CL2006002831A1 - Compuestos derivados de sulfonamida: proceso de preparacion; composicion farmaceutica; y uso en el tratamiento de una enfermedad mediada por el receptor de glucocorticoides. - Google Patents
Compuestos derivados de sulfonamida: proceso de preparacion; composicion farmaceutica; y uso en el tratamiento de una enfermedad mediada por el receptor de glucocorticoides.Info
- Publication number
- CL2006002831A1 CL2006002831A1 CL200602831A CL2006002831A CL2006002831A1 CL 2006002831 A1 CL2006002831 A1 CL 2006002831A1 CL 200602831 A CL200602831 A CL 200602831A CL 2006002831 A CL2006002831 A CL 2006002831A CL 2006002831 A1 CL2006002831 A1 CL 2006002831A1
- Authority
- CL
- Chile
- Prior art keywords
- sulfonamide
- treatment
- pharmaceutical composition
- preparation process
- glucocorticoid receptor
- Prior art date
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- C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
- C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
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- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
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- Diabetes (AREA)
- Immunology (AREA)
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- Cardiology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Heart & Thoracic Surgery (AREA)
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Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SE0502325 | 2005-10-20 | ||
SE0600747 | 2006-04-03 |
Publications (1)
Publication Number | Publication Date |
---|---|
CL2006002831A1 true CL2006002831A1 (es) | 2008-02-22 |
Family
ID=37962757
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CL200602831A CL2006002831A1 (es) | 2005-10-20 | 2006-10-19 | Compuestos derivados de sulfonamida: proceso de preparacion; composicion farmaceutica; y uso en el tratamiento de una enfermedad mediada por el receptor de glucocorticoides. |
Country Status (10)
Country | Link |
---|---|
US (1) | US20090124607A1 (es) |
EP (1) | EP1940800A4 (es) |
JP (1) | JP2009512687A (es) |
AR (1) | AR056877A1 (es) |
CA (1) | CA2628577A1 (es) |
CL (1) | CL2006002831A1 (es) |
PE (1) | PE20070712A1 (es) |
TW (1) | TW200815361A (es) |
UY (1) | UY29875A1 (es) |
WO (1) | WO2007046747A1 (es) |
Families Citing this family (27)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE10238722A1 (de) | 2002-08-23 | 2004-03-11 | Bayer Ag | Selektive Phosphodiesterase 9A-Inhibitoren als Arzneimittel zur Verbesserung kognitiver Prozesse |
GB0620385D0 (en) * | 2006-10-13 | 2006-11-22 | Glaxo Group Ltd | Novel compounds |
CN101573340A (zh) | 2006-11-01 | 2009-11-04 | 百时美施贵宝公司 | 糖皮质激素受体AP-1和/或NF-κB活性的调节剂及其用途 |
TW200829578A (en) * | 2006-11-23 | 2008-07-16 | Astrazeneca Ab | Chemical compounds 537 |
JO2754B1 (en) * | 2006-12-21 | 2014-03-15 | استرازينكا ايه بي | Amylendazoleil derivatives for the treatment of glucocorticoid-mediated disorders |
GB0704407D0 (en) | 2007-03-07 | 2007-04-18 | Glaxo Group Ltd | Compounds |
EP2136634A4 (en) * | 2007-04-10 | 2011-07-06 | Boehringer Ingelheim Int | MIMETIC GLUCOCORTICOID SUBSTANCES, PREPARATION METHODS THEREOF, PHARMACEUTICAL COMPOSITIONS AND USES THEREOF |
GB0720557D0 (en) * | 2007-10-19 | 2007-11-28 | Glaxo Group Ltd | Novel compounds |
GB0720549D0 (en) * | 2007-10-19 | 2007-11-28 | Glaxo Group Ltd | Novel compounds |
GB0720556D0 (en) * | 2007-10-19 | 2007-11-28 | Glaxo Group Ltd | Novel compounds |
JP5498392B2 (ja) | 2007-11-30 | 2014-05-21 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 1,5−ジヒドロ−ピラゾロ[3,4−d]ピリミジン−4−オン誘導体及びcns障害の治療のためのpde9aモジュレーターとしてのそれらの使用 |
GB0724254D0 (en) * | 2007-12-12 | 2008-01-23 | Glaxo Group Ltd | Novel compounds |
CA2716136A1 (en) * | 2008-03-06 | 2009-09-11 | William P. Dankulich | Hexahydrocyclopentyl[f]indazole sulfonamides and derivatives thereof as selective glucocorticoid receptor modulators |
