HUP0003632A2 - Eljárás szubsztituált 2-nitro-guanidin-származékok és intermedierjeik előállítására - Google Patents

Eljárás szubsztituált 2-nitro-guanidin-származékok és intermedierjeik előállítására

Info

Publication number
HUP0003632A2
HUP0003632A2 HU0003632A HUP0003632A HUP0003632A2 HU P0003632 A2 HUP0003632 A2 HU P0003632A2 HU 0003632 A HU0003632 A HU 0003632A HU P0003632 A HUP0003632 A HU P0003632A HU P0003632 A2 HUP0003632 A2 HU P0003632A2
Authority
HU
Hungary
Prior art keywords
general formula
group
alkyl
optionally substituted
intermediates
Prior art date
Application number
HU0003632A
Other languages
English (en)
Inventor
Peter Maienfisch
Original Assignee
Novartis Ag.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag. filed Critical Novartis Ag.
Publication of HUP0003632A2 publication Critical patent/HUP0003632A2/hu
Publication of HUP0003632A3 publication Critical patent/HUP0003632A3/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C211/00—Compounds containing amino groups bound to a carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/61—Halogen atoms or nitro radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D251/00—Heterocyclic compounds containing 1,3,5-triazine rings
    • C07D251/02—Heterocyclic compounds containing 1,3,5-triazine rings not condensed with other rings
    • C07D251/08—Heterocyclic compounds containing 1,3,5-triazine rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pyridine Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Furan Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

A találmány tárgya eljárás egy általános képletű vegyület - aképletben R1 hidrogénatom vagy alkilcsoport; R2 hidrogénatom, alkil-, cikloalkil- vagy -CH2B általános képletűcsoport; A adott esetben szubsztituált aromás vagy nemaromás, mono- vagybiciklusos heterogyűrűs csoport; és B adott esetben szubsztituált fenil-, 3-piridil- vagy tiazolilcsoport-előállítására. Az eljárás során egy általános képletű vegyületet -amely képletben R1, R2 és A az (I) általános képletnél megadott; R3 adott esetben szubsztituált alkil-, cikloalkil-, alkenil-,alkinilcsoport, -N(R4)R5 általános képletű csoport, adott esetbenszubsztituált arilcsoport vagy heterogyűrűs csoport; R4 hidrogénatom vagy alkilcsoport; R5 hidrogénatom, alkil-, alkil-karbonil- vagy alkoxi-karbonil-csoport- hidrolizálnak. A találmány tárgya továbbá eljárás a (II) általánosképletű intermedierek, valamint ez utóbbiak kiindulási anyagainak, aáltalános képletű vegyületeknek az előállítására. Az (I) általánosképletű vegyületek peszticid hatóanyagok előállítására használhatók. Ó
HU0003632A 1997-08-20 1998-08-18 Method for producing substituted 2-nitroguanidine derivatives and their intermediates HUP0003632A3 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH195197 1997-08-20

Publications (2)

Publication Number Publication Date
HUP0003632A2 true HUP0003632A2 (hu) 2001-02-28
HUP0003632A3 HUP0003632A3 (en) 2002-11-28

Family

ID=4222414

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0003632A HUP0003632A3 (en) 1997-08-20 1998-08-18 Method for producing substituted 2-nitroguanidine derivatives and their intermediates

Country Status (12)

Country Link
EP (1) EP1005456A1 (hu)
JP (1) JP2001515066A (hu)
KR (1) KR20010023053A (hu)
CN (1) CN1271346A (hu)
AU (1) AU741658B2 (hu)
BR (1) BR9811966A (hu)
CA (1) CA2301172A1 (hu)
HU (1) HUP0003632A3 (hu)
ID (1) ID24319A (hu)
IL (1) IL134502A0 (hu)
PL (1) PL338778A1 (hu)
WO (1) WO1999009009A1 (hu)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19806469A1 (de) * 1998-02-17 1999-08-19 Bayer Ag Verfahren zur Herstellung von 1,3-disubstituierten 2-Nitroguanidinen
US6518433B1 (en) * 1998-03-19 2003-02-11 Syngenta Crop Protection, Inc. Process for the preparation of nitroguanidine derivatives
DE19961604A1 (de) 1999-12-21 2001-07-05 Bayer Ag Verfahren zur Herstellung von 1,3-disubstituierten 2-Nitroguanidinen
DE10121652A1 (de) * 2001-05-03 2002-11-07 Bayer Ag Verfahren zur Herstellung von 1,3-disubstituierten 2-Nitroguanidinen
ES2266618T3 (es) * 2001-08-23 2007-03-01 Bayer Cropscience S.A. Propargilaminas substituidas.
CN102070629A (zh) * 2010-12-28 2011-05-25 上海师范大学 新烟碱噻虫胺类似物杀虫剂及其制备方法
CN103254171A (zh) * 2013-04-16 2013-08-21 中国农业大学 一类含芳杂环三嗪类(反)-β-法尼烯类似物及其应用

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2779403B2 (ja) * 1988-11-29 1998-07-23 日本バイエルアグロケム株式会社 殺虫性ニトロ化合物
IE71183B1 (en) * 1988-12-27 1997-01-29 Takeda Chemical Industries Ltd Guanidine derivatives their production and insecticides
DE69004452T2 (de) * 1989-02-13 1994-03-10 Bayer Agrochem Kk Nitroverbindungen als Insektizide.
AU6044790A (en) * 1989-07-28 1991-03-11 Nippon Soda Co., Ltd. Triazine derivatives
AU628229B2 (en) * 1989-11-10 1992-09-10 Agro-Kanesho Co. Ltd. Hexahydrotriazine compounds and insecticides
JPH0674249B2 (ja) * 1990-04-05 1994-09-21 アグロカネショウ株式会社 置換ニトログアニジン類の製造法
IL99576A0 (en) * 1990-10-05 1992-08-18 Ciba Geigy Ag Triazacyclohexane derivatives
TW198724B (hu) * 1990-10-24 1993-01-21 Ciba Geigy Ag
JP2766848B2 (ja) * 1993-10-26 1998-06-18 三井化学株式会社 フラニル系殺虫剤
JP3258502B2 (ja) * 1993-10-26 2002-02-18 三井化学株式会社 殺虫性テトラヒドロフラン誘導体

Also Published As

Publication number Publication date
JP2001515066A (ja) 2001-09-18
PL338778A1 (en) 2000-11-20
CA2301172A1 (en) 1999-02-25
EP1005456A1 (de) 2000-06-07
BR9811966A (pt) 2000-08-15
AU741658B2 (en) 2001-12-06
KR20010023053A (ko) 2001-03-26
IL134502A0 (en) 2001-04-30
ID24319A (id) 2000-07-13
WO1999009009A1 (de) 1999-02-25
AU9344298A (en) 1999-03-08
CN1271346A (zh) 2000-10-25
HUP0003632A3 (en) 2002-11-28

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Legal Events

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FD9A Lapse of provisional protection due to non-payment of fees