IL143299A0 - Pharmaceutical composition comprising 5-[[4- [3-methyl-4-oxo-3, 4-dihydro-2-quinazolinyl] methoxy] phenyl-methyl] thiadiazolidine-2, 4-dione and the process for its preparation - Google Patents

Pharmaceutical composition comprising 5-[[4- [3-methyl-4-oxo-3, 4-dihydro-2-quinazolinyl] methoxy] phenyl-methyl] thiadiazolidine-2, 4-dione and the process for its preparation

Info

Publication number
IL143299A0
IL143299A0 IL14329999A IL14329999A IL143299A0 IL 143299 A0 IL143299 A0 IL 143299A0 IL 14329999 A IL14329999 A IL 14329999A IL 14329999 A IL14329999 A IL 14329999A IL 143299 A0 IL143299 A0 IL 143299A0
Authority
IL
Israel
Prior art keywords
methyl
thiadiazolidine
quinazolinyl
dione
dihydro
Prior art date
Application number
IL14329999A
Other languages
English (en)
Original Assignee
Novo Nordisk As
Reddy Research Foundation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novo Nordisk As, Reddy Research Foundation filed Critical Novo Nordisk As
Publication of IL143299A0 publication Critical patent/IL143299A0/xx

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/427—Thiazoles not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
    • A61P5/50—Drugs for disorders of the endocrine system of the pancreatic hormones for increasing or potentiating the activity of insulin

Landscapes

  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Diabetes (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Endocrinology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
IL14329999A 1998-12-01 1999-11-29 Pharmaceutical composition comprising 5-[[4- [3-methyl-4-oxo-3, 4-dihydro-2-quinazolinyl] methoxy] phenyl-methyl] thiadiazolidine-2, 4-dione and the process for its preparation IL143299A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DKPA199801580 1998-12-01
PCT/DK1999/000663 WO2000032191A1 (en) 1998-12-01 1999-11-29 New pharmaceutical composition and the process for its preparation

Publications (1)

Publication Number Publication Date
IL143299A0 true IL143299A0 (en) 2002-04-21

Family

ID=8106261

Family Applications (3)

Application Number Title Priority Date Filing Date
IL14329999A IL143299A0 (en) 1998-12-01 1999-11-29 Pharmaceutical composition comprising 5-[[4- [3-methyl-4-oxo-3, 4-dihydro-2-quinazolinyl] methoxy] phenyl-methyl] thiadiazolidine-2, 4-dione and the process for its preparation
IL143299A IL143299A (en) 1998-12-01 2001-05-22 Pharmaceutical preparation containing 5 - [[- [3-methyl - 4 - oxo - 3,4 - dehydro - quinazolinyl] methoxy] phenyl-methyl] thiadiazolidine - 2,4 - deion and process for its preparation
IL179865A IL179865A (en) 1998-12-01 2006-12-05 Pharmaceutical composition comprising 5 - [[4-[3 - methyl- 4- oxo - 3,4 - dihydro - 2 - quinazolinyl]methoxy] phenyl-methyl]thiadiazolidine-2,4- dione in the form of a tablet, a powder or a capsule and process for its preparation

Family Applications After (2)

Application Number Title Priority Date Filing Date
IL143299A IL143299A (en) 1998-12-01 2001-05-22 Pharmaceutical preparation containing 5 - [[- [3-methyl - 4 - oxo - 3,4 - dehydro - quinazolinyl] methoxy] phenyl-methyl] thiadiazolidine - 2,4 - deion and process for its preparation
IL179865A IL179865A (en) 1998-12-01 2006-12-05 Pharmaceutical composition comprising 5 - [[4-[3 - methyl- 4- oxo - 3,4 - dihydro - 2 - quinazolinyl]methoxy] phenyl-methyl]thiadiazolidine-2,4- dione in the form of a tablet, a powder or a capsule and process for its preparation

Country Status (21)

Country Link
US (1) US7439248B1 (xx)
EP (1) EP1135127B1 (xx)
JP (2) JP5524435B2 (xx)
KR (1) KR100690311B1 (xx)
CN (1) CN1158075C (xx)
AT (1) ATE316376T1 (xx)
AU (1) AU776299B2 (xx)
BR (1) BR9915835A (xx)
CA (1) CA2352430C (xx)
CZ (1) CZ300543B6 (xx)
DE (1) DE69929635T2 (xx)
ES (1) ES2257886T3 (xx)
HU (1) HUP0104544A3 (xx)
IL (3) IL143299A0 (xx)
NO (1) NO329909B1 (xx)
PL (1) PL197077B1 (xx)
RU (1) RU2233659C2 (xx)
TW (1) TWI235657B (xx)
UA (1) UA75569C2 (xx)
WO (1) WO2000032191A1 (xx)
ZA (1) ZA200104261B (xx)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1158075C (zh) * 1998-12-01 2004-07-21 诺沃挪第克公司 新药物组合物及其制备方法
US20010047032A1 (en) * 1999-12-30 2001-11-29 Castillo Gerardo M. Polyhydroxylated aromatic compounds for the treatment of amyloidosis and alpha-synuclein fibril diseases
AU2001260083A1 (en) * 2000-05-26 2001-12-03 Dr. Reddy's Research Foundation New pharmaceutical composition and the process for its preparation
WO2001091751A1 (en) * 2000-05-30 2001-12-06 Novo Nordisk A/S New pharmaceutical composition and the process for its preparation
US20050118202A1 (en) * 2001-12-19 2005-06-02 Akio Yamashita Solid compositions containing compounds unstable to oxygen and method for stabilization thereof
WO2006002255A2 (en) * 2004-06-23 2006-01-05 Dr. Reddy's Laboratories Ltd. A pharmaceutical formulation of balaglitazone
CL2008000596A1 (es) * 2007-03-01 2008-09-05 Glaxo Group Ltd Forma de dosificacion que comprende 1-(6-[(3-ciclobutil-2,3,4,5-tetrahidro-1h-3-benzazepin-7-il)oxi]-3-piridinil)-2-pirrolidinona, un estabilizador, un excipiente; procedimiento de preparacion; y su uso para tratar enfermedades neurologicas.

