HUT65627A - Process for producing of alkynyl-derivatives of indolyl-methoxybenzoyl-benzenesulphonemide compounds and pharmaceutical compositions comprising them - Google Patents

Process for producing of alkynyl-derivatives of indolyl-methoxybenzoyl-benzenesulphonemide compounds and pharmaceutical compositions comprising them Download PDF

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Publication number
HUT65627A
HUT65627A HU9203343A HU9203343A HUT65627A HU T65627 A HUT65627 A HU T65627A HU 9203343 A HU9203343 A HU 9203343A HU 9203343 A HU9203343 A HU 9203343A HU T65627 A HUT65627 A HU T65627A
Authority
HU
Hungary
Prior art keywords
formula
group
compound
benzenesulfonamide
ylmethyl
Prior art date
Application number
HU9203343A
Other languages
English (en)
Hungarian (hu)
Other versions
HU9203343D0 (en
Inventor
Rolf Schurter
Alfred Sallmann
Marc Gerspacher
Original Assignee
Ciba Geigy Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag
Publication of HU9203343D0 publication Critical patent/HU9203343D0/hu
Publication of HUT65627A publication Critical patent/HUT65627A/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/14—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/18—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D209/24—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals with an alkyl or cycloalkyl radical attached to the ring nitrogen atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/14—Decongestants or antiallergics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Communicable Diseases (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Oncology (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Indole Compounds (AREA)
HU9203343A 1991-10-25 1992-10-22 Process for producing of alkynyl-derivatives of indolyl-methoxybenzoyl-benzenesulphonemide compounds and pharmaceutical compositions comprising them HUT65627A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH313591 1991-10-25

Publications (2)

Publication Number Publication Date
HU9203343D0 HU9203343D0 (en) 1992-12-28
HUT65627A true HUT65627A (en) 1994-07-28

Family

ID=4249377

Family Applications (1)

Application Number Title Priority Date Filing Date
HU9203343A HUT65627A (en) 1991-10-25 1992-10-22 Process for producing of alkynyl-derivatives of indolyl-methoxybenzoyl-benzenesulphonemide compounds and pharmaceutical compositions comprising them

Country Status (13)

Country Link
US (1) US5248693A (enExample)
EP (1) EP0539329A1 (enExample)
JP (1) JPH05221980A (enExample)
KR (1) KR930007902A (enExample)
AU (1) AU2723292A (enExample)
CA (1) CA2081262A1 (enExample)
FI (1) FI924768L (enExample)
HU (1) HUT65627A (enExample)
IL (1) IL103524A0 (enExample)
MX (1) MX9206127A (enExample)
NO (1) NO924112L (enExample)
TW (1) TW207531B (enExample)
ZA (1) ZA928201B (enExample)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2072125T3 (es) * 1991-10-25 1995-07-01 Ciba Geigy Ag Procedimiento para la obtencion de indoles substituidos.
US5439929A (en) * 1994-03-01 1995-08-08 Pfizer Inc. Bicyclic carbamates, pharmaceutical compositions and use
GB9804648D0 (en) 1998-03-06 1998-04-29 Zeneca Ltd Chemical compounds
GB9805520D0 (en) * 1998-03-17 1998-05-13 Zeneca Ltd Chemical compounds
GB9811427D0 (en) 1998-05-29 1998-07-22 Zeneca Ltd Chemical compounds
ES2273725T3 (es) 1999-09-04 2007-05-16 Astrazeneca Ab Derivados de hidroxiacetamidobencenosulfonamida.
ES2307528T3 (es) 1999-09-04 2008-12-01 Astrazeneca Ab Amidas como inhibidores para la piruvato deshidrogenasa.
ES2216940T3 (es) 1999-09-04 2004-11-01 Astrazeneca Ab Derivados n-fenilicos de 2-hidroxi-2-metil-3,3,3-trifluoropropanamida sustituidos que elevan la actividad de piruvato deshidrogenasa.
GB0120471D0 (en) * 2001-08-23 2001-10-17 Astrazeneca Ab Chemical compounds
EP2981324B1 (en) * 2013-04-05 2020-01-01 Miller, Leonard B. Methods and articles of manufacture for the treatment of skin
CN108084077B (zh) * 2017-12-20 2020-04-14 江汉大学 一种扎鲁司特中间体的合成方法
CN112516080B (zh) * 2018-01-23 2023-09-19 盛元医药广州有限公司 一种眼用药物组合物及其制备方法和应用
CN115458713B (zh) * 2022-10-21 2024-04-19 深圳市山木新能源科技股份有限公司 一种聚阴离子钠离子电池电极

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8607294D0 (en) * 1985-04-17 1986-04-30 Ici America Inc Heterocyclic amide derivatives
DK496086A (da) * 1985-10-17 1987-04-18 Ici America Inc Heterocykliske forbindelser
GB8623429D0 (en) * 1985-10-17 1986-11-05 Ici America Inc Carboximide derivatives
GB8906032D0 (en) * 1988-04-14 1989-04-26 Ici America Inc Hetera-aliphatic carboxamides
DE59103389D1 (de) * 1990-05-04 1994-12-08 Ciba Geigy Ag Substituierte Indole.

Also Published As

Publication number Publication date
TW207531B (enExample) 1993-06-11
US5248693A (en) 1993-09-28
FI924768A0 (fi) 1992-10-21
HU9203343D0 (en) 1992-12-28
IL103524A0 (en) 1993-03-15
KR930007902A (ko) 1993-05-20
FI924768A7 (fi) 1993-04-26
AU2723292A (en) 1993-04-29
NO924112L (no) 1993-04-26
JPH05221980A (ja) 1993-08-31
CA2081262A1 (en) 1993-04-26
EP0539329A1 (de) 1993-04-28
MX9206127A (es) 1993-08-01
FI924768L (fi) 1993-04-26
ZA928201B (en) 1993-04-28
NO924112D0 (no) 1992-10-23

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Legal Events

Date Code Title Description
DFD9 Temporary protection cancelled due to non-payment of fee