HRP20140558T1 - Novi postupci za proizvodnju derivata benzofenona - Google Patents

Novi postupci za proizvodnju derivata benzofenona Download PDF

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Publication number
HRP20140558T1
HRP20140558T1 HRP20140558AT HRP20140558T HRP20140558T1 HR P20140558 T1 HRP20140558 T1 HR P20140558T1 HR P20140558A T HRP20140558A T HR P20140558AT HR P20140558 T HRP20140558 T HR P20140558T HR P20140558 T1 HRP20140558 T1 HR P20140558T1
Authority
HR
Croatia
Prior art keywords
compound
formula
preparation
followed
iii
Prior art date
Application number
HRP20140558AT
Other languages
English (en)
Croatian (hr)
Inventor
Lars Eklund
Jonas Nilsson
Original Assignee
Cambrex Karlskoga Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43827282&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HRP20140558(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Cambrex Karlskoga Ab filed Critical Cambrex Karlskoga Ab
Publication of HRP20140558T1 publication Critical patent/HRP20140558T1/hr

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C41/00Preparation of ethers; Preparation of compounds having groups, groups or groups
    • C07C41/01Preparation of ethers
    • C07C41/18Preparation of ethers by reactions not forming ether-oxygen bonds
    • C07C41/30Preparation of ethers by reactions not forming ether-oxygen bonds by increasing the number of carbon atoms, e.g. by oligomerisation
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/12Drugs for genital or sexual disorders; Contraceptives for climacteric disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/30Oestrogens
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/67Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
    • C07C45/68Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms
    • C07C45/72Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms by reaction of compounds containing >C = O groups with the same or other compounds containing >C = O groups

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Endocrinology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Diabetes (AREA)
  • Reproductive Health (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
HRP20140558AT 2010-01-19 2011-01-19 Novi postupci za proizvodnju derivata benzofenona HRP20140558T1 (hr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US29609610P 2010-01-19 2010-01-19
PCT/GB2011/000058 WO2011089385A1 (en) 2010-01-19 2011-01-19 New processes for producing benzophenone derivatives

Publications (1)

Publication Number Publication Date
HRP20140558T1 true HRP20140558T1 (hr) 2014-08-01

Family

ID=43827282

Family Applications (1)

Application Number Title Priority Date Filing Date
HRP20140558AT HRP20140558T1 (hr) 2010-01-19 2011-01-19 Novi postupci za proizvodnju derivata benzofenona

Country Status (13)

Country Link
US (1) US9085519B2 (enExample)
EP (1) EP2526080B1 (enExample)
JP (1) JP5850857B2 (enExample)
CN (1) CN102770402B (enExample)
BR (1) BR112012017845A2 (enExample)
DK (1) DK2526080T3 (enExample)
ES (1) ES2460022T3 (enExample)
HR (1) HRP20140558T1 (enExample)
PL (1) PL2526080T3 (enExample)
PT (1) PT2526080E (enExample)
RS (1) RS53353B (enExample)
SI (1) SI2526080T1 (enExample)
WO (1) WO2011089385A1 (enExample)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20150321983A1 (en) * 2012-10-19 2015-11-12 Fermion Oy A process for the preparation of ospemifene
US9321712B2 (en) 2012-10-19 2016-04-26 Fermion Oy Process for the preparation of ospemifene
CN104030896A (zh) * 2013-03-07 2014-09-10 天津药物研究院 一种简易去除欧司哌米芬特异杂质的方法
MX2017003290A (es) * 2014-09-16 2017-06-21 Shionogi & Co Proceso para la preparacion de derivados de trifenilbuteno.
JP6697467B2 (ja) * 2014-12-29 2020-05-20 オロン エス.ピー.エー. オスペミフェン及びフィスペミフェンを調製するためのプロセス
WO2016110805A1 (en) * 2015-01-09 2016-07-14 Glenmark Pharmaceuticals Limited Process for preparation of ospemifene
JP2019500362A (ja) 2015-12-15 2019-01-10 ビーエーエスエフ ソシエタス・ヨーロピアBasf Se ヒドロキシベンゾフェノンポリグリコールエーテル(メタ)アクリレートの製造方法
EA039048B1 (ru) * 2016-03-15 2021-11-26 Сионоги Энд Ко., Лтд. Способ получения производных феноксиэтанола

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2182786A (en) 1938-09-14 1939-12-12 Dow Chemical Co Hydroxy-alkyl ethers of benzophenone
US2831768A (en) 1956-01-19 1958-04-22 Eastman Kodak Co Polymeric light-sensitive photographic elements
CS196471B1 (cs) 1977-11-28 1980-03-31 Ivan Lukac Nové p-acylované fenoxyetanoly
EP0072475B1 (de) 1981-08-17 1986-08-20 F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft Carbaminsäureester, Verfahren zu deren Herstellung, Schädlingsbekämpfungsmittel, die diese Verbindungen als Wirkstoffe enthalten, sowie Verwendung solcher Verbindungen und Mittel zur Bekämpfung von Schädlingen
GB2126576B (en) 1982-06-25 1985-06-19 Farmos Group Limited Alkane and alkene derivatives
US4625048A (en) * 1982-08-13 1986-11-25 Hoffmann-La Roche Inc. Carbamic acid esters
DE3814781A1 (de) * 1988-04-30 1989-11-09 Basf Ag Verfahren zur herstellung von 2-hydroxy-4-(2'-hydroxyethoxy)-benzophenonen
DE3936592A1 (de) 1989-11-03 1991-05-08 Basf Ag Verfahren zur herstellung und reinigung von 2-hydroxy-4-(2'-hydroxy-ethoxy)phenylarylketonen
GB9418067D0 (en) * 1994-09-07 1994-10-26 Orion Yhtymae Oy Triphenylethylenes for the prevention and treatment of osteoporosis
GB9803521D0 (en) 1998-02-19 1998-04-15 Orion Yhtymo Oy New compounds and pharmaceutical compositions thereof
TW593256B (en) * 1999-11-16 2004-06-21 Hormos Medical Oy Ltd Triphenylalkene derivatives and their use as selective estrogen receptor modulators
DE60104614T2 (de) 2000-02-17 2005-01-05 Appleton Papers Inc., Appleton Verfahren zur herstellung von alkoxy- oder arylmethoxy-aroxyethanen
EP2121553B1 (en) * 2007-02-14 2012-06-27 Hormos Medical Ltd. Method for the preparation of therapeutically valuable triphenylbutene derivatives
WO2008099060A2 (en) 2007-02-14 2008-08-21 Hormos Medical Ltd Methods for the preparation of fispemifene from ospemifene

Also Published As

Publication number Publication date
BR112012017845A2 (pt) 2016-03-29
PT2526080E (pt) 2014-05-06
JP2013517320A (ja) 2013-05-16
EP2526080B1 (en) 2014-03-26
CN102770402A (zh) 2012-11-07
RS53353B (sr) 2014-10-31
DK2526080T3 (da) 2014-04-28
WO2011089385A1 (en) 2011-07-28
US9085519B2 (en) 2015-07-21
PL2526080T3 (pl) 2014-08-29
HK1179244A1 (en) 2013-09-27
EP2526080A1 (en) 2012-11-28
JP5850857B2 (ja) 2016-02-03
ES2460022T3 (es) 2014-05-13
SI2526080T1 (sl) 2014-07-31
CN102770402B (zh) 2016-01-20
US20130035514A1 (en) 2013-02-07

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