HUP0003632A2 - Eljárás szubsztituált 2-nitro-guanidin-származékok és intermedierjeik előállítására - Google Patents
Eljárás szubsztituált 2-nitro-guanidin-származékok és intermedierjeik előállításáraInfo
- Publication number
- HUP0003632A2 HUP0003632A2 HU0003632A HUP0003632A HUP0003632A2 HU P0003632 A2 HUP0003632 A2 HU P0003632A2 HU 0003632 A HU0003632 A HU 0003632A HU P0003632 A HUP0003632 A HU P0003632A HU P0003632 A2 HUP0003632 A2 HU P0003632A2
- Authority
- HU
- Hungary
- Prior art keywords
- general formula
- group
- alkyl
- optionally substituted
- intermediates
- Prior art date
Links
- 238000004519 manufacturing process Methods 0.000 title abstract 3
- 239000000543 intermediate Substances 0.000 title abstract 2
- IDCPFAYURAQKDZ-UHFFFAOYSA-N 1-nitroguanidine Chemical class NC(=N)N[N+]([O-])=O IDCPFAYURAQKDZ-UHFFFAOYSA-N 0.000 title 1
- 125000000217 alkyl group Chemical group 0.000 abstract 4
- 150000001875 compounds Chemical class 0.000 abstract 4
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 4
- 238000000034 method Methods 0.000 abstract 3
- 125000003118 aryl group Chemical group 0.000 abstract 2
- 125000000753 cycloalkyl group Chemical group 0.000 abstract 2
- 125000003349 3-pyridyl group Chemical group N1=C([H])C([*])=C([H])C([H])=C1[H] 0.000 abstract 1
- 239000004480 active ingredient Substances 0.000 abstract 1
- 125000003342 alkenyl group Chemical group 0.000 abstract 1
- 125000004453 alkoxycarbonyl group Chemical group 0.000 abstract 1
- 125000004448 alkyl carbonyl group Chemical group 0.000 abstract 1
- 125000000304 alkynyl group Chemical group 0.000 abstract 1
- 125000002618 bicyclic heterocycle group Chemical group 0.000 abstract 1
- 125000000623 heterocyclic group Chemical group 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 125000002911 monocyclic heterocycle group Chemical group 0.000 abstract 1
- 239000000575 pesticide Substances 0.000 abstract 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
- 239000007858 starting material Substances 0.000 abstract 1
- 125000000547 substituted alkyl group Chemical group 0.000 abstract 1
- 125000003107 substituted aryl group Chemical group 0.000 abstract 1
- 125000000335 thiazolyl group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C211/00—Compounds containing amino groups bound to a carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/61—Halogen atoms or nitro radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D251/00—Heterocyclic compounds containing 1,3,5-triazine rings
- C07D251/02—Heterocyclic compounds containing 1,3,5-triazine rings not condensed with other rings
- C07D251/08—Heterocyclic compounds containing 1,3,5-triazine rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pyridine Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Furan Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Abstract
A találmány tárgya eljárás egy általános képletű vegyület - aképletben R1 hidrogénatom vagy alkilcsoport; R2 hidrogénatom, alkil-, cikloalkil- vagy -CH2B általános képletűcsoport; A adott esetben szubsztituált aromás vagy nemaromás, mono- vagybiciklusos heterogyűrűs csoport; és B adott esetben szubsztituált fenil-, 3-piridil- vagy tiazolilcsoport-előállítására. Az eljárás során egy általános képletű vegyületet -amely képletben R1, R2 és A az (I) általános képletnél megadott; R3 adott esetben szubsztituált alkil-, cikloalkil-, alkenil-,alkinilcsoport, -N(R4)R5 általános képletű csoport, adott esetbenszubsztituált arilcsoport vagy heterogyűrűs csoport; R4 hidrogénatom vagy alkilcsoport; R5 hidrogénatom, alkil-, alkil-karbonil- vagy alkoxi-karbonil-csoport- hidrolizálnak. A találmány tárgya továbbá eljárás a (II) általánosképletű intermedierek, valamint ez utóbbiak kiindulási anyagainak, aáltalános képletű vegyületeknek az előállítására. Az (I) általánosképletű vegyületek peszticid hatóanyagok előállítására használhatók. Ó
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CH195197 | 1997-08-20 |
Publications (2)
