HRP20171036T1 - Kombinacija dvaju antiviralnih sredstava za liječenje hepatitisa c - Google Patents

Kombinacija dvaju antiviralnih sredstava za liječenje hepatitisa c Download PDF

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Publication number
HRP20171036T1
HRP20171036T1 HRP20171036TT HRP20171036T HRP20171036T1 HR P20171036 T1 HRP20171036 T1 HR P20171036T1 HR P20171036T T HRP20171036T T HR P20171036TT HR P20171036 T HRP20171036 T HR P20171036T HR P20171036 T1 HRP20171036 T1 HR P20171036T1
Authority
HR
Croatia
Prior art keywords
daas
use according
patient
infected
hcv genotype
Prior art date
Application number
HRP20171036TT
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English (en)
Inventor
Barry M. Bernstein
Sandeep Dutta
Wei Liu
Thomas J. PODSADECKI
Andrew L. Campbell
Rajeev M. Menon
Chih-Wei Lin
Tianli WANG
Walid M. Awni
Sven MENSING
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Abbvie Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=50588882&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HRP20171036(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Abbvie Inc. filed Critical Abbvie Inc.
Publication of HRP20171036T1 publication Critical patent/HRP20171036T1/hr

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4985Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/41841,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/498Pyrazines or piperazines ortho- and peri-condensed with carbocyclic ring systems, e.g. quinoxaline, phenazine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Peptides Or Proteins (AREA)
  • Enzymes And Modification Thereof (AREA)
  • Micro-Organisms Or Cultivation Processes Thereof (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Claims (15)

1. Najmanje dva antivirusna sredstva koja djeluju izravno (DAA) za primjenu u metodi za liječenje HCV infekcije, naznačena time, da navedeni postupak obuhvaća davanje najmanje dva DAA pacijentu koji boluje od HCV infekcije, pri čemu se navedenom pacijentu ne daje interferon niti ribavirin tijekom navedenog liječenja, a navedeni tretman traje 8, 9, 10, 11 ili 12 tjedana, i pri čemu navedeni najmanje dva DAA sadržavaju: [image] ili njegove farmaceutski prihvatljive soli, i [image] ili njegove farmaceutski prihvatljive soli.
2. Najmanje dva DAA za uporabu u skladu s patentnim zahtjevom 1, naznačena time, da navedeno liječenje traje 12 tjedana.
3. Najmanje dva DAA za uporabu u skladu s patentnim zahtjevom 1, naznačena time, da navedeno liječenje traje 8 tjedana.
4. Najmanje dva DAA za uporabu u skladu s bilo kojim od patentnih zahtjeva 1 do 3, naznačena time, da je navedeni pacijent inficiran s HCV genotipom 1.
5. Najmanje dva DAA za uporabu u skladu s bilo kojim od patentnih zahtjeva 1 do 3, naznačena time, da je navedeni pacijent inficiran s HCV genotipom la.
6. Najmanje dva DAA za uporabu u skladu s bilo kojim od patentnih zahtjeva 1 do 3, naznačena time, da je navedeni pacijent inficiran s HCV genotipom 2.
7. Najmanje dva DAA za uporabu u skladu s bilo kojim od patentnih zahtjeva 1 do 3, naznačena time, da je navedeni pacijent inficiran s HCV genotipom 3.
8. Najmanje dva DAA za uporabu u skladu s bilo kojim od patentnih zahtjeva 1 do 3, naznačena time, da je navedeni pacijent inficiran HCV genotipom 4.
9. Najmanje dva DAA za uporabu u skladu s bilo kojim od patentnih zahtjeva 1 do 3, naznačena time, da je navedeni pacijent inficiran HCV genotipom 5.
10. Najmanje dva DAA za uporabu u skladu s bilo kojim od patentnih zahtjeva 1 do 3, naznačena time, da je navedeni pacijent inficiran s HCV genotipom 6.
11. Najmanje dva DAA za uporabu u skladu s bilo kojim od patentnih zahtjeva 1 do 3, naznačena time, da navedeni pacijent nema cirozu.
12. Najmanje dva DAA za uporabu u skladu s bilo kojim od patentnih zahtjeva 1 do 3, naznačena time, da navedeni pacijent ima kompenziranu cirozu.
13. Najmanje dva DAA za uporabu u skladu s bilo kojim od patentnih zahtjeva 1 do 3, naznačena time, da navedeni pacijent prije toga nije bio podvrgnut drugom liječenju HCV infekcije.
14. Najmanje dva DAA za uporabu u skladu s bilo kojim od patentnih zahtjeva 1 do 3, naznačena time, da navedeni pacijent ne reagira na interferon.
15. Najmanje dva DAA za upotrebu prema bilo kojem od patentnih zahtjeva 1 do 14, naznačena time, da se navedena najmanje dva DAA sastoje od (1) Spoja 1 ili njegove farmaceutski prihvatljive soli i (2) Spoja 2 ili njegova farmaceutski prihvatljiva sol .
HRP20171036TT 2013-03-14 2014-03-14 Kombinacija dvaju antiviralnih sredstava za liječenje hepatitisa c HRP20171036T1 (hr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201361783376P 2013-03-14 2013-03-14
PCT/US2014/027423 WO2014152514A1 (en) 2013-03-14 2014-03-14 Combination of two antivirals for treating hepatitis c
EP14719977.2A EP2968301B1 (en) 2013-03-14 2014-03-14 Combination of two antivirals for treating hepatitis c

