BR112012017845A2 - novo processo para produção de derivados de benzofenona - Google Patents

novo processo para produção de derivados de benzofenona

Info

Publication number
BR112012017845A2
BR112012017845A2 BR112012017845A BR112012017845A BR112012017845A2 BR 112012017845 A2 BR112012017845 A2 BR 112012017845A2 BR 112012017845 A BR112012017845 A BR 112012017845A BR 112012017845 A BR112012017845 A BR 112012017845A BR 112012017845 A2 BR112012017845 A2 BR 112012017845A2
Authority
BR
Brazil
Prior art keywords
new process
benzophenone derivatives
production
derivatives
compounds
Prior art date
Application number
BR112012017845A
Other languages
English (en)
Inventor
Lars Eklund
Original Assignee
Cambrex Karlskoga Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43827282&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BR112012017845(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Cambrex Karlskoga Ab filed Critical Cambrex Karlskoga Ab
Publication of BR112012017845A2 publication Critical patent/BR112012017845A2/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C41/00—Preparation of ethers; Preparation of compounds having groups, groups or groups
    • C07C41/01—Preparation of ethers
    • C07C41/18—Preparation of ethers by reactions not forming ether-oxygen bonds
    • C07C41/30—Preparation of ethers by reactions not forming ether-oxygen bonds by increasing the number of carbon atoms, e.g. by oligomerisation
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/12—Drugs for genital or sexual disorders; Contraceptives for climacteric disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/30—Oestrogens
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/67—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
    • C07C45/68—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms
    • C07C45/72—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms by reaction of compounds containing >C = O groups with the same or other compounds containing >C = O groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Endocrinology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Reproductive Health (AREA)
  • Diabetes (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

patente de invenção para: "novo processo para produção de derivados de benzofenona". é proporcionado um processo paqra o preparo de um composto de fórmula i: são conforme descrito na descrição. tais compostos podem, por exemplo, ser medicamentos úteis (ou intermediários para medicamentos).
BR112012017845A 2010-01-19 2011-01-19 novo processo para produção de derivados de benzofenona BR112012017845A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US29609610P 2010-01-19 2010-01-19
PCT/GB2011/000058 WO2011089385A1 (en) 2010-01-19 2011-01-19 New processes for producing benzophenone derivatives

Publications (1)

Publication Number Publication Date
BR112012017845A2 true BR112012017845A2 (pt) 2016-03-29

Family

ID=43827282

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112012017845A BR112012017845A2 (pt) 2010-01-19 2011-01-19 novo processo para produção de derivados de benzofenona

Country Status (14)

Country Link
US (1) US9085519B2 (pt)
EP (1) EP2526080B1 (pt)
JP (1) JP5850857B2 (pt)
CN (1) CN102770402B (pt)
BR (1) BR112012017845A2 (pt)
DK (1) DK2526080T3 (pt)
ES (1) ES2460022T3 (pt)
HK (1) HK1179244A1 (pt)
HR (1) HRP20140558T1 (pt)
PL (1) PL2526080T3 (pt)
PT (1) PT2526080E (pt)
RS (1) RS53353B (pt)
SI (1) SI2526080T1 (pt)
WO (1) WO2011089385A1 (pt)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20150321983A1 (en) * 2012-10-19 2015-11-12 Fermion Oy A process for the preparation of ospemifene
WO2014060639A1 (en) 2012-10-19 2014-04-24 Fermion Oy A process for the preparation of ospemifene
CN104030896A (zh) * 2013-03-07 2014-09-10 天津药物研究院 一种简易去除欧司哌米芬特异杂质的方法
CN107074722A (zh) * 2014-09-16 2017-08-18 盐野义制药株式会社 三苯基丁烯衍生物的制造方法
EP3240771B1 (en) 2014-12-29 2019-02-20 OLON S.p.A. Process for the preparation of ospemifene and fispemifene
US10138190B2 (en) 2015-01-09 2018-11-27 Glenmark Pharmaceuticals Limited Process for preparation of ospemifene
EP3390338A1 (de) * 2015-12-15 2018-10-24 Basf Se Verfahren zur herstellung von hydroxybenzophenonpolyglykolether-(meth)acrylat
EP3835285A1 (en) 2016-03-15 2021-06-16 Shionogi & Co., Ltd Method for producing phenoxyethanol derivative

