BR9811966A - Método para a produção de derivados substituìdos de 2- nitroguanidina - Google Patents

Método para a produção de derivados substituìdos de 2- nitroguanidina

Info

Publication number
BR9811966A
BR9811966A BR9811966-4A BR9811966A BR9811966A BR 9811966 A BR9811966 A BR 9811966A BR 9811966 A BR9811966 A BR 9811966A BR 9811966 A BR9811966 A BR 9811966A
Authority
BR
Brazil
Prior art keywords
substituted
alkyl
formula
production
hydrogen
Prior art date
Application number
BR9811966-4A
Other languages
English (en)
Inventor
Peter Maienfisch
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of BR9811966A publication Critical patent/BR9811966A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C211/00—Compounds containing amino groups bound to a carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/61—Halogen atoms or nitro radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D251/00—Heterocyclic compounds containing 1,3,5-triazine rings
    • C07D251/02—Heterocyclic compounds containing 1,3,5-triazine rings not condensed with other rings
    • C07D251/08—Heterocyclic compounds containing 1,3,5-triazine rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pyridine Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Furan Compounds (AREA)

Abstract

Patente de Invenção: <B>"MéTODO PARA A PRODUçãO DE DERIVADOS SUBSTITUìDOS DE 2-NITROGUANIDINA"<D>. São descritos um método para a produção de um composto da fórmula: no qual R~ 1~ é hidrogênio ou C~ 1~-C~ 4~ alquila; R~ 2~ é hidrogênio, C~ 1~-C~ 6~ alquila, C~ 3~-C~ 6~ cicloalquila ou um radical -CH~ 2~B; A é um radical heterocíclico, não-substituído ou substituído, aromático ou não-aromático, monocíclico ou bicíclico; e B é fenila, 3-piridila ou tiazolila, as quais são substituídas; caracterizado em que um composto da fórmula: na qual R~ 1~, R~ 2~ e A têm o mesmo significado como os fornecidos para a fórmula (I), e R~ 3~ é C~ 11~-C~ 22~ alquila, C~ 7~-C~ 16~ cicloalquila, C~ 3~-C~ 20~ alquenila, C~ 3~-C~ 20~ alquinila, N(R~ 4~)R~ 5~ não-substituídos ou substituídos, arila opcionalmente substituída, ou um radical heterocíclico opcionalmente substituído; R~ 4~ é hidrogênio ou C~ 1~-C~ 12~ alquila; R~ 5~ é hidrogênio, C~ 1~-C~ 12~ alquila, C~ 1~-C~ 12~ alquilcarbonila ou C~ 1~-C~ 12~ alcóxicarbonila; é hidrolizado; Um método para a produção de compostos das fórmulas (II) e (III), bem como um método para o controle de pragas com a utilização dos compostos da fórmula (II) são descritos. Os compostos da fórmula (I) são adequados para a produção de misturas pesticidas.
BR9811966-4A 1997-08-20 1998-08-18 Método para a produção de derivados substituìdos de 2- nitroguanidina BR9811966A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH195197 1997-08-20
PCT/EP1998/005248 WO1999009009A1 (de) 1997-08-20 1998-08-18 Verfahren zur herstellung von substituierten 2-nitroguanidinderivaten

Publications (1)

Publication Number Publication Date
BR9811966A true BR9811966A (pt) 2000-08-15

Family

ID=4222414

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9811966-4A BR9811966A (pt) 1997-08-20 1998-08-18 Método para a produção de derivados substituìdos de 2- nitroguanidina

Country Status (12)

Country Link
EP (1) EP1005456A1 (pt)
JP (1) JP2001515066A (pt)
KR (1) KR20010023053A (pt)
CN (1) CN1271346A (pt)
AU (1) AU741658B2 (pt)
BR (1) BR9811966A (pt)
CA (1) CA2301172A1 (pt)
HU (1) HUP0003632A3 (pt)
ID (1) ID24319A (pt)
IL (1) IL134502A0 (pt)
PL (1) PL338778A1 (pt)
WO (1) WO1999009009A1 (pt)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19806469A1 (de) * 1998-02-17 1999-08-19 Bayer Ag Verfahren zur Herstellung von 1,3-disubstituierten 2-Nitroguanidinen
KR20010041996A (ko) * 1998-03-19 2001-05-25 한스 루돌프 하우스, 헨리테 브룬너, 베아트리체 귄터 니트로구아니딘 유도체의 제조 방법
DE19961604A1 (de) * 1999-12-21 2001-07-05 Bayer Ag Verfahren zur Herstellung von 1,3-disubstituierten 2-Nitroguanidinen
DE10121652A1 (de) * 2001-05-03 2002-11-07 Bayer Ag Verfahren zur Herstellung von 1,3-disubstituierten 2-Nitroguanidinen
WO2003017764A1 (de) * 2001-08-23 2003-03-06 Bayer Cropscience S.A. Substituierte propargylamine
CN102070629A (zh) * 2010-12-28 2011-05-25 上海师范大学 新烟碱噻虫胺类似物杀虫剂及其制备方法
CN103254171A (zh) * 2013-04-16 2013-08-21 中国农业大学 一类含芳杂环三嗪类(反)-β-法尼烯类似物及其应用

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2779403B2 (ja) * 1988-11-29 1998-07-23 日本バイエルアグロケム株式会社 殺虫性ニトロ化合物
IE960442L (en) * 1988-12-27 1990-06-27 Takeda Chemical Industries Ltd Guanidine derivatives, their production and insecticides
DK0383091T3 (da) * 1989-02-13 1994-02-07 Bayer Agrochem Kk Insecticidt virksomme nitroforbindelser
AU6044790A (en) * 1989-07-28 1991-03-11 Nippon Soda Co., Ltd. Triazine derivatives
AU628229B2 (en) * 1989-11-10 1992-09-10 Agro-Kanesho Co. Ltd. Hexahydrotriazine compounds and insecticides
JPH0674249B2 (ja) * 1990-04-05 1994-09-21 アグロカネショウ株式会社 置換ニトログアニジン類の製造法
IL99576A0 (en) * 1990-10-05 1992-08-18 Ciba Geigy Ag Triazacyclohexane derivatives
TW198724B (pt) * 1990-10-24 1993-01-21 Ciba Geigy Ag
JP2766848B2 (ja) * 1993-10-26 1998-06-18 三井化学株式会社 フラニル系殺虫剤
JP3258502B2 (ja) * 1993-10-26 2002-02-18 三井化学株式会社 殺虫性テトラヒドロフラン誘導体

Also Published As

Publication number Publication date
HUP0003632A2 (hu) 2001-02-28
CN1271346A (zh) 2000-10-25
JP2001515066A (ja) 2001-09-18
IL134502A0 (en) 2001-04-30
PL338778A1 (en) 2000-11-20
ID24319A (id) 2000-07-13
AU741658B2 (en) 2001-12-06
KR20010023053A (ko) 2001-03-26
AU9344298A (en) 1999-03-08
EP1005456A1 (de) 2000-06-07
CA2301172A1 (en) 1999-02-25
HUP0003632A3 (en) 2002-11-28
WO1999009009A1 (de) 1999-02-25

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Legal Events

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B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 8A E 9A ANUIDADES

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 1912 DE 28/08/2007.