IL169314A0 - Process for the production of 3'-nucleoside prodrugs - Google Patents

Process for the production of 3'-nucleoside prodrugs

Info

Publication number
IL169314A0
IL169314A0 IL169314A IL16931405A IL169314A0 IL 169314 A0 IL169314 A0 IL 169314A0 IL 169314 A IL169314 A IL 169314A IL 16931405 A IL16931405 A IL 16931405A IL 169314 A0 IL169314 A0 IL 169314A0
Authority
IL
Israel
Prior art keywords
production
nucleoside prodrugs
nucleoside
prodrugs
Prior art date
Application number
IL169314A
Other languages
English (en)
Original Assignee
Idenix Cayman Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Idenix Cayman Ltd filed Critical Idenix Cayman Ltd
Publication of IL169314A0 publication Critical patent/IL169314A0/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
IL169314A 2002-12-23 2005-06-21 Process for the production of 3'-nucleoside prodrugs IL169314A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US43615002P 2002-12-23 2002-12-23
PCT/US2003/041603 WO2004058792A1 (en) 2002-12-23 2003-12-23 Process for the production of 3'-nucleoside prodrugs

Publications (1)

Publication Number Publication Date
IL169314A0 true IL169314A0 (en) 2007-07-04

Family

ID=32682350

Family Applications (1)

Application Number Title Priority Date Filing Date
IL169314A IL169314A0 (en) 2002-12-23 2005-06-21 Process for the production of 3'-nucleoside prodrugs

Country Status (16)

Country Link
US (1) US20040181051A1 (enExample)
EP (1) EP1575971A4 (enExample)
JP (1) JP2006514038A (enExample)
KR (1) KR20050110611A (enExample)
CN (1) CN100335492C (enExample)
AU (1) AU2003300434A1 (enExample)
BR (1) BR0316868A (enExample)
CA (1) CA2511616A1 (enExample)
IL (1) IL169314A0 (enExample)
MX (1) MXPA05006865A (enExample)
NO (1) NO20053557L (enExample)
NZ (1) NZ540913A (enExample)
PL (1) PL377608A1 (enExample)
RU (1) RU2005123395A (enExample)
WO (1) WO2004058792A1 (enExample)
ZA (1) ZA200505040B (enExample)

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PT1576138T (pt) 2002-11-15 2017-05-03 Idenix Pharmaceuticals Llc 2'-metil-nucleósidos em combinação com interferão e mutação de flaviviridae
RU2005121904A (ru) 2002-12-12 2006-01-20 Айденикс (Кайман) Лимитед (Ky) Способ получения 2`-разветвленных нуклеозидов
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CA2637879A1 (en) * 2006-02-14 2007-08-23 Merck & Co., Inc. Nucleoside aryl phosphoramidates for the treatment of rna-dependent rna viral infection
JP2009532411A (ja) 2006-04-04 2009-09-10 エフ．ホフマン−ラ ロシュ アーゲー Ｈｃｖ治療のための３’，５’−ジ−ｏ−アシル化ヌクレオシド
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US8716263B2 (en) 2008-12-23 2014-05-06 Gilead Pharmasset Llc Synthesis of purine nucleosides
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US8551973B2 (en) 2008-12-23 2013-10-08 Gilead Pharmasset Llc Nucleoside analogs
CA2749394A1 (en) 2009-01-09 2010-07-15 University College Of Cardiff Consultants Limited Phosphoramidate derivatives of guanosine nucleoside compounds for treatment of viral infections
WO2011123668A2 (en) 2010-03-31 2011-10-06 Pharmasset, Inc. Stereoselective synthesis of phosphorus containing actives
SG11201901457TA (en) 2016-09-07 2019-03-28 Atea Pharmaceuticals Inc 2'-substituted-n6-substituted purine nucleotides for rna virus treatment
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Also Published As

Publication number Publication date
WO2004058792A1 (en) 2004-07-15
PL377608A1 (pl) 2006-02-06
NZ540913A (en) 2008-02-29
KR20050110611A (ko) 2005-11-23
BR0316868A (pt) 2005-10-25
CN100335492C (zh) 2007-09-05
CN1751058A (zh) 2006-03-22
NO20053557L (no) 2005-09-08
ZA200505040B (en) 2006-04-26
AU2003300434A1 (en) 2004-07-22
MXPA05006865A (es) 2005-12-12
EP1575971A1 (en) 2005-09-21
CA2511616A1 (en) 2004-07-15
US20040181051A1 (en) 2004-09-16
RU2005123395A (ru) 2006-01-27
EP1575971A4 (en) 2008-03-05
JP2006514038A (ja) 2006-04-27

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