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2182786A (en) 1938-09-14 1939-12-12 Dow Chemical Co Hydroxy-alkyl ethers of benzophenone
US2831768A (en) 1956-01-19 1958-04-22 Eastman Kodak Co Polymeric light-sensitive photographic elements
CS196471B1 (cs) 1977-11-28 1980-03-31 Ivan Lukac Nové p-acylované fenoxyetanoly
DE3272723D1 (en) 1981-08-17 1986-09-25 Hoffmann La Roche Carbamic esters, preparation thereof, pesticidal compositions on the basis of these compounds and their use in combating pests
GB2126576B (en) 1982-06-25 1985-06-19 Farmos Group Limited Alkane and alkene derivatives
US4625048A (en) 1982-08-13 1986-11-25 Hoffmann-La Roche Inc. Carbamic acid esters
DE3814781A1 (de) * 1988-04-30 1989-11-09 Basf Ag Verfahren zur herstellung von 2-hydroxy-4-(2'-hydroxyethoxy)-benzophenonen
DE3936592A1 (de) * 1989-11-03 1991-05-08 Basf Ag Verfahren zur herstellung und reinigung von 2-hydroxy-4-(2'-hydroxy-ethoxy)phenylarylketonen
GB9418067D0 (en) * 1994-09-07 1994-10-26 Orion Yhtymae Oy Triphenylethylenes for the prevention and treatment of osteoporosis
GB9803521D0 (en) 1998-02-19 1998-04-15 Orion Yhtymo Oy New compounds and pharmaceutical compositions thereof
TW593256B (en) * 1999-11-16 2004-06-21 Hormos Medical Oy Ltd Triphenylalkene derivatives and their use as selective estrogen receptor modulators
ATE272600T1 (de) 2000-02-17 2004-08-15 Appleton Paper Inc Verfahren zur herstellung von alkoxy- oder arylmethoxy-aroxyethanen
WO2008099060A2 (en) 2007-02-14 2008-08-21 Hormos Medical Ltd Methods for the preparation of fispemifene from ospemifene
CN101636372B (zh) * 2007-02-14 2013-03-27 霍尔莫斯医疗有限公司 有治疗价值的三苯基丁烯衍生物的制备方法

Also Published As

Publication number Publication date
CN102770402B (zh) 2016-01-20
PT2526080E (pt) 2014-05-06
WO2011089385A1 (en) 2011-07-28
EP2526080A1 (en) 2012-11-28
US9085519B2 (en) 2015-07-21
EP2526080B1 (en) 2014-03-26
US20130035514A1 (en) 2013-02-07
HRP20140558T1 (hr) 2014-08-01
RS53353B (en) 2014-10-31
SI2526080T1 (sl) 2014-07-31
CN102770402A (zh) 2012-11-07
DK2526080T3 (da) 2014-04-28
JP2013517320A (ja) 2013-05-16
ES2460022T3 (es) 2014-05-13
PL2526080T3 (pl) 2014-08-29
HK1179244A1 (en) 2013-09-27
JP5850857B2 (ja) 2016-02-03

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Legal Events

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B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]

Free format text: DE ACORDO COM O ARTIGO 229-C DA LEI NO 10196/2001, QUE MODIFICOU A LEI NO 9279/96, A CONCESSAO DA PATENTE ESTA CONDICIONADA A ANUENCIA PREVIA DA ANVISA. CONSIDERANDO A APROVACAO DOS TERMOS DO PARECER NO 337/PGF/EA/2010, BEM COMO A PORTARIA INTERMINISTERIAL NO 1065 DE 24/05/2012, ENCAMINHA-SE O PRESENTE PEDIDO PARA AS PROVIDENCIAS CABIVEIS.

B07E Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]
B06U Preliminary requirement: requests with searches performed by other patent offices: procedure suspended [chapter 6.21 patent gazette]
B06A Patent application procedure suspended [chapter 6.1 patent gazette]
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 11A ANUIDADE.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2653 DE 09-11-2021 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.