminoquinazolin
Prior art date
Application number
IL193322A
Other languages
English (en)
Hebrew (he)
Other versions
IL193322A0 (en
Inventor
Kazuki Miyazaki
Kazutomi Kusano
Yasutaka Takase
Osamu Asano
Manabu Shirato
Hisashi Wakita
Takao Saeki
Naoto Ishii
Original Assignee
Eisai R&D Man Co Ltd
Kazuki Miyazaki
Kazutomi Kusano
Yasutaka Takase
Osamu Asano
Manabu Shirato
Hisashi Wakita
Takao Saeki
Naoto Ishii
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/JP2007/053066 external-priority patent/WO2007097317A1/ja
Application filed by Eisai R&D Man Co Ltd, Kazuki Miyazaki, Kazutomi Kusano, Yasutaka Takase, Osamu Asano, Manabu Shirato, Hisashi Wakita, Takao Saeki, Naoto Ishii filed Critical Eisai R&D Man Co Ltd
Publication of IL193322A0 publication Critical patent/IL193322A0/en
Publication of IL193322A publication Critical patent/IL193322A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/78Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 2
    • C07D239/84Nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
IL193322A 2006-02-21 2008-08-07 Derivatives of 4– (3 – benzoylaminophenyl) –7,6 – domethoxy – 2– methylaminoquinazoline IL193322A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2006043273 2006-02-21
PCT/JP2007/053066 WO2007097317A1 (ja) 2006-02-21 2007-02-20 4-(3-ベンゾイルアミノフェニル)-6,7-ジメトキシ-2-メチルアミノキナゾリン誘導体

Publications (2)

Publication Number Publication Date
IL193322A0 IL193322A0 (en) 2009-05-04
IL193322A true IL193322A (en) 2014-04-30

Family

ID=42137992

Family Applications (1)

Application Number Title Priority Date Filing Date
IL193322A IL193322A (en) 2006-02-21 2008-08-07 Derivatives of 4– (3 – benzoylaminophenyl) –7,6 – domethoxy – 2– methylaminoquinazoline

Country Status (18)

Country Link
JP (1) JP4778550B2 (el)
KR (1) KR101278852B1 (el)
AT (1) ATE517875T1 (el)
BR (1) BRPI0708098B8 (el)
CY (1) CY1112554T1 (el)
DK (1) DK1992622T3 (el)
ES (1) ES2368089T3 (el)
HK (1) HK1122025A1 (el)
HR (1) HRP20110604T1 (el)
IL (1) IL193322A (el)
JO (1) JO2726B1 (el)
MY (1) MY146275A (el)
NZ (1) NZ569936A (el)
PT (1) PT1992622E (el)
RS (1) RS51969B (el)
RU (1) RU2431632C2 (el)
SI (1) SI1992622T1 (el)
TW (1) TWI404709B (el)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2678477A1 (en) 2007-02-16 2008-08-21 Eisai R&D Management Co., Ltd. Crystal, amorphous form and salt of methyl n-[3-(6,7-dimethoxy-2-methylaminoquinazolin-4-yl)phenyl]terephthalamic acid
ATE538102T1 (de) 2007-08-17 2012-01-15 Eisai R&D Man Co Ltd Verfahren zur herstellung eines chinazolinderivats
EP2202229B1 (en) 2007-08-17 2012-03-14 Eisai R&D Management Co., Ltd. Novel preparation for external use

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR015966A1 (es) * 1997-10-17 2001-05-30 Smithkline Beecham Corp Uso de un compuesto inhibidor de pde4 para la preparacion de un medicamento util para el tratamiento de prurito
JPH11209350A (ja) 1998-01-26 1999-08-03 Eisai Co Ltd 含窒素複素環誘導体およびその医薬

Also Published As

Publication number Publication date
MY146275A (en) 2012-07-31
RU2008137654A (ru) 2010-03-27
DK1992622T3 (da) 2011-09-05
SI1992622T1 (sl) 2011-11-30
JPWO2007097317A1 (ja) 2009-07-16
BRPI0708098B8 (pt) 2021-05-25
NZ569936A (en) 2010-07-30
HRP20110604T1 (hr) 2011-09-30
HK1122025A1 (el) 2009-05-08
ES2368089T3 (es) 2011-11-14
JP4778550B2 (ja) 2011-09-21
TW200812980A (en) 2008-03-16
ATE517875T1 (de) 2011-08-15
BRPI0708098B1 (pt) 2019-08-06
KR101278852B1 (ko) 2013-07-01
TWI404709B (zh) 2013-08-11
JO2726B1 (en) 2013-09-15
IL193322A0 (en) 2009-05-04
CY1112554T1 (el) 2016-02-10
RS51969B (en) 2012-02-29
KR20080094811A (ko) 2008-10-24
RU2431632C2 (ru) 2011-10-20
BRPI0708098A2 (pt) 2011-05-17
PT1992622E (pt) 2011-09-19

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