HUT77318A - 1-Acil-4-/(alifás amino)-piperidin/-származékok, e vegyületeket tartalmazó gyógyszerkészítmények, eljárás előállításukra és alkalmazásuk - Google Patents

1-Acil-4-/(alifás amino)-piperidin/-származékok, e vegyületeket tartalmazó gyógyszerkészítmények, eljárás előállításukra és alkalmazásuk

Info

Publication number
HUT77318A
HUT77318A HU9701800A HU9701800A HUT77318A HU T77318 A HUT77318 A HU T77318A HU 9701800 A HU9701800 A HU 9701800A HU 9701800 A HU9701800 A HU 9701800A HU T77318 A HUT77318 A HU T77318A
Authority
HU
Hungary
Prior art keywords
alkyl
amino
substituted
alkylene
lower alkyl
Prior art date
Application number
HU9701800A
Other languages
English (en)
Inventor
Silvio Ofner
Siem Jacob Veenstra
Original Assignee
Novartis Ag.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag. filed Critical Novartis Ag.
Publication of HUT77318A publication Critical patent/HUT77318A/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/56—Nitrogen atoms
    • C07D211/58—Nitrogen atoms attached in position 4
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Plural Heterocyclic Compounds (AREA)
HU9701800A 1994-09-30 1995-09-19 1-Acil-4-/(alifás amino)-piperidin/-származékok, e vegyületeket tartalmazó gyógyszerkészítmények, eljárás előállításukra és alkalmazásuk HUT77318A (hu)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH296694 1994-09-30

Publications (1)

Publication Number Publication Date
HUT77318A true HUT77318A (hu) 1998-03-30

Family

ID=4245651

Family Applications (1)

Application Number Title Priority Date Filing Date
HU9701800A HUT77318A (hu) 1994-09-30 1995-09-19 1-Acil-4-/(alifás amino)-piperidin/-származékok, e vegyületeket tartalmazó gyógyszerkészítmények, eljárás előállításukra és alkalmazásuk

Country Status (14)

Country Link
US (1) US5935951A (hu)
EP (1) EP0783490B1 (hu)
JP (1) JPH10506399A (hu)
AT (1) ATE212981T1 (hu)
AU (1) AU3607895A (hu)
CA (1) CA2198382A1 (hu)
DE (1) DE69525355T2 (hu)
DK (1) DK0783490T3 (hu)
ES (1) ES2172595T3 (hu)
FI (1) FI971260A (hu)
HU (1) HUT77318A (hu)
NO (1) NO971383L (hu)
PT (1) PT783490E (hu)
WO (1) WO1996010562A1 (hu)

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JP4879988B2 (ja) 2005-09-29 2012-02-22 メルク・シャープ・エンド・ドーム・コーポレイション メラノコルチン−４受容体モジュレーターとしてのアシル化スピロピペリジン誘導体
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GEP20115337B (en) 2007-01-10 2011-11-25 St Di Ricerche Di Biologia Molecolare P Angeletti Spa Amide substituted indazoles as poly(adp-ribose)polymerase (parp) inhibitors
JP5319518B2 (ja) 2007-04-02 2013-10-16 Ｍｓｄ株式会社 インドールジオン誘導体
US8389553B2 (en) 2007-06-27 2013-03-05 Merck Sharp & Dohme Corp. 4-carboxybenzylamino derivatives as histone deacetylase inhibitors
EP2247185B1 (en) 2008-03-03 2014-04-16 Tiger Pharmatech Tyrosine kinase inhibitors
US9156812B2 (en) 2008-06-04 2015-10-13 Bristol-Myers Squibb Company Crystalline form of 6-[(4S)-2-methyl-4-(2-naphthyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]pyridazin-3-amine
WO2010114780A1 (en) 2009-04-01 2010-10-07 Merck Sharp & Dohme Corp. Inhibitors of akt activity
KR20130009577A (ko) 2009-04-20 2013-01-23 오스펙스 파마슈티컬즈 엘엘씨 야누스 키나아제 3의 피페리딘 억제제
JP5739415B2 (ja) 2009-05-12 2015-06-24 ブリストル−マイヤーズ スクウィブ カンパニー （Ｓ）−７−（［１，２，４］トリアゾロ［１，５−ａ］ピリジン−６−イル）−４−（３，４−ジクロロフェニル）−１，２，３，４−テトラヒドロイソキノリンの結晶形態およびその使用
EA020553B1 (ru) 2009-05-12 2014-12-30 Олбани Молекьюлар Рисерч, Инк. 7-([1,2,4]ТРИАЗОЛО[1,5-α]ПИРИДИН-6-ИЛ)-4-(3,4-ДИХЛОРФЕНИЛ)-1,2,3,4-ТЕТРАГИДРОИЗОХИНОЛИН, ФАРМАЦЕВТИЧЕСКАЯ КОМПОЗИЦИЯ НА ЕГО ОСНОВЕ И СПОСОБЫ ЛЕЧЕНИЯ НЕВРОЛОГИЧЕСКИХ И ПСИХИЧЕСКИХ РАССТРОЙСТВ
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Also Published As

Publication number Publication date
EP0783490A1 (en) 1997-07-16
JPH10506399A (ja) 1998-06-23
CA2198382A1 (en) 1996-04-11
US5935951A (en) 1999-08-10
MX9702092A (es) 1997-10-31
WO1996010562A1 (en) 1996-04-11
PT783490E (pt) 2002-06-28
AU3607895A (en) 1996-04-26
ES2172595T3 (es) 2002-10-01
FI971260A0 (fi) 1997-03-26
DE69525355T2 (de) 2002-09-19
NO971383D0 (no) 1997-03-24
DE69525355D1 (de) 2002-03-21
NO971383L (no) 1997-05-14
DK0783490T3 (da) 2002-05-13
EP0783490B1 (en) 2002-02-06
ATE212981T1 (de) 2002-02-15
FI971260A (fi) 1997-03-26

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Legal Events

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