Publications (1)

Publication Number Publication Date
HRP20171036T1 true HRP20171036T1 (hr) 2017-10-06

Family

ID=50588882

Family Applications (2)

Application Number Title Priority Date Filing Date
HRP20171036TT HRP20171036T1 (hr) 2013-03-14 2014-03-14 Kombinacija dvaju antiviralnih sredstava za liječenje hepatitisa c
HRP20201575TT HRP20201575T1 (hr) 2013-03-14 2020-10-05 Kombinacija dva protuvirusna sredstva namijenjena liječenju hepatitisa c

Family Applications After (1)

Application Number Title Priority Date Filing Date
HRP20201575TT HRP20201575T1 (hr) 2013-03-14 2020-10-05 Kombinacija dva protuvirusna sredstva namijenjena liječenju hepatitisa c

Country Status (25)

Country Link
US (1) US20140275099A1 (hr)
EP (3) EP3766495A1 (hr)
JP (4) JP6441303B2 (hr)
KR (2) KR20210013344A (hr)
CN (2) CN105073113B (hr)
AU (2) AU2014239563B2 (hr)
BR (1) BR112015023017B1 (hr)
CA (1) CA2901810C (hr)
CY (2) CY1119025T1 (hr)
DK (2) DK3213750T3 (hr)
EA (2) EA033257B1 (hr)
ES (2) ES2624980T3 (hr)
HR (2) HRP20171036T1 (hr)
HU (2) HUE033010T2 (hr)
IL (1) IL240419B (hr)
LT (2) LT3213750T (hr)
MX (3) MX373314B (hr)
NZ (2) NZ631155A (hr)
PL (2) PL2968301T3 (hr)
PT (2) PT2968301T (hr)
RS (2) RS56202B1 (hr)
SG (2) SG11201507364SA (hr)
SI (2) SI3213750T1 (hr)
TW (2) TWI642436B (hr)
WO (1) WO2014152514A1 (hr)

Families Citing this family (21)

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Publication number Priority date Publication date Assignee Title
DK3213750T3 (da) 2013-03-14 2020-10-19 Abbvie Inc Kombination af to antivirale midler til behandling af hepatitis c
US11484534B2 (en) 2013-03-14 2022-11-01 Abbvie Inc. Methods for treating HCV
MX2015017953A (es) * 2013-07-02 2016-10-28 Abbvie Inc Metodos para tratar el virus de hepatitis c.
CN105658219A (zh) * 2013-10-25 2016-06-08 艾伯维公司 用于治疗hcv的方法
US20150174194A1 (en) * 2013-12-19 2015-06-25 Abbvie Inc. Methods for treating liver transplant recipients
CA2943054A1 (en) * 2014-04-02 2015-10-08 Abbvie Inc. Methods for treating hcv
MX388482B (es) * 2014-04-02 2025-03-20 Abbvie Inc Métodos para tratar el virus de la hepatitis c.
US20160375017A1 (en) 2015-06-26 2016-12-29 Abbvie Inc. Solid Pharmaceutical Compositions for Treating HCV
HK1250627A1 (zh) * 2015-06-26 2019-01-11 Abbvie Inc. 用於治疗hcv的固体药物组合物
US20180177779A1 (en) * 2015-07-08 2018-06-28 Abbvie Inc. Methods for Treating HCV
US20230385268A1 (en) * 2022-05-17 2023-11-30 Abbvie Inc. Methods for Treating HCV
EA201890334A1 (ru) * 2015-07-17 2018-06-29 Эббви Инк. Твердые фармацевтические композиции для лечения вируса гепатита с
JP7129703B2 (ja) 2016-04-28 2022-09-02 エモリー ユニバーシティー アルキン含有ヌクレオチド及びヌクレオシド治療組成物並びにそれらに関連した使用
JP2019529426A (ja) * 2016-09-23 2019-10-17 アッヴィ・インコーポレイテッド 用量調整
CA2994496A1 (en) * 2017-02-14 2018-08-14 Abbvie Inc. Methods for treating hcv
CA2981993A1 (en) * 2017-08-02 2019-02-02 Abbvie Inc. Methods for treating hcv
WO2019200005A1 (en) * 2018-04-10 2019-10-17 Atea Pharmaceuticals, Inc. Treatment of hcv infected patients with cirrhosis
AU2019384793A1 (en) 2018-11-20 2021-06-10 Abbvie Inc. Methods for treating acute HCV
KR102077833B1 (ko) 2018-12-10 2020-02-14 류형준 기능성 식품조성물
CN111688355B (zh) 2019-03-15 2022-04-12 精工爱普生株式会社 液体吸收体、液体吸收器以及液体喷出装置
AU2020271791A1 (en) * 2019-04-08 2021-11-04 Abbvie Inc. Solid pharmaceutical compositions for treating HCV

