HU194175B - Process for preparing n-phenyl-pyridine-amino-derivatives - Google Patents

Process for preparing n-phenyl-pyridine-amino-derivatives Download PDF

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Publication number
HU194175B
HU194175B HU86638A HU63886A HU194175B HU 194175 B HU194175 B HU 194175B HU 86638 A HU86638 A HU 86638A HU 63886 A HU63886 A HU 63886A HU 194175 B HU194175 B HU 194175B
Authority
HU
Hungary
Prior art keywords
preparation
starting compounds
pyridinyl
formula
appropriate starting
Prior art date
Application number
HU86638A
Other languages
English (en)
Hungarian (hu)
Other versions
HUT40420A (en
Inventor
Jun Roy T Chandler
Sek L Young
Original Assignee
Robins Co Inc A H
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Robins Co Inc A H filed Critical Robins Co Inc A H
Publication of HUT40420A publication Critical patent/HUT40420A/hu
Publication of HU194175B publication Critical patent/HU194175B/hu

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/74—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/75—Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/81—Amides; Imides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Psychiatry (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
HU86638A 1982-07-02 1983-05-12 Process for preparing n-phenyl-pyridine-amino-derivatives HU194175B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/394,551 US4558132A (en) 1982-07-02 1982-07-02 Nitro, amino and aroylamino-N-phenylpyridinamines in a process for preparing pyrido[1,4]benzodiazepines

Publications (2)

Publication Number Publication Date
HUT40420A HUT40420A (en) 1986-12-28
HU194175B true HU194175B (en) 1988-01-28

Family

ID=23559432

Family Applications (2)

Application Number Title Priority Date Filing Date
HU86638A HU194175B (en) 1982-07-02 1983-05-12 Process for preparing n-phenyl-pyridine-amino-derivatives
HU831647A HU191837B (en) 1982-07-02 1983-05-12 Process for preparing 6-phenyl-11h-pyrido/2,3-b//1,4/-benzodiazepines

Family Applications After (1)

Application Number Title Priority Date Filing Date
HU831647A HU191837B (en) 1982-07-02 1983-05-12 Process for preparing 6-phenyl-11h-pyrido/2,3-b//1,4/-benzodiazepines

Country Status (20)

Country Link
US (1) US4558132A (cg-RX-API-DMAC7.html)
EP (1) EP0099614A3 (cg-RX-API-DMAC7.html)
JP (1) JPS597166A (cg-RX-API-DMAC7.html)
KR (1) KR880001282B1 (cg-RX-API-DMAC7.html)
AU (1) AU550950B2 (cg-RX-API-DMAC7.html)
CA (1) CA1198424A (cg-RX-API-DMAC7.html)
DK (1) DK547782A (cg-RX-API-DMAC7.html)
ES (2) ES518376A0 (cg-RX-API-DMAC7.html)
FI (1) FI78076C (cg-RX-API-DMAC7.html)
GR (1) GR77822B (cg-RX-API-DMAC7.html)
HU (2) HU194175B (cg-RX-API-DMAC7.html)
IE (1) IE54618B1 (cg-RX-API-DMAC7.html)
IL (1) IL67508A (cg-RX-API-DMAC7.html)
IN (1) IN156481B (cg-RX-API-DMAC7.html)
NO (1) NO158062C (cg-RX-API-DMAC7.html)
NZ (1) NZ202800A (cg-RX-API-DMAC7.html)
PH (1) PH21401A (cg-RX-API-DMAC7.html)
PL (4) PL141485B1 (cg-RX-API-DMAC7.html)
PT (1) PT76093B (cg-RX-API-DMAC7.html)
ZA (1) ZA829155B (cg-RX-API-DMAC7.html)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3409237A1 (de) * 1984-03-14 1985-09-19 Dr. Karl Thomae Gmbh, 7950 Biberach Kondensierte diazepinone, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
DE3626095A1 (de) * 1986-07-31 1988-02-11 Thomae Gmbh Dr K Neue substituierte pyrido(2,3-b)(1,4)benzodiazepin-6-one, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
US4749788A (en) * 1987-04-13 1988-06-07 A. H. Robins Company, Incorporated Process for the preparation of aryl-pyrido(1,4) benzodiazepines

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2785172A (en) * 1953-06-17 1957-03-12 Searle & Co Dialkylaminoalkylphenetidinopyridine
GB907646A (en) * 1959-01-23 1962-10-10 Wander S A A Method of production of new derivatives of diazepin
FR8363M (cg-RX-API-DMAC7.html) * 1967-02-01 1971-02-15
GB1192995A (en) * 1967-04-12 1970-05-28 Egyt Gyogyszervegyeszeti Gyar Formimino Ethers
GB1268772A (en) * 1968-03-15 1972-03-29 Glaxo Lab Ltd NOVEL alpha-CARBOLINE DERIVATIVES, THE PREPARATION THEREOF AND COMPOSITIONS CONTAINING THE SAME
AT327200B (de) * 1972-09-06 1976-01-26 Degussa Verfahren zur herstellung von neuen aza-10,11-dihydro-5h-dibenzo (b,e)-(1,4) diazepinen sowie deren salzen
AT325052B (de) * 1972-12-07 1975-10-10 Degussa Verfahren zur herstellung von neuen 6-azabenzo-1,5-diazepinen und ihren salzen
DK209976A (da) * 1975-05-28 1976-11-29 Merck & Co Inc Fremgangsmade til fremstilling af 3h-1,2,2-triazol(4,5-b)pyridiner

Also Published As

Publication number Publication date
ES531221A0 (es) 1985-09-01
AU550950B2 (en) 1986-04-10
CA1198424A (en) 1985-12-24
GR77822B (cg-RX-API-DMAC7.html) 1984-09-25
ES8507496A1 (es) 1985-09-01
DK547782A (da) 1984-01-03
NO158062B (no) 1988-03-28
PL241785A1 (en) 1985-02-27
EP0099614A3 (en) 1985-05-29
PL144137B1 (en) 1988-04-30
FI824247A0 (fi) 1982-12-10
PT76093B (en) 1986-01-09
FI824247L (fi) 1984-01-03
HU191837B (en) 1987-04-28
US4558132A (en) 1985-12-10
PL143959B1 (en) 1988-03-31
PL141485B1 (en) 1987-07-31
FI78076B (fi) 1989-02-28
PL144138B1 (en) 1988-04-30
IN156481B (cg-RX-API-DMAC7.html) 1985-08-10
IE54618B1 (en) 1989-12-20
AU9163382A (en) 1984-01-05
PL250096A1 (en) 1985-09-10
PH21401A (en) 1987-10-15
JPS597166A (ja) 1984-01-14
NO824115L (no) 1984-01-03
ES8406441A1 (es) 1984-08-01
EP0099614A2 (en) 1984-02-01
IL67508A (en) 1986-02-28
KR880001282B1 (ko) 1988-07-18
PL250097A1 (en) 1985-09-10
FI78076C (fi) 1989-06-12
PT76093A (en) 1983-02-01
HUT34477A (en) 1985-03-28
ZA829155B (en) 1983-09-28
PL250095A1 (en) 1985-09-10
NZ202800A (en) 1987-07-31
HUT40420A (en) 1986-12-28
NO158062C (no) 1988-07-06
KR840002837A (ko) 1984-07-21
IE822918L (en) 1984-01-02
ES518376A0 (es) 1984-08-01

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Legal Events

Date Code Title Description
HU90 Patent valid on 900628
HMM4 Cancellation of final prot. due to non-payment of fee