CL2009001137A1 - Compuestos derivados de cicloheptanocarboniloxi-1-azonia-biciclo[2.2.2]-octano, moduladores de receptores muscarinicos; composiciones farmaceuticas; proceso de preparacion de dicha composicion; y uso en el tratamiento de una enfermedad pulmonar obstructiva cronica. - Google Patents
Compuestos derivados de cicloheptanocarboniloxi-1-azonia-biciclo[2.2.2]-octano, moduladores de receptores muscarinicos; composiciones farmaceuticas; proceso de preparacion de dicha composicion; y uso en el tratamiento de una enfermedad pulmonar obstructiva cronica.Info
- Publication number
- CL2009001137A1 CL2009001137A1 CL2009001137A CL2009001137A CL2009001137A1 CL 2009001137 A1 CL2009001137 A1 CL 2009001137A1 CL 2009001137 A CL2009001137 A CL 2009001137A CL 2009001137 A CL2009001137 A CL 2009001137A CL 2009001137 A1 CL2009001137 A1 CL 2009001137A1
- Authority
- CL
- Chile
- Prior art keywords
- composition
- cycloheptanecarbonyloxy
- azonia
- bicyclo
- modulators
- Prior art date
Links
- 208000006545 Chronic Obstructive Pulmonary Disease Diseases 0.000 title abstract 2
- 102000014415 Muscarinic acetylcholine receptor Human genes 0.000 title abstract 2
- 108050003473 Muscarinic acetylcholine receptor Proteins 0.000 title abstract 2
- 150000001875 compounds Chemical class 0.000 title abstract 2
- -1 cycloheptanecarbonyloxy-1-azonia-bicyclo [2.2.2] -octane Chemical compound 0.000 title abstract 2
- 238000000034 method Methods 0.000 title abstract 2
- 239000000203 mixture Substances 0.000 title abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
- C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
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- Health & Medical Sciences (AREA)
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- Veterinary Medicine (AREA)
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Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PCT/GB2008/001647 WO2009138707A1 (en) | 2008-05-13 | 2008-05-13 | Quinuclidine derivatives as muscarinic m3 receptor antagonists |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CL2009001137A1 true CL2009001137A1 (es) | 2009-11-27 |
Family
ID=40361403
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CL2009001137A CL2009001137A1 (es) | 2008-05-13 | 2009-05-11 | Compuestos derivados de cicloheptanocarboniloxi-1-azonia-biciclo[2.2.2]-octano, moduladores de receptores muscarinicos; composiciones farmaceuticas; proceso de preparacion de dicha composicion; y uso en el tratamiento de una enfermedad pulmonar obstructiva cronica. |
Country Status (17)
| Country | Link |
|---|---|
| US (2) | US8329729B2 (https=) |
| EP (1) | EP2300464A1 (https=) |
| JP (1) | JP4837800B2 (https=) |
| CN (1) | CN102089304A (https=) |
| AU (1) | AU2008356409B2 (https=) |
| BR (1) | BRPI0822693A2 (https=) |
| CA (1) | CA2723981A1 (https=) |
| CL (1) | CL2009001137A1 (https=) |
| EA (1) | EA017627B1 (https=) |
| EC (1) | ECSP10010606A (https=) |
| HN (1) | HN2010002403A (https=) |
| IL (1) | IL209126A0 (https=) |
| MX (1) | MX2010012189A (https=) |
| NI (1) | NI201000195A (https=) |
| NZ (1) | NZ589091A (https=) |
| WO (1) | WO2009138707A1 (https=) |
| ZA (1) | ZA201007988B (https=) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5807670A (en) * | 1995-08-14 | 1998-09-15 | Abbott Laboratories | Detection of hepatitis GB virus genotypes |
| TW200825084A (en) | 2006-11-14 | 2008-06-16 | Astrazeneca Ab | New compounds 521 |
| CN102088976B (zh) * | 2008-05-13 | 2012-12-26 | 阿斯利康(瑞典)有限公司 | 包含毒蕈碱性受体拮抗剂和β2-肾上腺素受体激动剂的药物产品 |
