IL121969A - 10,13,15-trioxatricyclo¬9.2.1.1.9.6¾-pentadecanone derivatives their preparation and pharmaceutical compositions containing these compounds - Google Patents
10,13,15-trioxatricyclo¬9.2.1.1.9.6¾-pentadecanone derivatives their preparation and pharmaceutical compositions containing these compoundsInfo
- Publication number
- IL121969A IL121969A IL12196997A IL12196997A IL121969A IL 121969 A IL121969 A IL 121969A IL 12196997 A IL12196997 A IL 12196997A IL 12196997 A IL12196997 A IL 12196997A IL 121969 A IL121969 A IL 121969A
- Authority
- IL
- Israel
- Prior art keywords
- trioxatricyclo
- pentadecanone
- derivatives
- compounds
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/06—Anti-spasmodics, e.g. drugs for colics, esophagic dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H1/00—Processes for the preparation of sugar derivatives
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Molecular Biology (AREA)
- Biochemistry (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Genetics & Genomics (AREA)
- Public Health (AREA)
- Biotechnology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19644195A DE19644195A1 (de) | 1996-10-24 | 1996-10-24 | 10,13,15-Trioxatricyclo[9.2.1.1.·9·.·6·]-pentadecanon-Derivate, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel |
Publications (2)
Publication Number | Publication Date |
---|---|
IL121969A0 IL121969A0 (en) | 1998-03-10 |
IL121969A true IL121969A (en) | 2000-06-29 |
Family
ID=7809858
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IL12196997A IL121969A (en) | 1996-10-24 | 1997-10-14 | 10,13,15-trioxatricyclo¬9.2.1.1.9.6¾-pentadecanone derivatives their preparation and pharmaceutical compositions containing these compounds |
Country Status (27)
Country | Link |
---|---|
US (1) | US5912235A (ja) |
EP (1) | EP0838469B1 (ja) |
JP (1) | JP4175682B2 (ja) |
KR (1) | KR100466495B1 (ja) |
CN (1) | CN1093133C (ja) |
AR (1) | AR009809A1 (ja) |
AT (1) | ATE211745T1 (ja) |
AU (1) | AU726092B2 (ja) |
BR (2) | BR9705143A (ja) |
CA (1) | CA2219311C (ja) |
CZ (1) | CZ291768B6 (ja) |
DE (2) | DE19644195A1 (ja) |
DK (1) | DK0838469T3 (ja) |
DZ (1) | DZ2322A1 (ja) |
ES (1) | ES2170318T3 (ja) |
HK (1) | HK1010885A1 (ja) |
HU (1) | HU222540B1 (ja) |
IL (1) | IL121969A (ja) |
MX (1) | MX9707974A (ja) |
NO (1) | NO308362B1 (ja) |
NZ (1) | NZ328979A (ja) |
PL (1) | PL184693B1 (ja) |
PT (1) | PT838469E (ja) |
RU (1) | RU2181727C2 (ja) |
SK (1) | SK283114B6 (ja) |
UA (1) | UA44310C2 (ja) |
ZA (1) | ZA979059B (ja) |
Families Citing this family (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1998023629A1 (fr) * | 1996-11-26 | 1998-06-04 | Chugai Seiyaku Kabushiki Kaisha | Composes de macrolides comportant une chaine a 13 elements, medicament les contenant et leur procede de preparation |
PT1489090E (pt) * | 2000-08-17 | 2006-05-31 | Kitasato Inst | Novos derivados de pseudoeritromicina |
JP2003007917A (ja) * | 2001-06-19 | 2003-01-10 | Sanyo Electric Co Ltd | 回路装置の製造方法 |
US6986882B2 (en) * | 2002-01-17 | 2006-01-17 | Astrazeneca Ab | Therapy for functional dyspepsia |
US7521420B2 (en) | 2003-06-18 | 2009-04-21 | Tranzyme Pharma, Inc. | Macrocyclic antagonists of the motilin receptor |
GB0611907D0 (en) | 2006-06-15 | 2006-07-26 | Glaxo Group Ltd | Compounds |
JP2009501199A (ja) | 2005-07-12 | 2009-01-15 | グラクソ グループ リミテッド | Gpr38アゴニストとしてのピペラジンヘテロアリール誘導体 |
MX2008001211A (es) | 2005-07-26 | 2008-03-24 | Glaxo Group Ltd | Derivados de bencilpiperazina y su uso medico. |
CA2632779A1 (en) * | 2005-12-08 | 2007-06-14 | Pfizer Inc. | Method for demethylating the 3'-dimethylamino group of erythromycin compounds |
