HN2010002403A - Derivados de quinuclidina como antagonistas de receptores muscarinicos m3 - Google Patents

Derivados de quinuclidina como antagonistas de receptores muscarinicos m3

Info

Publication number
HN2010002403A
HN2010002403A HN2010002403A HN2010002403A HN2010002403A HN 2010002403 A HN2010002403 A HN 2010002403A HN 2010002403 A HN2010002403 A HN 2010002403A HN 2010002403 A HN2010002403 A HN 2010002403A HN 2010002403 A HN2010002403 A HN 2010002403A
Authority
HN
Honduras
Prior art keywords
muscarinic receptors
quinuclidine derivatives
receptors antagonists
pharmaceutical compositions
quinuclidine
Prior art date
Application number
HN2010002403A
Other languages
English (en)
Spanish (es)
Inventor
Lee Ford Rhonan
Nigel Mather Andrew
Mete Antonio
James Bull Richard
Anne Skidmore Elizabeth
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of HN2010002403A publication Critical patent/HN2010002403A/es

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • A—HUMAN NECESSITIES
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    • A61P1/02—Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
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    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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  • Health & Medical Sciences (AREA)
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  • Neurosurgery (AREA)
  • Dermatology (AREA)
  • Diabetes (AREA)
  • Urology & Nephrology (AREA)
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  • Orthopedic Medicine & Surgery (AREA)
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  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
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HN2010002403A 2008-05-13 2010-11-12 Derivados de quinuclidina como antagonistas de receptores muscarinicos m3 HN2010002403A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/GB2008/001647 WO2009138707A1 (en) 2008-05-13 2008-05-13 Quinuclidine derivatives as muscarinic m3 receptor antagonists

Publications (1)

Publication Number Publication Date
HN2010002403A true HN2010002403A (es) 2013-01-28

Family

ID=40361403

Family Applications (1)

Application Number Title Priority Date Filing Date
HN2010002403A HN2010002403A (es) 2008-05-13 2010-11-12 Derivados de quinuclidina como antagonistas de receptores muscarinicos m3

Country Status (17)

Country Link
US (2) US8329729B2 (https=)
EP (1) EP2300464A1 (https=)
JP (1) JP4837800B2 (https=)
CN (1) CN102089304A (https=)
AU (1) AU2008356409B2 (https=)
BR (1) BRPI0822693A2 (https=)
CA (1) CA2723981A1 (https=)
CL (1) CL2009001137A1 (https=)
EA (1) EA017627B1 (https=)
EC (1) ECSP10010606A (https=)
HN (1) HN2010002403A (https=)
IL (1) IL209126A0 (https=)
MX (1) MX2010012189A (https=)
NI (1) NI201000195A (https=)
NZ (1) NZ589091A (https=)
WO (1) WO2009138707A1 (https=)
ZA (1) ZA201007988B (https=)

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TW200825084A (en) 2006-11-14 2008-06-16 Astrazeneca Ab New compounds 521
CN102088976B (zh) * 2008-05-13 2012-12-26 阿斯利康(瑞典)有限公司 包含毒蕈碱性受体拮抗剂和β2-肾上腺素受体激动剂的药物产品
EA017627B1 (ru) 2008-05-13 2013-01-30 Астразенека Аб Хинуклидиновые производные в качестве антагонистов мускаринового м3 рецептора
TW201036957A (en) 2009-02-20 2010-10-16 Astrazeneca Ab Novel salt 628
GB201016912D0 (en) 2010-10-07 2010-11-24 Astrazeneca Ab Novel combination
CN103265478B (zh) * 2013-05-20 2015-09-30 中国人民解放军第二军医大学 巯基烟酸类化合物及其制备方法
CN114716380B (zh) * 2022-04-01 2024-06-21 新乡医学院 一种相转移催化的4-取代吡唑酮类化合物不对称氟化方法
WO2025171311A1 (en) * 2024-02-09 2025-08-14 University Of Florida Research Foundation, Incorporated Aryl and pyridyl amide pesticides and compositions thereof

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FR2155927A1 (en) 1971-10-15 1973-05-25 Synthelabo 1-phenylcyclo hexane carboxylic acid esters - with antispasmodic and anticholinergic activity
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US20110172237A1 (en) 2011-07-14
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US20130030001A1 (en) 2013-01-31
ECSP10010606A (es) 2010-12-30
WO2009138707A1 (en) 2009-11-19
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JP2011520853A (ja) 2011-07-21
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EP2300464A1 (en) 2011-03-30
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AU2008356409A1 (en) 2009-11-19
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EA017627B1 (ru) 2013-01-30
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