| EA017627B1 (ru) | 2008-05-13 | 2013-01-30 | Астразенека Аб | Хинуклидиновые производные в качестве антагонистов мускаринового м3 рецептора |
| TW201036957A (en) | 2009-02-20 | 2010-10-16 | Astrazeneca Ab | Novel salt 628 |
| GB201016912D0 (en) | 2010-10-07 | 2010-11-24 | Astrazeneca Ab | Novel combination |
| CN103265478B (zh) * | 2013-05-20 | 2015-09-30 | 中国人民解放军第二军医大学 | 巯基烟酸类化合物及其制备方法 |
| CN114716380B (zh) * | 2022-04-01 | 2024-06-21 | 新乡医学院 | 一种相转移催化的4-取代吡唑酮类化合物不对称氟化方法 |
| WO2025171311A1 (en) * | 2024-02-09 | 2025-08-14 | University Of Florida Research Foundation, Incorporated | Aryl and pyridyl amide pesticides and compositions thereof |
Family Cites Families (81)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NL62140C (https=) * | 1942-12-16 | |||
| DE2104179C3 (de) | 1971-01-29 | 1980-10-02 | Knoll Ag, 6700 Ludwigshafen | exo-2-Phenyl-bicyclo- [2,2,1] -heptan-2- (N-methylpiperidol-4)-carbonsäureester und dessen Salze, Verfahren zu deren Herstellung sowie diese enthaltende Arzneimittel |
| FR2155927A1 (en) | 1971-10-15 | 1973-05-25 | Synthelabo | 1-phenylcyclo hexane carboxylic acid esters - with antispasmodic and anticholinergic activity |
| FR2168881A1 (en) | 1972-01-25 | 1973-09-07 | Synthelabo | Tropanol 1-phenylcycloalkane carboxylic ester salts - spasmolytics and cholinergics |
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-
2008
- 2008-05-13 EA EA201001645A patent/EA017627B1/ru not_active IP Right Cessation
- 2008-05-13 EP EP08750581A patent/EP2300464A1/en not_active Withdrawn
- 2008-05-13 WO PCT/GB2008/001647 patent/WO2009138707A1/en not_active Ceased
- 2008-05-13 BR BRPI0822693-8A patent/BRPI0822693A2/pt not_active IP Right Cessation
- 2008-05-13 CA CA2723981A patent/CA2723981A1/en not_active Abandoned
- 2008-05-13 JP JP2011508991A patent/JP4837800B2/ja not_active Expired - Fee Related
- 2008-05-13 CN CN2008801303428A patent/CN102089304A/zh active Pending
- 2008-05-13 US US12/992,045 patent/US8329729B2/en not_active Expired - Fee Related
- 2008-05-13 NZ NZ589091A patent/NZ589091A/en not_active IP Right Cessation
- 2008-05-13 MX MX2010012189A patent/MX2010012189A/es not_active Application Discontinuation
- 2008-05-13 AU AU2008356409A patent/AU2008356409B2/en not_active Ceased
-
2009
- 2009-05-11 CL CL2009001137A patent/CL2009001137A1/es unknown
-
2010
- 2010-11-04 IL IL209126A patent/IL209126A0/en unknown
- 2010-11-08 ZA ZA2010/07988A patent/ZA201007988B/en unknown
- 2010-11-12 HN HN2010002403A patent/HN2010002403A/es unknown
- 2010-11-12 NI NI201000195A patent/NI201000195A/es unknown
- 2010-11-12 EC EC2010010606A patent/ECSP10010606A/es unknown
-
2012
- 2012-08-01 US US13/564,194 patent/US20130030001A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| US8329729B2 (en) | 2012-12-11 |
| HN2010002403A (es) | 2013-01-28 |
| US20110172237A1 (en) | 2011-07-14 |
| EA201001645A1 (ru) | 2011-06-30 |
| US20130030001A1 (en) | 2013-01-31 |
| ECSP10010606A (es) | 2010-12-30 |
| WO2009138707A1 (en) | 2009-11-19 |
| MX2010012189A (es) | 2011-03-02 |
| JP2011520853A (ja) | 2011-07-21 |
| IL209126A0 (en) | 2011-01-31 |
| JP4837800B2 (ja) | 2011-12-14 |
| WO2009138707A9 (en) | 2010-01-28 |
| EP2300464A1 (en) | 2011-03-30 |
| BRPI0822693A2 (pt) | 2015-07-07 |
| CN102089304A (zh) | 2011-06-08 |
| AU2008356409A1 (en) | 2009-11-19 |
| NZ589091A (en) | 2011-07-29 |
| CA2723981A1 (en) | 2009-11-19 |
| ZA201007988B (en) | 2011-07-27 |
| AU2008356409B2 (en) | 2012-01-19 |
| EA017627B1 (ru) | 2013-01-30 |
| NI201000195A (es) | 2012-08-16 |
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