HUP0004819A2 - Mikrobicid N-alfa-szulfonil-N-{[(alkinil-oxi)-fenil]-etil}-glicin-amid-származékok, intermedierjeik, előállításuk és alkalmazásuk - Google Patents

Mikrobicid N-alfa-szulfonil-N-{[(alkinil-oxi)-fenil]-etil}-glicin-amid-származékok, intermedierjeik, előállításuk és alkalmazásuk

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Publication number
HUP0004819A2
HUP0004819A2 HU0004819A HUP0004819A HUP0004819A2 HU P0004819 A2 HUP0004819 A2 HU P0004819A2 HU 0004819 A HU0004819 A HU 0004819A HU P0004819 A HUP0004819 A HU P0004819A HU P0004819 A2 HUP0004819 A2 HU P0004819A2
Authority
HU
Hungary
Prior art keywords
group
cycloalkyl
alkyl
optionally substituted
alkyl group
Prior art date
Application number
HU0004819A
Other languages
English (en)
Inventor
André Jeanguenat
Martin Zeller
Original Assignee
Novartis Ag.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag. filed Critical Novartis Ag.
Publication of HUP0004819A2 publication Critical patent/HUP0004819A2/hu
Publication of HUP0004819A3 publication Critical patent/HUP0004819A3/hu

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/01Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms
    • C07C311/02Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
    • C07C311/03Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atoms of the sulfonamide groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C311/06Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atoms of the sulfonamide groups bound to hydrogen atoms or to acyclic carbon atoms to acyclic carbon atoms of hydrocarbon radicals substituted by carboxyl groups
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N41/00Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a sulfur atom bound to a hetero atom
    • A01N41/02Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a sulfur atom bound to a hetero atom containing a sulfur-to-oxygen double bond
    • A01N41/04Sulfonic acids; Derivatives thereof
    • A01N41/06Sulfonic acid amides
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/02Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms
    • A01N43/04Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom
    • A01N43/06Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom five-membered rings
    • A01N43/10Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom five-membered rings with sulfur as the ring hetero atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C217/00Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton
    • C07C217/54Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups bound to carbon atoms of at least one six-membered aromatic ring and amino groups bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton
    • C07C217/56Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups bound to carbon atoms of at least one six-membered aromatic ring and amino groups bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton with amino groups linked to the six-membered aromatic ring, or to the condensed ring system containing that ring, by carbon chains not further substituted by singly-bound oxygen atoms
    • C07C217/60Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups bound to carbon atoms of at least one six-membered aromatic ring and amino groups bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton with amino groups linked to the six-membered aromatic ring, or to the condensed ring system containing that ring, by carbon chains not further substituted by singly-bound oxygen atoms linked by carbon chains having two carbon atoms between the amino groups and the six-membered aromatic ring or the condensed ring system containing that ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C237/00Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
    • C07C237/02Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C237/04Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being acyclic and saturated
    • C07C237/08Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being acyclic and saturated having the nitrogen atom of at least one of the carboxamide groups bound to an acyclic carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C307/00Amides of sulfuric acids, i.e. compounds having singly-bound oxygen atoms of sulfate groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C307/04Diamides of sulfuric acids
    • C07C307/06Diamides of sulfuric acids having nitrogen atoms of the sulfamide groups bound to acyclic carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/01Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms
    • C07C311/11Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic unsaturated carbon skeleton
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C313/00Sulfinic acids; Sulfenic acids; Halides, esters or anhydrides thereof; Amides of sulfinic or sulfenic acids, i.e. compounds having singly-bound oxygen atoms of sulfinic or sulfenic groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C313/02Sulfinic acids; Derivatives thereof
    • C07C313/06Sulfinamides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/14Radicals substituted by singly bound hetero atoms other than halogen
    • C07D333/16Radicals substituted by singly bound hetero atoms other than halogen by oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00Systems containing only non-condensed rings
    • C07C2601/12Systems containing only non-condensed rings with a six-membered ring
    • C07C2601/14The ring being saturated