Family Cites Families (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4280997A (en) * 1978-12-08 1981-07-28 Johannes Van Leverink Extrusion process for the preparation of anhydrous stable lactose
DE3433239A1 (de) * 1984-09-11 1986-03-20 Bayer Ag, 5090 Leverkusen Feste arzneizubereitung enthaltend nitrendipin und verfahren zu ihrer herstellung
CA2019324C (en) * 1989-07-10 1996-08-20 Robert L. Jerzewski Fosinopril tablet formulations
IT1238072B (it) * 1990-01-19 1993-07-03 Sclavo Spa Composizioni farmaceutiche e forme di dosaggio per la somministrazione orale di calcitonina
AU665944B2 (en) * 1991-04-04 1996-01-25 Procter & Gamble Company, The Chewable antacid compositions
CZ227093A3 (en) * 1991-04-29 1994-03-16 Merck & Co Inc Mixture suitable for the preparation of tablets by direct moulding
TW268952B (xx) * 1993-02-26 1996-01-21 Takeda Pharm Industry Co Ltd
DE69431662T2 (de) * 1993-09-03 2003-09-18 Smithkline Beecham Corp Stabilisierte tablettenformulierung
US5532256A (en) 1994-05-18 1996-07-02 American Home Products Corporation New azolidinediones and thiadiazolidinediones as antihyperglycemic agents
ES2079327B1 (es) * 1994-12-13 1996-08-01 Lilly Sa Formulaciones farmaceuticas de cefaclor.
ATE199495T1 (de) * 1994-12-14 2001-03-15 Enbalt Trading Ltd Pharmazeutische zubereitung zur direktverpressung
US6395303B1 (en) * 1996-06-10 2002-05-28 Edward Mendell Co., Inc. Process for preparing a directly compressible solid dosage form containing microcrystalline cellulose
JPH09249561A (ja) * 1996-03-15 1997-09-22 Teikoku Chem Ind Corp Ltd 医薬組成物
HU222109B1 (hu) * 1996-09-10 2003-04-28 EGIS Gyógyszergyár Rt. Captopriltartalmú tabletták és eljárás ezek előállítására
HUP0301101A3 (en) * 1996-12-31 2009-03-30 Reddy S Res Foundation Novel heterocyclic compounds process for their preparation and pharmaceutical compositions containing them and their use in the treatment of diabetes and related diseases
DE69824756T2 (de) 1997-12-02 2005-07-14 Dr. Reddy's Laboratories Ltd. Substituierte thiazolidinedione und oxazolidinedione mit antidiabetischen,hypolipidämischen und antihypertensiven eigenschaften
EP0945134A1 (de) * 1998-03-27 1999-09-29 Boehringer Ingelheim Pharma KG Neue galenische Zubereitungsformen von Meloxicam zur oralen Applikation
CN1158075C (zh) * 1998-12-01 2004-07-21 诺沃挪第克公司 新药物组合物及其制备方法
AU2001260083A1 (en) * 2000-05-26 2001-12-03 Dr. Reddy's Research Foundation New pharmaceutical composition and the process for its preparation
WO2006002255A2 (en) 2004-06-23 2006-01-05 Dr. Reddy's Laboratories Ltd. A pharmaceutical formulation of balaglitazone

Also Published As

Publication number Publication date
EP1135127B1 (en) 2006-01-25
NO20012673D0 (no) 2001-05-31
KR20010099827A (ko) 2001-11-09
TWI235657B (en) 2005-07-11
JP5524435B2 (ja) 2014-06-18
CZ300543B6 (cs) 2009-06-10
NO329909B1 (no) 2011-01-24
PL348601A1 (en) 2002-06-03
JP2012144560A (ja) 2012-08-02
HUP0104544A3 (en) 2003-12-29
JP2002531404A (ja) 2002-09-24
IL179865A0 (en) 2007-05-15
ES2257886T3 (es) 2006-08-01
ATE316376T1 (de) 2006-02-15
AU1376200A (en) 2000-06-19
CA2352430A1 (en) 2000-06-08
KR100690311B1 (ko) 2007-03-09
IL143299A (en) 2006-12-31
BR9915835A (pt) 2001-08-21
CZ20011832A3 (cs) 2001-10-17
UA75569C2 (en) 2006-05-15
RU2233659C2 (ru) 2004-08-10
NO20012673L (no) 2001-05-31
IL179865A (en) 2009-12-24
EP1135127A1 (en) 2001-09-26
CN1158075C (zh) 2004-07-21
DE69929635D1 (de) 2006-04-13
ZA200104261B (en) 2002-05-24
CN1356901A (zh) 2002-07-03
WO2000032191A1 (en) 2000-06-08
US7439248B1 (en) 2008-10-21
AU776299B2 (en) 2004-09-02
DE69929635T2 (de) 2006-09-21
PL197077B1 (pl) 2008-02-29
HUP0104544A2 (en) 2002-08-28
CA2352430C (en) 2008-11-18

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Legal Events

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FF Patent granted
KB Patent renewed