HUE053911T2 - Tofacitinibet tartalmazó orális, nyújtott hatóanyag-felszabadulású adagolási formák - Google Patents

Tofacitinibet tartalmazó orális, nyújtott hatóanyag-felszabadulású adagolási formák

Info

Publication number
HUE053911T2
HUE053911T2 HUE14726410A HUE14726410A HUE053911T2 HU E053911 T2 HUE053911 T2 HU E053911T2 HU E14726410 A HUE14726410 A HU E14726410A HU E14726410 A HUE14726410 A HU E14726410A HU E053911 T2 HUE053911 T2 HU E053911T2
Authority
HU
Hungary
Prior art keywords
dosage forms
sustained release
release dosage
oral sustained
tofacitinib
Prior art date
Application number
HUE14726410A
Other languages
English (en)
Inventor
Scott Max Herbig
Sriram Krishnaswami
Iv Joseph Kushner
Manisha Lamba
Thomas C Stock
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=50819757&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HUE053911(T2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer filed Critical Pfizer
Publication of HUE053911T4 publication Critical patent/HUE053911T4/hu
Publication of HUE053911T2 publication Critical patent/HUE053911T2/hu

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52—Purines, e.g. adenine
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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    • A61K9/0002—Galenical forms characterised by the drug release technique; Application systems commanded by energy
    • A61K9/0004—Osmotic delivery systems; Sustained release driven by osmosis, thermal energy or gas
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    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
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    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
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    • A61K9/2022—Organic macromolecular compounds
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    • A61K9/2806—Coating materials
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HUE14726410A 2013-03-16 2014-03-12 Tofacitinibet tartalmazó orális, nyújtott hatóanyag-felszabadulású adagolási formák HUE053911T2 (hu)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201361802479P 2013-03-16 2013-03-16
US201361864059P 2013-08-09 2013-08-09
US201461934428P 2014-01-31 2014-01-31

Publications (2)

Publication Number Publication Date
HUE053911T4 HUE053911T4 (hu) 2021-06-28
HUE053911T2 true HUE053911T2 (hu) 2021-07-28

Family

ID=50819757

Family Applications (1)

Application Number Title Priority Date Filing Date
HUE14726410A HUE053911T2 (hu) 2013-03-16 2014-03-12 Tofacitinibet tartalmazó orális, nyújtott hatóanyag-felszabadulású adagolási formák

Country Status (23)

Country Link
US (4) US9937181B2 (hu)
EP (3) EP4249055A3 (hu)
JP (3) JP6041823B2 (hu)
KR (5) KR102151842B1 (hu)
CN (2) CN111419817A (hu)
AU (2) AU2014233850B2 (hu)
BR (1) BR112015020453B1 (hu)
CA (2) CA2905604C (hu)
CY (1) CY1124007T1 (hu)
DK (1) DK2968155T3 (hu)
ES (1) ES2865134T3 (hu)
HK (1) HK1217297A1 (hu)
HU (1) HUE053911T2 (hu)
IL (3) IL241400B (hu)
MX (1) MX2021000550A (hu)
NZ (2) NZ751227A (hu)
PL (1) PL2968155T3 (hu)
PT (1) PT2968155T (hu)
SG (2) SG11201506103UA (hu)
SI (1) SI2968155T1 (hu)
TW (1) TWI619516B (hu)
WO (1) WO2014147526A1 (hu)
ZA (2) ZA201505468B (hu)

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