IL109144A - Glycoprotein IIB/IIIA inhibiting 4-pyridylamino heterocyclic derivatives process for their preparation and pharmaceutical compositions containing them - Google Patents

Glycoprotein IIB/IIIA inhibiting 4-pyridylamino heterocyclic derivatives process for their preparation and pharmaceutical compositions containing them

Info

Publication number
IL109144A
IL109144A IL10914494A IL10914494A IL109144A IL 109144 A IL109144 A IL 109144A IL 10914494 A IL10914494 A IL 10914494A IL 10914494 A IL10914494 A IL 10914494A IL 109144 A IL109144 A IL 109144A
Authority
IL
Israel
Prior art keywords
iiia
pyridylamino
inhibiting
preparation
pharmaceutical compositions
Prior art date
Application number
IL10914494A
Other languages
English (en)
Other versions
IL109144A0 (en
Original Assignee
Zeneca Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB939306453A external-priority patent/GB9306453D0/en
Priority claimed from GB939325605A external-priority patent/GB9325605D0/en
Application filed by Zeneca Ltd filed Critical Zeneca Ltd
Publication of IL109144A0 publication Critical patent/IL109144A0/xx
Publication of IL109144A publication Critical patent/IL109144A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/74—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Emulsifying, Dispersing, Foam-Producing Or Wetting Agents (AREA)
  • Electrochromic Elements, Electrophoresis, Or Variable Reflection Or Absorption Elements (AREA)
  • Electroluminescent Light Sources (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyridine Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
IL10914494A 1993-03-29 1994-03-28 Glycoprotein IIB/IIIA inhibiting 4-pyridylamino heterocyclic derivatives process for their preparation and pharmaceutical compositions containing them IL109144A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB939306453A GB9306453D0 (en) 1993-03-29 1993-03-29 Heterocyclic derivatives
GB939325605A GB9325605D0 (en) 1993-12-15 1993-12-15 Heterocyclic derivatives

Publications (2)

Publication Number Publication Date
IL109144A0 IL109144A0 (en) 1994-06-24
IL109144A true IL109144A (en) 2000-02-29

Family

ID=26302668

Family Applications (1)

Application Number Title Priority Date Filing Date
IL10914494A IL109144A (en) 1993-03-29 1994-03-28 Glycoprotein IIB/IIIA inhibiting 4-pyridylamino heterocyclic derivatives process for their preparation and pharmaceutical compositions containing them

Country Status (26)

Country Link
US (1) US5556977A (ref)
EP (2) EP0825184B1 (ref)
JP (1) JPH08508291A (ref)
KR (1) KR100231089B1 (ref)
CN (1) CN1120334A (ref)
AT (2) ATE202345T1 (ref)
AU (1) AU692438B2 (ref)
BR (1) BR9406613A (ref)
CA (1) CA2156070A1 (ref)
CZ (1) CZ250995A3 (ref)
DE (2) DE69411900T2 (ref)
DK (2) DK0691959T3 (ref)
ES (2) ES2119184T3 (ref)
FI (1) FI954616A7 (ref)
GB (1) GB9406143D0 (ref)
GR (2) GR3027751T3 (ref)
HU (2) HUT72088A (ref)
IL (1) IL109144A (ref)
NO (1) NO305244B1 (ref)
NZ (1) NZ262941A (ref)
PL (1) PL310889A1 (ref)
PT (1) PT825184E (ref)
SK (1) SK120895A3 (ref)
TW (1) TW276254B (ref)
WO (1) WO1994022834A1 (ref)
ZW (1) ZW4294A1 (ref)