Publication Number | Publication Date |
---|---|
HUP0003632A2 true HUP0003632A2 (hu) | 2001-02-28 |
HUP0003632A3 HUP0003632A3 (en) | 2002-11-28 |
Family
ID=4222414
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HU0003632A HUP0003632A3 (en) | 1997-08-20 | 1998-08-18 | Method for producing substituted 2-nitroguanidine derivatives and their intermediates |
Country Status (12)
Country | Link |
---|---|
EP (1) | EP1005456A1 (hu) |
JP (1) | JP2001515066A (hu) |
KR (1) | KR20010023053A (hu) |
CN (1) | CN1271346A (hu) |
AU (1) | AU741658B2 (hu) |
BR (1) | BR9811966A (hu) |
CA (1) | CA2301172A1 (hu) |
HU (1) | HUP0003632A3 (hu) |
ID (1) | ID24319A (hu) |
IL (1) | IL134502A0 (hu) |
PL (1) | PL338778A1 (hu) |
WO (1) | WO1999009009A1 (hu) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE19806469A1 (de) * | 1998-02-17 | 1999-08-19 | Bayer Ag | Verfahren zur Herstellung von 1,3-disubstituierten 2-Nitroguanidinen |
IL138343A0 (en) * | 1998-03-19 | 2001-10-31 | Novartis Ag | Process for the preparation of nitroguanidine derivatives |
DE19961604A1 (de) | 1999-12-21 | 2001-07-05 | Bayer Ag | Verfahren zur Herstellung von 1,3-disubstituierten 2-Nitroguanidinen |
DE10121652A1 (de) * | 2001-05-03 | 2002-11-07 | Bayer Ag | Verfahren zur Herstellung von 1,3-disubstituierten 2-Nitroguanidinen |
ES2266618T3 (es) * | 2001-08-23 | 2007-03-01 | Bayer Cropscience S.A. | Propargilaminas substituidas. |
CN102070629A (zh) * | 2010-12-28 | 2011-05-25 | 上海师范大学 | 新烟碱噻虫胺类似物杀虫剂及其制备方法 |
CN103254171A (zh) * | 2013-04-16 | 2013-08-21 | 中国农业大学 | 一类含芳杂环三嗪类(反)-β-法尼烯类似物及其应用 |
Family Cites Families (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2779403B2 (ja) * | 1988-11-29 | 1998-07-23 | 日本バイエルアグロケム株式会社 | 殺虫性ニトロ化合物 |
IE71183B1 (en) * | 1988-12-27 | 1997-01-29 | Takeda Chemical Industries Ltd | Guanidine derivatives their production and insecticides |
DE69004452T2 (de) * | 1989-02-13 | 1994-03-10 | Bayer Agrochem Kk | Nitroverbindungen als Insektizide. |
WO1991001978A1 (en) * | 1989-07-28 | 1991-02-21 | Nippon Soda Co., Ltd. | Triazine derivatives |
US6187773B1 (en) * | 1989-11-10 | 2001-02-13 | Agro-Kanesho Co., Ltd. | Hexahydrotriazine compounds and insecticides |
JPH0674249B2 (ja) * | 1990-04-05 | 1994-09-21 | アグロカネショウ株式会社 | 置換ニトログアニジン類の製造法 |
EP0483055A1 (de) * | 1990-10-05 | 1992-04-29 | Ciba-Geigy Ag | Triazacyclohexanderivate |
TW198724B (hu) * | 1990-10-24 | 1993-01-21 | Ciba Geigy Ag | |
JP3258502B2 (ja) * | 1993-10-26 | 2002-02-18 | 三井化学株式会社 | 殺虫性テトラヒドロフラン誘導体 |
JP2766848B2 (ja) * | 1993-10-26 | 1998-06-18 | 三井化学株式会社 | フラニル系殺虫剤 |
-
1998
- 1998-08-18 AU AU93442/98A patent/AU741658B2/en not_active Ceased
- 1998-08-18 JP JP2000509693A patent/JP2001515066A/ja active Pending
- 1998-08-18 EP EP98946375A patent/EP1005456A1/de not_active Withdrawn
- 1998-08-18 IL IL13450298A patent/IL134502A0/xx unknown
- 1998-08-18 HU HU0003632A patent/HUP0003632A3/hu unknown
- 1998-08-18 CN CN98809316A patent/CN1271346A/zh active Pending
- 1998-08-18 WO PCT/EP1998/005248 patent/WO1999009009A1/de not_active Application Discontinuation
- 1998-08-18 BR BR9811966-4A patent/BR9811966A/pt not_active IP Right Cessation
- 1998-08-18 CA CA002301172A patent/CA2301172A1/en not_active Abandoned
- 1998-08-18 KR KR1020007001670A patent/KR20010023053A/ko not_active Application Discontinuation
- 1998-08-18 ID IDW20000316A patent/ID24319A/id unknown
- 1998-08-18 PL PL98338778A patent/PL338778A1/xx unknown
Also Published As
Publication number | Publication date |
---|---|
KR20010023053A (ko) | 2001-03-26 |
CN1271346A (zh) | 2000-10-25 |
EP1005456A1 (de) | 2000-06-07 |
JP2001515066A (ja) | 2001-09-18 |
HUP0003632A3 (en) | 2002-11-28 |
CA2301172A1 (en) | 1999-02-25 |
IL134502A0 (en) | 2001-04-30 |
AU741658B2 (en) | 2001-12-06 |
BR9811966A (pt) | 2000-08-15 |
PL338778A1 (en) | 2000-11-20 |
WO1999009009A1 (de) | 1999-02-25 |
ID24319A (id) | 2000-07-13 |
AU9344298A (en) | 1999-03-08 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FD9A | Lapse of provisional protection due to non-payment of fees |