ID28343A - Kaprolaktam tersubstitusi tertentu, komposisi farmasi yang mengandungnya dan penggunaannya dalam pengobatan tumor - Google Patents

Kaprolaktam tersubstitusi tertentu, komposisi farmasi yang mengandungnya dan penggunaannya dalam pengobatan tumor

Info

Publication number
ID28343A
ID28343A IDW00200100966A ID20010966A ID28343A ID 28343 A ID28343 A ID 28343A ID W00200100966 A IDW00200100966 A ID W00200100966A ID 20010966 A ID20010966 A ID 20010966A ID 28343 A ID28343 A ID 28343A
Authority
ID
Indonesia
Prior art keywords
capacolakam
certained
substituted
tumor treatment
pharmacy composition
Prior art date
Application number
IDW00200100966A
Other languages
English (en)
Inventor
Frederick R Kinder
Kenneth W Bair
Christopher T Jagoe
Richard W Versace
Sompong Wattanasin
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of ID28343A publication Critical patent/ID28343A/id

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D223/00Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
    • C07D223/02Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D223/06Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom not condensed with other rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D223/08Oxygen atoms
    • C07D223/10Oxygen atoms attached in position 2
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
IDW00200100966A 1998-11-17 1999-11-15 Kaprolaktam tersubstitusi tertentu, komposisi farmasi yang mengandungnya dan penggunaannya dalam pengobatan tumor ID28343A (id)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US19335498A 1998-11-17 1998-11-17

Publications (1)

Publication Number Publication Date
ID28343A true ID28343A (id) 2001-05-17

Family

ID=22713307

Family Applications (1)

Application Number Title Priority Date Filing Date
IDW00200100966A ID28343A (id) 1998-11-17 1999-11-15 Kaprolaktam tersubstitusi tertentu, komposisi farmasi yang mengandungnya dan penggunaannya dalam pengobatan tumor

Country Status (25)

Country Link
EP (1) EP1131297B1 (id)
JP (1) JP3550545B2 (id)
KR (1) KR20010080461A (id)
CN (1) CN1187333C (id)
AR (1) AR023914A1 (id)
AT (1) ATE264309T1 (id)
AU (1) AU748016B2 (id)
BR (1) BR9915436A (id)
CA (1) CA2347773C (id)
CO (1) CO5140099A1 (id)
CZ (1) CZ20011707A3 (id)
DE (1) DE69916488T2 (id)
ES (1) ES2221463T3 (id)
HU (1) HUP0104224A3 (id)
ID (1) ID28343A (id)
IL (1) IL142701A0 (id)
NO (1) NO20012428L (id)
PE (1) PE20001241A1 (id)
PL (1) PL347633A1 (id)
PT (1) PT1131297E (id)
SK (1) SK6692001A3 (id)
TR (1) TR200101366T2 (id)
UY (2) UY25807A1 (id)
WO (1) WO2000029382A1 (id)
ZA (1) ZA200103419B (id)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1191237C (zh) * 2000-05-11 2005-03-02 诺瓦提斯公司 取代的己内酰胺碳酸酯与醚和它们作为抗肿瘤剂的用途
WO2002072555A1 (en) * 2001-03-12 2002-09-19 Novartis Ag Process for preparing certain substituted caprolactams
CN1856486A (zh) 2003-07-25 2006-11-01 诺瓦提斯公司 取代的内酰胺和它们作为抗癌剂的用途
US7153846B2 (en) 2003-10-24 2006-12-26 Sanofi-Aventis Deutschland Gmbh Bengamide derivatives, process for preparing them, and their use
DE10349669B3 (de) * 2003-10-24 2005-05-25 Aventis Pharma Deutschland Gmbh Bengamide-Derivate, Verfahren zu ihrer Herstellung und ihre Verwendung
FR2878528B1 (fr) * 2004-11-29 2008-05-16 Aventis Pharma Sa 2-alcoxy-3,4,5-trihydroxy-alkylamides, leur preparation, compositions les contenant et utilisation
FR2878525B1 (fr) * 2004-11-29 2007-02-23 Aventis Pharma Sa Bengamides possedant un cycle caprolactame substitue, procede de preparation, compositions les contenant et utilisation
FR2901556A1 (fr) * 2006-05-24 2007-11-30 Sanofi Aventis Sa Derives de 2-alcoxy-3,4,5-trihydroxy-alkylamide, leur preparation, compositions les contenant et utilisation
FR2901555A1 (fr) 2006-05-24 2007-11-30 Sanofi Aventis Sa 2-alcoxy-3,4,5-trihydroxy-alkylamide-benzothiazepine, leur preparation, compositions les contenant et utilisation
FR2901554B1 (fr) 2006-05-24 2011-04-01 Sanofi Aventis 2-alcoxy-3,4,5-trihydroxy-alkylamide-benzazepine, leur preparation, compositions les contenant et utilisation
US20130090342A1 (en) 2010-06-17 2013-04-11 Novartis Ag Biphenyl substituted 1,3-dihydro-benzoimidazol-2-ylideneamine derivatives
JP2013532149A (ja) 2010-06-17 2013-08-15 ノバルティス アーゲー ピペリジニル置換1,3−ジヒドロ−ベンゾイミダゾール−2−イリデンアミン誘導体

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9411841D0 (en) * 1994-06-14 1994-08-03 Pharma Mar Sa New antitumoral compounds from jaspis sponge

Also Published As

Publication number Publication date
EP1131297B1 (en) 2004-04-14
CN1187333C (zh) 2005-02-02
JP2002529536A (ja) 2002-09-10
SK6692001A3 (en) 2001-10-08
DE69916488D1 (de) 2004-05-19
AU748016B2 (en) 2002-05-30
WO2000029382A1 (en) 2000-05-25
CA2347773A1 (en) 2000-05-25
HUP0104224A2 (hu) 2002-03-28
CN1326445A (zh) 2001-12-12
IL142701A0 (en) 2002-03-10
KR20010080461A (ko) 2001-08-22
NO20012428L (no) 2001-07-17
CO5140099A1 (es) 2002-03-22
UY26036A1 (es) 2001-06-29
BR9915436A (pt) 2001-08-07
ES2221463T3 (es) 2004-12-16
PT1131297E (pt) 2004-08-31
ZA200103419B (en) 2002-06-26
HUP0104224A3 (en) 2002-04-29
PL347633A1 (en) 2002-04-22
TR200101366T2 (tr) 2001-10-22
CZ20011707A3 (cs) 2001-08-15
CA2347773C (en) 2009-03-10
NO20012428D0 (no) 2001-05-16
JP3550545B2 (ja) 2004-08-04
AR023914A1 (es) 2002-09-04
ATE264309T1 (de) 2004-04-15
PE20001241A1 (es) 2000-11-24
UY25807A1 (es) 2001-08-27
DE69916488T2 (de) 2005-03-24
EP1131297A1 (en) 2001-09-12
AU1506000A (en) 2000-06-05

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