EP2489660A1 (en) * | 2008-03-20 | 2012-08-22 | Abbott Laboratories | Methods for making central nervous system agents that are TRPV1 antagonists |
UA105362C2 (en) | 2008-04-02 | 2014-05-12 | Бьорингер Ингельхайм Интернациональ Гмбх | 1-heterocyclyl-1, 5-dihydro-pyrazolo [3, 4-d] pyrimidin-4-one derivatives and their use as pde9a modulators |
TWI445705B (zh) * | 2008-05-20 | 2014-07-21 | Astrazeneca Ab | 經苯基及苯并二基取代之吲唑衍生物 |
WO2009142588A1 (en) * | 2008-05-20 | 2009-11-26 | Astrazeneca Ab | Combination of (a) a chemokine receptor 1 (ccr1) antagonist and (b) glucocorticoid receptor modulator |
WO2009142589A1 (en) * | 2008-05-20 | 2009-11-26 | Astrazeneca Ab | Combination of (a) glucocorticoid receptor modulator and (b) a muscarinic antagonist |
WO2009142568A1 (en) * | 2008-05-20 | 2009-11-26 | Astrazeneca Ab | Combination of (a) glucocorticoid receptor modulator and (b) a b2-agonist |
NZ590788A (en) | 2008-09-08 | 2012-11-30 | Boehringer Ingelheim Int | Pyrazolopyrimidines and their use for the treatment of cns disorders |
MX2011010184A (es) | 2009-03-31 | 2011-10-28 | Boehringer Ingelheim Int | Derivados de 1-heterociclil-1,5-dihidro-pirazolo[3,4-d]pirimidin-4 -ona y su uso como moduladores de pde9a. |
CN105541849B (zh) | 2010-08-12 | 2018-03-23 | 勃林格殷格翰国际有限公司 | 6‑环烷基‑1,5‑二氢‑吡唑并[3,4‑d]嘧啶‑4‑酮衍生物及其作为PDE9A抑制剂的用途 |
US8809345B2 (en) | 2011-02-15 | 2014-08-19 | Boehringer Ingelheim International Gmbh | 6-cycloalkyl-pyrazolopyrimidinones for the treatment of CNS disorders |
US9149346B1 (en) * | 2014-10-17 | 2015-10-06 | Kelly Walter Lee Caldiero | Method for synthetic polymer tooth replacement |
KR102412146B1 (ko) | 2015-02-11 | 2022-06-22 | 주식회사 아이엔테라퓨틱스 | 소디움 채널 차단제 |
WO2017161518A1 (en) | 2016-03-23 | 2017-09-28 | Astrazeneca Ab | New physical form |
CA3125929A1 (en) * | 2019-01-11 | 2020-07-16 | Grunenthal Gmbh | Substituted pyrrolidine amides iii |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3992441A (en) * | 1972-12-26 | 1976-11-16 | Pfizer Inc. | Sulfamylbenzoic acids |
DE3535167A1 (de) * | 1985-10-02 | 1987-04-09 | Boehringer Mannheim Gmbh | Neue sulfonyl-phenyl(alkyl)amine, verfahren zu ihrer herstellung sowie arzneimittel |
GB9504854D0 (en) * | 1994-03-31 | 1995-04-26 | Zeneca Ltd | Nitrogen derivatives |
DE19856475A1 (de) * | 1998-11-27 | 2000-05-31 | Schering Ag | Nichtsteroidale Entzündungshemmer |
ATE473740T1 (de) * | 2002-08-29 | 2010-07-15 | Boehringer Ingelheim Pharma | 3-(sulfonamidoethyl)-indol-derivate zur verwendung als glucocorticoid-mimetika bei der behandlung von entzündlichen, allergischen und proliferativen erkrankungen |
-
2006
- 2006-10-16 TW TW095138026A patent/TW200815361A/zh unknown
- 2006-10-18 CA CA002628577A patent/CA2628577A1/en not_active Abandoned
- 2006-10-18 EP EP06799780A patent/EP1940800A4/en not_active Withdrawn
- 2006-10-18 US US12/090,442 patent/US20090124607A1/en not_active Abandoned
- 2006-10-18 JP JP2008536543A patent/JP2009512687A/ja active Pending
- 2006-10-18 WO PCT/SE2006/001181 patent/WO2007046747A1/en active Application Filing
- 2006-10-19 UY UY29875A patent/UY29875A1/es not_active Application Discontinuation
- 2006-10-19 CL CL200602831A patent/CL2006002831A1/es unknown
- 2006-10-19 PE PE2006001271A patent/PE20070712A1/es not_active Application Discontinuation
- 2006-10-20 AR ARP060104613A patent/AR056877A1/es not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
WO2007046747A1 (en) | 2007-04-26 |
US20090124607A1 (en) | 2009-05-14 |
JP2009512687A (ja) | 2009-03-26 |
EP1940800A1 (en) | 2008-07-09 |
PE20070712A1 (es) | 2007-09-21 |
TW200815361A (en) | 2008-04-01 |
UY29875A1 (es) | 2007-05-31 |
CA2628577A1 (en) | 2007-04-26 |
EP1940800A4 (en) | 2009-12-30 |
AR056877A1 (es) | 2007-10-31 |
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