HN2007015177A - Derivados de triazolopirazina - Google Patents

Derivados de triazolopirazina

Info

Publication number
HN2007015177A
HN2007015177A HN2007015177A HN2007015177A HN2007015177A HN 2007015177 A HN2007015177 A HN 2007015177A HN 2007015177 A HN2007015177 A HN 2007015177A HN 2007015177 A HN2007015177 A HN 2007015177A HN 2007015177 A HN2007015177 A HN 2007015177A
Authority
HN
Honduras
Prior art keywords
triazolopirazine
derivatives
canceres
mammals
useful
Prior art date
Application number
HN2007015177A
Other languages
English (en)
Inventor
Cheng Hengmiao
Jean Cui Jingrong
Elizabeth Hoffman Jacqui
Jia Lei
Catherine Johnson Mary
Steven Kania Robert
Thi Quy Le Phuong
David Nambu Mitchell
Alan Pairish Mason
Shen Hong
Bich Tran-Dube Michelle
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of HN2007015177A publication Critical patent/HN2007015177A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/50—Pyridazines; Hydrogenated pyridazines
    • A61K31/5025—Pyridazines; Hydrogenated pyridazines ortho- or peri-condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

ESTA INVENCION SE REFIERE A NUEVOS DERIVADOS DE TRIAZOLOPIRAZINA QUE SON UTILES EN EL TRATAMIENTO DE ENFERMEDADES HIPERPROLIFERATIVAS, TALES COMO CANCERES EN MAMIFEROS.
HN2007015177A 2006-05-11 2007-05-09 Derivados de triazolopirazina HN2007015177A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US79996606P 2006-05-11 2006-05-11
US89323107P 2007-03-06 2007-03-06

Publications (1)

Publication Number Publication Date
HN2007015177A true HN2007015177A (es) 2010-06-09

Family

ID=38441445

Family Applications (1)

Application Number Title Priority Date Filing Date
HN2007015177A HN2007015177A (es) 2006-05-11 2007-05-09 Derivados de triazolopirazina

Country Status (32)

Country Link
US (2) US7732604B2 (es)
EP (1) EP2018383B1 (es)
JP (1) JP4377962B2 (es)
KR (1) KR101099161B1 (es)
CN (1) CN101443331A (es)
AP (1) AP2008004674A0 (es)
AR (1) AR060994A1 (es)
AT (1) ATE532785T1 (es)
AU (1) AU2007251283A1 (es)
BR (1) BRPI0711809A2 (es)
CA (1) CA2651363C (es)
CR (1) CR10383A (es)
EA (1) EA016204B1 (es)
EC (1) ECSP088871A (es)
ES (1) ES2376913T3 (es)
GE (1) GEP20115174B (es)
GT (1) GT200700039A (es)
HN (1) HN2007015177A (es)
IL (1) IL194813A0 (es)
MA (1) MA30411B1 (es)
ME (1) MEP36508A (es)
MX (1) MX2008014399A (es)
NL (1) NL2000613C2 (es)
NO (1) NO20085060L (es)
NZ (1) NZ572361A (es)
PE (1) PE20080067A1 (es)
RS (1) RS20080533A (es)
TN (1) TNSN08445A1 (es)
TW (1) TWI346115B (es)
UY (1) UY30334A1 (es)
WO (1) WO2007132308A1 (es)
ZA (1) ZA200809020B (es)

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DE102008019907A1 (de) 2008-04-21 2009-10-22 Merck Patent Gmbh Pyridazinonderivate
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US8592448B2 (en) 2008-11-20 2013-11-26 OSI Pharmaceuticals, LLC Substituted pyrrolo[2,3-b]-pyridines and -pyrazines
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CN107922396B (zh) * 2015-07-20 2022-08-05 建新公司 集落刺激因子-1受体(csf-1r)抑制剂
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JP6659850B2 (ja) * 2015-12-31 2020-03-04 シャンハイ ファーマシューティカルズ ホールディング カンパニー，リミティド キノリン系化合物の塩、その結晶形、調製方法、組成物及び用途
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Also Published As

Publication number Publication date
TNSN08445A1 (fr) 2010-04-14
KR20090006187A (ko) 2009-01-14
TWI346115B (en) 2011-08-01
MEP36508A (en) 2011-02-10
WO2007132308A1 (en) 2007-11-22
PE20080067A1 (es) 2008-03-10
BRPI0711809A2 (pt) 2011-12-06
EA200870423A1 (ru) 2009-04-28
CR10383A (es) 2008-11-11
ECSP088871A (es) 2008-12-30
US20070265272A1 (en) 2007-11-15
EA016204B1 (ru) 2012-03-30
GEP20115174B (en) 2011-03-10
ATE532785T1 (de) 2011-11-15
IL194813A0 (en) 2009-08-03
CA2651363A1 (en) 2007-11-22
ZA200809020B (en) 2009-12-30
MX2008014399A (es) 2008-11-27
AR060994A1 (es) 2008-07-30
RS20080533A (en) 2009-09-08
AP2008004674A0 (en) 2008-12-31
ES2376913T3 (es) 2012-03-20
JP2009536636A (ja) 2009-10-15
NL2000613C2 (nl) 2007-11-20
TW200804384A (en) 2008-01-16
CA2651363C (en) 2011-07-12
UY30334A1 (es) 2008-01-02
US7732604B2 (en) 2010-06-08
KR101099161B1 (ko) 2011-12-27
MA30411B1 (fr) 2009-05-04
EP2018383A1 (en) 2009-01-28
GT200700039A (es) 2008-06-02
CN101443331A (zh) 2009-05-27
NO20085060L (no) 2008-12-03
AU2007251283A1 (en) 2007-11-22
JP4377962B2 (ja) 2009-12-02
US20100105656A1 (en) 2010-04-29
EP2018383B1 (en) 2011-11-09
NZ572361A (en) 2012-02-24

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