HUE037343T2 - Policiklusos karmaboilpiridon vegyületek és alkalmazásuk HIV fertõzések kezelésére - Google Patents

Policiklusos karmaboilpiridon vegyületek és alkalmazásuk HIV fertõzések kezelésére

Info

Publication number
HUE037343T2
HUE037343T2 HUE14745053A HUE14745053A HUE037343T2 HU E037343 T2 HUE037343 T2 HU E037343T2 HU E14745053 A HUE14745053 A HU E14745053A HU E14745053 A HUE14745053 A HU E14745053A HU E037343 T2 HUE037343 T2 HU E037343T2
Authority
HU
Hungary
Prior art keywords
karmaboylpyridone
polycyclic
compounds
treatment
hiv infections
Prior art date
Application number
HUE14745053A
Other languages
English (en)
Hungarian (hu)
Inventor
Mingzhe Ji
Teresa Alejandra Trejo Martin
Manoj C Desai
Haolun Jin
Hyung-Jung Pyun
Original Assignee
Gilead Sciences Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gilead Sciences Inc filed Critical Gilead Sciences Inc
Publication of HUE037343T2 publication Critical patent/HUE037343T2/hu

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/18—Bridged systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • AIDS & HIV (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyridine Compounds (AREA)
HUE14745053A 2013-07-12 2014-07-11 Policiklusos karmaboilpiridon vegyületek és alkalmazásuk HIV fertõzések kezelésére HUE037343T2 (hu)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201361845807P 2013-07-12 2013-07-12

Publications (1)

Publication Number Publication Date
HUE037343T2 true HUE037343T2 (hu) 2018-08-28

Family

ID=51257630

Family Applications (1)

Application Number Title Priority Date Filing Date
HUE14745053A HUE037343T2 (hu) 2013-07-12 2014-07-11 Policiklusos karmaboilpiridon vegyületek és alkalmazásuk HIV fertõzések kezelésére

Country Status (18)

Country Link
US (6) US9458159B2 (enExample)
EP (2) EP3252053B1 (enExample)
JP (1) JP6411492B2 (enExample)
AU (3) AU2014286995B2 (enExample)
CA (1) CA2918055C (enExample)
CY (1) CY1119545T1 (enExample)
DK (1) DK3019499T3 (enExample)
ES (2) ES2647216T3 (enExample)
HR (1) HRP20171807T1 (enExample)
HU (1) HUE037343T2 (enExample)
LT (1) LT3019499T (enExample)
NO (1) NO2865735T3 (enExample)
PL (1) PL3019499T3 (enExample)
PT (1) PT3019499T (enExample)
RS (1) RS56539B1 (enExample)
SI (2) SI3019499T1 (enExample)
SM (1) SMT201700525T1 (enExample)
WO (1) WO2015006733A1 (enExample)

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TWI902729B (zh) 2019-11-28 2025-11-01 日商鹽野義製藥股份有限公司 以組合整合酶阻礙劑及抗ｈｉｖ藥為特徵之ｈｉｖ感染症的預防及治療用醫藥
JP7453399B2 (ja) 2020-02-24 2024-03-19 ギリアード サイエンシーズ， インコーポレイテッド Ｈｉｖ感染症を治療するための四環式化合物及びその使用
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