IL162596A0 - 1-Alkyl-1-azoniabicyclo Ä2.2.2Ü octane carbamate derivatives and their use as muscarinic receptor ntagonists - Google Patents

1-Alkyl-1-azoniabicyclo Ä2.2.2Ü octane carbamate derivatives and their use as muscarinic receptor ntagonists

Info

Publication number
IL162596A0
IL162596A0 IL16259602A IL16259602A IL162596A0 IL 162596 A0 IL162596 A0 IL 162596A0 IL 16259602 A IL16259602 A IL 16259602A IL 16259602 A IL16259602 A IL 16259602A IL 162596 A0 IL162596 A0 IL 162596A0
Authority
IL
Israel
Prior art keywords
ntagonists
azoniabicyclo
octane
alkyl
muscarinic receptor
Prior art date
Application number
IL16259602A
Other languages
English (en)
Original Assignee
S A L V A T Lab Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by S A L V A T Lab Sa filed Critical S A L V A T Lab Sa
Publication of IL162596A0 publication Critical patent/IL162596A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/02—Nasal agents, e.g. decongestants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/10—Drugs for disorders of the urinary system of the bladder
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/12—Antidiuretics, e.g. drugs for diabetes insipidus
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • C07D453/04—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems having a quinolyl-4, a substituted quinolyl-4 or a alkylenedioxy-quinolyl-4 radical linked through only one carbon atom, attached in position 2, e.g. quinine

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pulmonology (AREA)
  • Diabetes (AREA)
  • Epidemiology (AREA)
  • Urology & Nephrology (AREA)
  • Hematology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
IL16259602A 2001-12-20 2002-12-18 1-Alkyl-1-azoniabicyclo Ä2.2.2Ü octane carbamate derivatives and their use as muscarinic receptor ntagonists IL162596A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
ES200200043 2001-12-20
PCT/EP2002/014470 WO2003053966A2 (en) 2001-12-20 2002-12-18 1-alkyl-1-azoniabicyclo [2.2.2] octane carbamate derivatives and their use as muscarinic receptor antagonists

Publications (1)

Publication Number Publication Date
IL162596A0 true IL162596A0 (en) 2005-11-20

Family

ID=32480019

Family Applications (1)

Application Number Title Priority Date Filing Date
IL16259602A IL162596A0 (en) 2001-12-20 2002-12-18 1-Alkyl-1-azoniabicyclo Ä2.2.2Ü octane carbamate derivatives and their use as muscarinic receptor ntagonists

Country Status (21)

Country Link
US (1) US7452904B2 (xx)
EP (1) EP1461336B1 (xx)
JP (1) JP4505227B2 (xx)
KR (1) KR100944580B1 (xx)
CN (1) CN1832948B (xx)
BR (1) BR0215348A (xx)
CA (1) CA2470956C (xx)
EA (1) EA006505B1 (xx)
ES (1) ES2425347T3 (xx)
GE (1) GEP20063958B (xx)
HK (1) HK1070057A1 (xx)
HR (1) HRP20040661A2 (xx)
HU (1) HUP0500107A3 (xx)
IL (1) IL162596A0 (xx)
MA (1) MA26385A1 (xx)
MX (1) MXPA04006206A (xx)
NO (1) NO329664B1 (xx)
PL (1) PL211250B1 (xx)
RS (1) RS52522B (xx)
UA (1) UA76571C2 (xx)
WO (1) WO2003053966A2 (xx)

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Also Published As

Publication number Publication date
KR100944580B1 (ko) 2010-02-25
AU2002361158A1 (en) 2003-07-09
KR20040091614A (ko) 2004-10-28
NO329664B1 (no) 2010-11-29
MA26385A1 (fr) 2004-11-01
EA006505B1 (ru) 2005-12-29
EA200400832A1 (ru) 2004-12-30
PL370972A1 (en) 2005-06-13
GEP20063958B (en) 2006-11-10
PL211250B1 (pl) 2012-04-30
CN1832948A (zh) 2006-09-13
WO2003053966A2 (en) 2003-07-03
WO2003053966A3 (en) 2003-11-13
MXPA04006206A (es) 2004-12-06
HUP0500107A3 (en) 2011-05-30
NO20043064L (no) 2004-09-17
US20050043349A1 (en) 2005-02-24
HRP20040661A2 (en) 2005-06-30
JP2005516954A (ja) 2005-06-09
CN1832948B (zh) 2011-06-15
CA2470956C (en) 2011-08-02
EP1461336B1 (en) 2013-05-22
ES2425347T3 (es) 2013-10-14
CA2470956A1 (en) 2003-07-03
EP1461336A2 (en) 2004-09-29
RS53904A (xx) 2006-12-15
BR0215348A (pt) 2004-11-16
JP4505227B2 (ja) 2010-07-21
HK1070057A1 (xx) 2005-06-10
HUP0500107A2 (hu) 2005-05-30
WO2003053966A8 (en) 2004-06-24
UA76571C2 (en) 2006-08-15
RS52522B (en) 2013-04-30
US7452904B2 (en) 2008-11-18

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