Family Cites Families (8)

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Publication number Priority date Publication date Assignee Title
US8937150B2 (en) * 2009-06-11 2015-01-20 Abbvie Inc. Anti-viral compounds
US9394279B2 (en) * 2009-06-11 2016-07-19 Abbvie Inc. Anti-viral compounds
PL2618831T3 (pl) * 2010-09-21 2016-06-30 Enanta Pharm Inc Makrocykliczne inhibitory proteazy serynowej HCV pochodzące od proliny
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PH12014500833A1 (en) 2011-10-21 2014-05-26 Abbvie Inc Methods for treating hcv
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RU2665365C2 (ru) * 2012-09-18 2018-08-29 Эббви Инк. Способы лечения гепатита с
DK3213750T3 (da) 2013-03-14 2020-10-19 Abbvie Inc Kombination af to antivirale midler til behandling af hepatitis c

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Publication number Publication date
AU2016202823B2 (en) 2017-11-23
CN105073113B (zh) 2018-01-02
LT3213750T (lt) 2020-10-26
PL3213750T3 (pl) 2020-12-14
EP3213750B1 (en) 2020-08-12
HUE052113T2 (hu) 2021-04-28
JP2019048868A (ja) 2019-03-28
SI2968301T1 (sl) 2017-07-31
ES2624980T3 (es) 2017-07-18
US20140275099A1 (en) 2014-09-18
KR20210013344A (ko) 2021-02-03
JP6441303B2 (ja) 2018-12-19
JP2020037589A (ja) 2020-03-12
AU2014239563A1 (en) 2015-08-27
CN108159393A (zh) 2018-06-15
KR102210935B1 (ko) 2021-02-02
IL240419B (en) 2019-03-31
HK1223817A1 (en) 2017-08-11
JP6621902B2 (ja) 2019-12-18
EP2968301A1 (en) 2016-01-20
HRP20201575T1 (hr) 2020-12-11
AU2014239563B2 (en) 2016-05-05
MX2015012538A (es) 2016-02-10
MX2020005054A (es) 2020-08-20
DK2968301T3 (en) 2017-07-24
KR20150129032A (ko) 2015-11-18
EP3766495A1 (en) 2021-01-20
CY1119025T1 (el) 2018-01-10
CA2901810A1 (en) 2014-09-25
AU2016202823A1 (en) 2016-05-19
TWI686196B (zh) 2020-03-01
SG11201507364SA (en) 2015-10-29
MX362616B (es) 2019-01-28
RS60881B1 (sr) 2020-11-30
TWI642436B (zh) 2018-12-01
HUE033010T2 (en) 2017-11-28
NZ631155A (en) 2016-05-27
CN105073113A (zh) 2015-11-18
ES2824473T3 (es) 2021-05-12
EA033257B1 (ru) 2019-09-30
PT3213750T (pt) 2020-10-19
HK1244668A1 (en) 2018-08-17
IL240419A0 (en) 2015-09-24
BR112015023017B1 (pt) 2022-08-30
EA201591702A1 (ru) 2016-09-30
PT2968301T (pt) 2017-07-17
TW201834656A (zh) 2018-10-01
EA201991174A1 (ru) 2020-01-31
SG10201708306WA (en) 2017-11-29
CY1123387T1 (el) 2021-12-31
JP2016513695A (ja) 2016-05-16
RS56202B1 (sr) 2017-11-30
CA2901810C (en) 2019-01-08
NZ719137A (en) 2017-11-24
WO2014152514A1 (en) 2014-09-25
MX373314B (es) 2020-05-20
LT2968301T (lt) 2017-05-25
EP2968301B1 (en) 2017-04-19
SI3213750T1 (sl) 2020-11-30
TW201511759A (zh) 2015-04-01
JP2021130720A (ja) 2021-09-09
DK3213750T3 (da) 2020-10-19
EP3213750A1 (en) 2017-09-06
BR112015023017A2 (pt) 2017-07-18
PL2968301T3 (pl) 2017-09-29

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