HUP0003141A3 - 4-phenylpiperidine derivatives, process for producing them and pharmaceutical compositions containing them - Google Patents

4-phenylpiperidine derivatives, process for producing them and pharmaceutical compositions containing them

Info

Publication number
HUP0003141A3
HUP0003141A3 HU0003141A HUP0003141A HUP0003141A3 HU P0003141 A3 HUP0003141 A3 HU P0003141A3 HU 0003141 A HU0003141 A HU 0003141A HU P0003141 A HUP0003141 A HU P0003141A HU P0003141 A3 HUP0003141 A3 HU P0003141A3
Authority
HU
Hungary
Prior art keywords
producing
pharmaceutical compositions
compositions containing
phenylpiperidine derivatives
phenylpiperidine
Prior art date
Application number
HU0003141A
Other languages
English (en)
Hungarian (hu)
Original Assignee
Synthon Bv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26647319&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HUP0003141(A3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Synthon Bv filed Critical Synthon Bv
Publication of HUP0003141A2 publication Critical patent/HUP0003141A2/hu
Publication of HUP0003141A3 publication Critical patent/HUP0003141A3/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/06—Antimigraine agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
    • C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D211/20—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Pain & Pain Management (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
HU0003141A 1997-06-10 1997-06-10 4-phenylpiperidine derivatives, process for producing them and pharmaceutical compositions containing them HUP0003141A3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US08/872,023 US5874447A (en) 1997-06-10 1997-06-10 4-Phenylpiperidine compounds for treating depression
PCT/NL1997/000328 WO1998056787A1 (en) 1997-06-10 1997-06-10 4-Phenylpiperidine compounds

Publications (2)

Publication Number Publication Date
HUP0003141A2 HUP0003141A2 (en) 2001-03-28
HUP0003141A3 true HUP0003141A3 (en) 2001-04-28

Family

ID=26647319

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0003141A HUP0003141A3 (en) 1997-06-10 1997-06-10 4-phenylpiperidine derivatives, process for producing them and pharmaceutical compositions containing them

Country Status (25)

Country Link
US (4) US5874447A (OSRAM)
EP (2) EP1078925A1 (OSRAM)
JP (1) JP2002503248A (OSRAM)
KR (1) KR100543614B1 (OSRAM)
AT (1) ATE200781T1 (OSRAM)
AU (1) AU3108097A (OSRAM)
BG (1) BG64315B1 (OSRAM)
BR (1) BR9714787A (OSRAM)
CA (1) CA2293247C (OSRAM)
CZ (1) CZ295301B6 (OSRAM)
DE (2) DE29724281U1 (OSRAM)
DK (1) DK0994872T3 (OSRAM)
EE (2) EE03970B1 (OSRAM)
ES (1) ES2155995T3 (OSRAM)
GR (1) GR3035784T3 (OSRAM)
HU (1) HUP0003141A3 (OSRAM)
IL (1) IL133366A (OSRAM)
IS (2) IS1927B (OSRAM)
NO (3) NO317371B1 (OSRAM)
PL (1) PL188450B1 (OSRAM)
PT (1) PT994872E (OSRAM)
SI (1) SI0994872T1 (OSRAM)
SK (1) SK283394B6 (OSRAM)
TR (2) TR200201156T2 (OSRAM)
WO (1) WO1998056787A1 (OSRAM)

Families Citing this family (53)

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KR20010042552A (ko) * 1998-04-09 2001-05-25 피터 기딩스 파록세틴 말레에이트
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US20010023252A1 (en) * 1998-07-02 2001-09-20 Smithkline Beecham Plc Novel compound
GB9814316D0 (en) * 1998-07-02 1998-09-02 Smithkline Beecham Plc Novel compounds
CH689805A8 (fr) * 1998-07-02 2000-02-29 Smithkline Beecham Plc Méthanesulfonate de paroxétine, procédé pour sa préparation et compositions pharmaceutiques le contenant.
WO2000008016A1 (en) * 1998-08-08 2000-02-17 Smithkline Beecham Plc Paroxetine salts
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WO2000078290A2 (en) * 1999-06-22 2000-12-28 Smithkline Beecham P.L.C. Pharmaceutical composition comprising a salt of paroxetine
ES2159260B1 (es) * 1999-06-22 2002-05-01 Smithkline Beechan Plc Nueva composicion de metanosulfonato de paroxetina
GB9914585D0 (en) * 1999-06-22 1999-08-25 Smithkline Beecham Plc Novel process
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GB9919052D0 (en) * 1999-08-12 1999-10-13 Smithkline Beecham Plc Novel compound composition and process
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DE60007782T2 (de) * 2000-05-12 2004-12-09 Synthon B.V. Piperidinverbindungen und verfahren zu deren herstellung
IL154422A0 (en) * 2000-08-28 2003-09-17 Synthon Bv Paroxetine compositions and processes for making the same
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Also Published As

Publication number Publication date
PT994872E (pt) 2001-09-28
SK161999A3 (en) 2000-08-14
US7598271B1 (en) 2009-10-06
EE03970B1 (et) 2003-02-17
CZ295301B6 (cs) 2005-07-13
GR3035784T3 (en) 2001-07-31
US5874447A (en) 1999-02-23
PL188450B1 (pl) 2005-02-28
DK0994872T3 (da) 2001-05-28
IS7098A (is) 2004-01-08
EE9900570A (et) 2000-08-15
TR199903025T2 (xx) 2000-07-21
DE69704679T2 (de) 2001-09-13
BG64315B1 (bg) 2004-09-30
IS1927B (is) 2004-04-15
HUP0003141A2 (en) 2001-03-28
CZ429599A3 (cs) 2000-04-12
KR20010013615A (ko) 2001-02-26
NO20033765L (no) 2000-02-09
EE200200633A (et) 2003-02-17
US20090326233A1 (en) 2009-12-31
SI0994872T1 (OSRAM) 2001-08-31
WO1998056787A1 (en) 1998-12-17
PL336895A1 (en) 2000-07-17
IS5249A (is) 1999-11-16
ES2155995T3 (es) 2001-06-01
DE29724281U1 (de) 2000-08-10
NO20033765D0 (no) 2003-08-25
NO317371B1 (no) 2004-10-18
IL133366A (en) 2005-11-20
CA2293247C (en) 2005-04-12
KR100543614B1 (ko) 2006-01-20
NO995455D0 (no) 1999-11-08
NO20033766D0 (no) 2003-08-25
TR200201156T2 (tr) 2002-07-22
DE69704679D1 (de) 2001-05-31
CA2293247A1 (en) 1998-12-17
EP0994872B1 (en) 2001-04-25
HK1027352A1 (en) 2001-01-12
EP0994872B9 (en) 2001-12-05
NO20033766L (no) 2000-02-09
EP0994872A1 (en) 2000-04-26
BG103980A (en) 2000-07-31
BR9714787A (pt) 2000-07-18
AU3108097A (en) 1998-12-30
ATE200781T1 (de) 2001-05-15
IL133366A0 (en) 2001-04-30
SK283394B6 (sk) 2003-07-01
US6900327B2 (en) 2005-05-31
JP2002503248A (ja) 2002-01-29
EP1078925A1 (en) 2001-02-28
US20010031767A1 (en) 2001-10-18
NO995455L (no) 2000-02-09

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