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US6232322B1 (en) 1998-05-12 2001-05-15 American Home Products Corporation Biphenyl oxo-acetic acids useful in the treatment of insulin resistance and hyperglycemia
US6110963A (en) * 1998-05-12 2000-08-29 American Home Products Corporation Aryl-oxo-acetic acids useful in the treatment of insulin resistance and hyperglycemia
US6699896B1 (en) 1998-05-12 2004-03-02 Wyeth Oxazole-aryl-carboxylic acids useful in the treatment of insulin resistance and hyperglycemia
JP2002521444A (ja) 1998-07-31 2002-07-16 イーライ・リリー・アンド・カンパニー 複素環スルホンアミド誘導体
GB9902989D0 (en) 1999-02-11 1999-03-31 Zeneca Ltd Heterocyclic derivatives
WO2000063161A1 (en) * 1999-04-19 2000-10-26 Coelacanth Corporation Ppar-(gamma) agonists as agents for the treatment of type ii diabetes
US6310081B1 (en) 1999-05-10 2001-10-30 American Home Products Corporation Biphenyl sulfonyl aryl carboxylic acids useful in the treatment of insulin resistance and hyperglycemia
DE60144284D1 (de) 2000-11-01 2011-05-05 Millennium Pharm Inc Stickstoffhaltige heterozyklische verbindungen und verfahren zu deren herstellung
DE202011000090U1 (de) 2011-01-14 2011-04-21 E-LEAD ELECTRONIC CO., LTD., Shengang Shiang Fahrzeug-Audiosystem mit auswechselbarem Plug-In-Computer
EP3684767B1 (en) 2017-09-22 2024-04-24 Jubilant Epipad LLC Heterocyclic compounds as pad inhibitors
WO2019077631A1 (en) 2017-10-18 2019-04-25 Jubilant Biosys Limited IMIDAZO-PYRIDINE COMPOUNDS FOR USE AS PAD INHIBITORS
BR112020008851A2 (pt) 2017-11-06 2020-10-20 Jubilant Prodel LLC composto da fórmula i, processo de preparação de compostos da fórmula i, composição farmacêutica, método para o tratamento e/ou prevenção de várias doenças, uso, método para o tratamento de câncer, método de tratamento de câncer e método para o tratamento e/ou prevenção de câncer e doenças infecciosas
SG11202004537UA (en) 2017-11-24 2020-06-29 Jubilant Episcribe Llc Heterocyclic compounds as prmt5 inhibitors
BR112020018610A2 (pt) 2018-03-13 2020-12-29 Jubilant Prodel LLC Compostos de fórmula i, fórmula ii, fórmula iii, fórmula iv, fórmula v, fórmula vi, ou seus polimorfos, estereoisômeros, tautômeros, profármacos, solvatos e sais farmaceuticamente aceitáveis dos mesmos e uso dos mesmos; processo de preparação; composição farmacêutica; e método para o tratamento e/ou prevenção de várias doenças, que incluem câncer e doenças infecciosas

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Also Published As

Publication number Publication date
ZW4294A1 (en) 1994-12-21
HU211336A9 (en) 1995-11-28
EP0825184B1 (en) 2001-06-20
FI954616A0 (fi) 1995-09-28
GB9406143D0 (en) 1994-05-18
CN1120334A (zh) 1996-04-10
ES2159798T3 (es) 2001-10-16
DE69411900T2 (de) 1998-12-10
PL310889A1 (en) 1996-01-08
EP0691959B1 (en) 1998-07-22
GR3027751T3 (en) 1998-11-30
FI954616L (fi) 1995-09-28
HUT72088A (en) 1996-03-28
CZ250995A3 (en) 1996-01-17
BR9406613A (pt) 1996-02-06
SK120895A3 (en) 1996-06-05
IL109144A0 (en) 1994-06-24
EP0825184A1 (en) 1998-02-25
WO1994022834A1 (en) 1994-10-13
FI954616A7 (fi) 1995-09-28
NO953837L (no) 1995-09-28
DE69427548D1 (de) 2001-07-26
ATE202345T1 (de) 2001-07-15
DK0825184T3 (da) 2001-09-10
DK0691959T3 (da) 1999-04-26
AU6288994A (en) 1994-10-24
US5556977A (en) 1996-09-17
NO953837D0 (no) 1995-09-28
JPH08508291A (ja) 1996-09-03
DE69427548T2 (de) 2002-04-18
GR3036640T3 (en) 2001-12-31
NZ262941A (en) 1997-07-27
EP0691959A1 (en) 1996-01-17
ES2119184T3 (es) 1998-10-01
PT825184E (pt) 2001-11-30
KR100231089B1 (ko) 1999-11-15
ATE168678T1 (de) 1998-08-15
AU692438B2 (en) 1998-06-11
NO305244B1 (no) 1999-04-26
TW276254B (ref) 1996-05-21
HU9502290D0 (en) 1995-10-30
CA2156070A1 (en) 1994-10-13
DE69411900D1 (de) 1998-08-27

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Legal Events

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