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

A találmány szerinti vegyületek (I) általánosképletében n 0 vagy 1; Rl adott esetben alkoxi-, alkil-tio-, alkil-szulfonil-cikloalkil-, ciano-, alkoxi-karbonil-, (alkenil-oxi)-karbonil- vagy (alkinil-oxi)-karbonil-csoporttal szubsztituáltalkilcsoport; cikloalkil-alkenil-, alkinil-, halogén-alkil- vagy -NR11R12 általános képletű csoport, amelyben R11 és R12 hidrogénatomvagy alkilcsoport, vagy R11 és R12 együtt tetra- vagy pentametilén-csoport; R2 és R3 hidrogénatom; adott esetben hidroxi-, alkoxi-merkapto- vagy alkil-tio-csoporttal szubsztituált alkilcsoport;alkenil-alkinil- cikloalkil-, cikloalkil-alkil-csoport vagy R2 és R3azzal a szénatommal együtt, amelyhez kapcsolódik, egy 3-8 tagú gyűrűtképez: R4, R5, R6 és R7 hidrogénatom vagy alkilcsoport; R8 alkil-,alkenil- vagy alkinilcsoport; A alkilincsoport; és B mono- vagypoliciklusos, adott esetben szubsztituált aril-csoport; mono- vagypoliciklusos, adott esetben szubsztituált heteroaril-csoport,alkilcsoport; vagy cikloalkil-csoport - és lehetséges izomereikre, valamint izomerkeverékeikre vonatkozik. Azúj vegyületek növények fitopatogén mikroorganizmusok által okozottfertőzésekkel szembeni védelmére alkalmazhatók. Ó
HU0004819A 1997-08-06 1998-08-04 Microbicidal n-sulfonylglycin alkynyloxyphenemethyl amide derivatives HUP0004819A3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH186497 1997-08-06
PCT/EP1998/004849 WO1999007674A2 (en) 1997-08-06 1998-08-04 Microbicidal n-sulfonylglycin alkynyloxyphenemethyl amide derivatives

Publications (2)

Publication Number Publication Date
HUP0004819A2 true HUP0004819A2 (hu) 2001-05-28
HUP0004819A3 HUP0004819A3 (en) 2002-01-28

Family

ID=4220395

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0004819A HUP0004819A3 (en) 1997-08-06 1998-08-04 Microbicidal n-sulfonylglycin alkynyloxyphenemethyl amide derivatives

Country Status (24)