DE602007006019D1 (de) | 2006-06-28 | 2010-06-02 | Glaxo Group Ltd | Für die behandlung von durch den gpr38-rezeptor vermittelten krankheiten geeignete piperazinylderivate |
JP5684474B2 (ja) | 2006-09-11 | 2015-03-11 | オセラ セラピューティクス, インコーポレイテッド | 胃腸の運動障害疾患の治療のためのモチリン受容体の大環状アンタゴニスト |
RU2533116C2 (ru) | 2009-02-27 | 2014-11-20 | Раквалиа Фарма Инк. | Оксииндольные производные, обладающие агонистической активностью в отношении мотилинового рецептора |
WO2014156339A1 (ja) * | 2013-03-25 | 2014-10-02 | ゼリア新薬工業株式会社 | 食後期の胃運動亢進剤 |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3725385A (en) * | 1970-11-02 | 1973-04-03 | Abbott Lab | Process for the demethylation of 3-amino macrolides |
US5106961A (en) * | 1987-05-26 | 1992-04-21 | Eli Lilly And Company | Erythromycin ring-contracted derivatives |
US4920102A (en) * | 1988-04-18 | 1990-04-24 | Eli Lilly And Company | Method for treating gastrointestinal disorders |
DE4200145A1 (de) * | 1992-01-07 | 1993-07-08 | Kali Chemie Pharma Gmbh | 7,10-epoxy-oxacyclododecan-derivate, verfahren und zwischenprodukte zu ihrer herstellung und diese verbindungen enthaltende arzneimittel |
-
1996
- 1996-10-24 DE DE19644195A patent/DE19644195A1/de not_active Withdrawn
-
1997
- 1997-09-23 AR ARP970104375A patent/AR009809A1/es active IP Right Grant
- 1997-09-29 DZ DZ970172A patent/DZ2322A1/xx active
- 1997-10-01 CZ CZ19973106A patent/CZ291768B6/cs not_active IP Right Cessation
- 1997-10-07 KR KR1019970051470A patent/KR100466495B1/ko not_active IP Right Cessation
- 1997-10-09 ZA ZA9709059A patent/ZA979059B/xx unknown
- 1997-10-14 IL IL12196997A patent/IL121969A/xx not_active IP Right Cessation
- 1997-10-16 MX MX9707974A patent/MX9707974A/es not_active IP Right Cessation
- 1997-10-17 AT AT97118000T patent/ATE211745T1/de not_active IP Right Cessation
- 1997-10-17 NZ NZ328979A patent/NZ328979A/xx unknown
- 1997-10-17 SK SK1419-97A patent/SK283114B6/sk not_active IP Right Cessation
- 1997-10-17 PT PT97118000T patent/PT838469E/pt unknown
- 1997-10-17 ES ES97118000T patent/ES2170318T3/es not_active Expired - Lifetime
- 1997-10-17 EP EP97118000A patent/EP0838469B1/de not_active Expired - Lifetime
- 1997-10-17 DE DE59705964T patent/DE59705964D1/de not_active Expired - Fee Related
- 1997-10-17 HU HU9701660A patent/HU222540B1/hu not_active IP Right Cessation
- 1997-10-17 DK DK97118000T patent/DK0838469T3/da active
- 1997-10-21 US US08/954,891 patent/US5912235A/en not_active Expired - Lifetime
- 1997-10-22 JP JP28986197A patent/JP4175682B2/ja not_active Expired - Fee Related
- 1997-10-22 AU AU42788/97A patent/AU726092B2/en not_active Ceased
- 1997-10-22 CN CN97121157A patent/CN1093133C/zh not_active Expired - Fee Related
- 1997-10-23 RU RU97117347/04A patent/RU2181727C2/ru not_active IP Right Cessation
- 1997-10-23 PL PL97322802A patent/PL184693B1/pl not_active IP Right Cessation
- 1997-10-23 UA UA97105178A patent/UA44310C2/uk unknown
- 1997-10-24 CA CA002219311A patent/CA2219311C/en not_active Expired - Fee Related
- 1997-10-24 BR BR9705143-8A patent/BR9705143A/pt active Search and Examination
- 1997-10-24 BR BR9705157-8A patent/BR9705157A/pt not_active Application Discontinuation
- 1997-10-24 NO NO974934A patent/NO308362B1/no not_active IP Right Cessation
-
1998
- 1998-11-10 HK HK98111873A patent/HK1010885A1/xx not_active IP Right Cessation
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FF | Patent granted | ||
KB | Patent renewed | ||
KB | Patent renewed | ||
MM9K | Patent not in force due to non-payment of renewal fees |