Country Link
US (1) US6482859B1 (hu)
EP (1) EP1003719B1 (hu)
JP (1) JP4163379B2 (hu)
KR (1) KR100609625B1 (hu)
CN (1) CN1215054C (hu)
AR (1) AR013391A1 (hu)
AT (1) ATE218540T1 (hu)
AU (1) AU738007B2 (hu)
BR (1) BR9811846B1 (hu)
CA (1) CA2293451A1 (hu)
DE (1) DE69805807T2 (hu)
DK (1) DK1003719T3 (hu)
ES (1) ES2178259T3 (hu)
GT (1) GT199800109A (hu)
HU (1) HUP0004819A3 (hu)
IL (1) IL134266A (hu)
NZ (1) NZ502508A (hu)
PL (1) PL195781B1 (hu)
PT (1) PT1003719E (hu)
RU (1) RU2221778C2 (hu)
TR (1) TR200000213T2 (hu)
TW (1) TW491832B (hu)
WO (1) WO1999007674A2 (hu)
ZA (1) ZA987017B (hu)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9826650D0 (en) * 1998-12-03 1999-01-27 Novartis Ag Organic compounds
TW564244B (en) * 1999-01-11 2003-12-01 Novartis Ag Novel propargylether derivatives
RU2002121647A (ru) * 2000-01-25 2004-01-10 Зингента Партисипейшнс Аг (Ch) 3-фенокси-1-фенилпроизводные ацетиленового ряда и их применение в качестве гербицидов
GB0011944D0 (en) * 2000-05-17 2000-07-05 Novartis Ag Organic compounds
US20030189958A1 (en) * 2000-09-12 2003-10-09 Cosima Nuninger Fungicidal compositions
GB0022338D0 (en) * 2000-09-12 2000-10-25 Novartis Ag Organic Compounds
GB0127554D0 (en) * 2001-11-16 2002-01-09 Syngenta Participations Ag Organic compounds
GB0227966D0 (en) * 2002-11-29 2003-01-08 Syngenta Participations Ag Organic Compounds
US7803889B2 (en) 2003-02-28 2010-09-28 Daikin Industries, Ltd. Granulated powder of low-molecular polytetrafluoro-ethylene and powder of low-molecular polytetrafluoro-ethylene and processes for producing both
GB0403864D0 (en) * 2004-02-20 2004-03-24 Ucl Ventures Modulator
WO2006024333A2 (en) * 2004-08-17 2006-03-09 Syngenta Participations Ag Aqueous neonicotinoid compositions for seed treatment
PE20060796A1 (es) 2004-11-25 2006-09-29 Basf Ag Procedimiento para intensificar la eficiencia de etaboxam
GB0516705D0 (en) * 2005-08-15 2005-09-21 Syngenta Participations Ag Process
JP5713677B2 (ja) 2008-09-30 2015-05-07 株式会社レイテック 成形加工が可能なポリテトラフルオロエチレン樹脂と応用製品およびその製造方法
CN101503381B (zh) * 2009-03-05 2012-09-05 中国农业大学 1-氧代四氢萘基-2-磺酰胺,其制备方法和作为杀菌剂的用途
GB0906515D0 (en) 2009-04-15 2009-05-20 Syngenta Participations Ag Fungical compositions
CA3006745C (en) 2010-11-05 2021-03-30 Oat Agrio Co., Ltd. Ethynylphenylamidine compound or salt thereof, method for producing same, and fungicide for agricultural and horticultural use
CN108503528B (zh) * 2018-05-14 2021-02-09 韦丽 一种抗凝血药物替卡格雷中间体原料的合成方法
CN108503508B (zh) * 2018-05-14 2021-02-02 广州润霖医药科技有限公司 一种抗凝血药物替卡格雷原料中间体的合成方法
CN115667236B (zh) * 2020-04-26 2024-04-26 江苏恩华药业股份有限公司 1,5-二氢-2,4-苯二氮䓬-3-酮衍生物及其应用
CN112110800B (zh) * 2020-09-25 2022-06-24 哈尔滨工业大学(深圳) 一种3-芳基-2-丙炔-1-醇类衍生物及其制备方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2140411C1 (ru) * 1994-05-04 1999-10-27 Новартис Аг Амиды n-сульфонил- и n-сульфиниламинокислот в качестве микробицидов
HUP9901137A3 (en) * 1995-10-18 2001-01-29 Novartis Ag N-sulphonyl and n-sulphinyl amino acid derivatives, preparation thereof, microbicide compositions containing these compounds as active ingredients and use thereof
ES2186145T3 (es) * 1997-02-25 2003-05-01 Syngenta Participations Ag Amidas de n-sulfonil y n-sulfinil aminoacidos como microbicidas.
DE69805774T2 (de) * 1997-02-25 2003-03-06 Syngenta Participations Ag N-sulphonyl- und n-sulphinylaminosaüreamide als microbiozide

Also Published As

Publication number Publication date
US6482859B1 (en) 2002-11-19
EP1003719B1 (en) 2002-06-05
CN1266426A (zh) 2000-09-13
CN1215054C (zh) 2005-08-17
TR200000213T2 (tr) 2000-08-21
ATE218540T1 (de) 2002-06-15
PL337827A1 (en) 2000-09-11
PT1003719E (pt) 2002-10-31
NZ502508A (en) 2002-05-31
JP4163379B2 (ja) 2008-10-08
GT199800109A (es) 2000-01-13
AU9338898A (en) 1999-03-01
KR100609625B1 (ko) 2006-08-09
BR9811846A (pt) 2000-08-08
DE69805807D1 (de) 2002-07-11
AU738007B2 (en) 2001-09-06
HUP0004819A3 (en) 2002-01-28
ZA987017B (en) 1999-02-08
AR013391A1 (es) 2000-12-27
PL195781B1 (pl) 2007-10-31
WO1999007674A2 (en) 1999-02-18
DK1003719T3 (da) 2002-10-14
WO1999007674A3 (en) 1999-04-15
IL134266A0 (en) 2001-04-30
ES2178259T3 (es) 2002-12-16
TW491832B (en) 2002-06-21
BR9811846B1 (pt) 2010-03-09
KR20010022635A (ko) 2001-03-26
EP1003719A2 (en) 2000-05-31
DE69805807T2 (de) 2003-02-06
RU2221778C2 (ru) 2004-01-20
JP2001513529A (ja) 2001-09-04
CA2293451A1 (en) 1999-02-18
IL134266A (en) 2005-11-20

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