HK82697A - 3-[2-(dimethylamino)ethyl]-N-methyl-1H-indole-5-methane-sulphonamide sulphate (2:1) - Google Patents

3-[2-(dimethylamino)ethyl]-N-methyl-1H-indole-5-methane-sulphonamide sulphate (2:1)

Info

Publication number
HK82697A
HK82697A HK82697A HK82697A HK82697A HK 82697 A HK82697 A HK 82697A HK 82697 A HK82697 A HK 82697A HK 82697 A HK82697 A HK 82697A HK 82697 A HK82697 A HK 82697A
Authority
HK
Hong Kong
Prior art keywords
sulphonamide
indole
sulphate
dimethylamino
methane
Prior art date
Application number
HK82697A
Other languages
English (en)
Inventor
Joanne Craig
Derek Leslie Crookes
Stephen John Skittrall
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of HK82697A publication Critical patent/HK82697A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/14—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
    • C07D209/16—Tryptamines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/06—Antimigraine agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A61P29/02—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID] without antiinflammatory effect

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Indole Compounds (AREA)
HK82697A 1990-12-12 1997-06-19 3-[2-(dimethylamino)ethyl]-N-methyl-1H-indole-5-methane-sulphonamide sulphate (2:1) HK82697A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB909026998A GB9026998D0 (en) 1990-12-12 1990-12-12 Medicaments

Publications (1)

Publication Number Publication Date
HK82697A true HK82697A (en) 1997-06-27

Family

ID=10686904

Family Applications (1)

Application Number Title Priority Date Filing Date
HK82697A HK82697A (en) 1990-12-12 1997-06-19 3-[2-(dimethylamino)ethyl]-N-methyl-1H-indole-5-methane-sulphonamide sulphate (2:1)

Country Status (36)

Country Link
US (2) US5554639A (el)
EP (1) EP0490689B1 (el)
JP (1) JP2994037B2 (el)
KR (1) KR100211479B1 (el)
CN (2) CN1030890C (el)
AP (1) AP230A (el)
AT (1) ATE119881T1 (el)
AU (1) AU650706B2 (el)
BE (1) BE1005085A3 (el)
CA (1) CA2098302C (el)
CH (1) CH684192A5 (el)
CY (1) CY2005A (el)
CZ (1) CZ281931B6 (el)
DE (1) DE69108200T2 (el)
DK (1) DK0490689T3 (el)
EG (1) EG20219A (el)
ES (1) ES2069836T3 (el)
FR (1) FR2670487B1 (el)
GB (2) GB9026998D0 (el)
GR (1) GR3015430T3 (el)
HK (1) HK82697A (el)
HU (1) HU211937A9 (el)
IE (1) IE62894B1 (el)
IL (1) IL100330A (el)
IS (1) IS1706B (el)
IT (1) IT1252868B (el)
MX (1) MX9102501A (el)
MY (1) MY109265A (el)
NL (1) NL9102071A (el)
NZ (1) NZ240942A (el)
PT (1) PT99757B (el)
RU (1) RU2108328C1 (el)
TW (2) TW300886B (el)
WO (1) WO1992010477A1 (el)
YU (1) YU48926B (el)
ZA (1) ZA919750B (el)

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US6187790B1 (en) 1999-03-04 2001-02-13 Neal R. Cutler Use of cilostazol for treatment of sexual dysfunction
US6426084B1 (en) * 2000-06-19 2002-07-30 Neal R. Cutler Treatment of sexual dysfunction in certain patient groups
US6132757A (en) * 1998-05-01 2000-10-17 Neal R. Cutler Treatment of sexual dysfunction in certain patient groups
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US6458804B1 (en) * 2001-01-26 2002-10-01 R.T. Alamo Venturesi, Llc Methods for the treatment of central nervous system disorders in certain patient groups
US6451813B1 (en) 2001-01-26 2002-09-17 R. T. Alamo Ventures I, Llc Treatment of gastroparesis in certain patient groups
US20040176359A1 (en) * 2001-02-20 2004-09-09 University Of Kentucky Research Foundation Intranasal Benzodiazepine compositions
US20030096748A1 (en) * 2001-06-04 2003-05-22 The Regents Of The University Of Michigan Methods and compositions for the treatment of diseases associated with signal transduction aberrations
DE60228294D1 (en) * 2001-06-05 2008-09-25 Ronald Aung-Din Topische migränetherapie
US8329734B2 (en) * 2009-07-27 2012-12-11 Afgin Pharma Llc Topical therapy for migraine
US7041677B2 (en) * 2002-03-01 2006-05-09 R.T. Alamo Ventures I, Llc Use of monochloroflosequinan in the treatment of sexual dysfunction
US7208628B2 (en) * 2002-05-13 2007-04-24 Kansas State University Research Foundation Compositions and methods for the treatment of hepatitis C virus infection
US7074893B2 (en) * 2002-06-03 2006-07-11 Regents Of The University Of Michigan Methods and compositions for the treatment of diseases associated with signal transduction aberrations
US20040068000A1 (en) * 2002-10-02 2004-04-08 Mintong Guo Compression coated tablets
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US20080213363A1 (en) * 2003-01-23 2008-09-04 Singh Nikhilesh N Methods and compositions for delivering 5-HT3 antagonists across the oral mucosa
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CA2529528A1 (en) 2003-06-20 2004-12-29 Ronald Aung-Din Topical therapy for the treatment of migraines, muscle sprains, muscle spasm, spasticity and related conditions
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WO2007070504A2 (en) * 2005-12-13 2007-06-21 Morton Grove Pharmaceuticals, Inc. Stable and palatable oral liquid sumatriptan compositions
US8716231B2 (en) 2005-12-19 2014-05-06 Janssen Pharmaceutica Nv Use of benzo-fused heterocycle sulfamide derivatives for the treatment of pain
US8937096B2 (en) 2005-12-19 2015-01-20 Janssen Pharmaceutica Nv Use of benzo-fused heterocyle sulfamide derivatives for the treatment of mania and bipolar disorder
AR058389A1 (es) 2005-12-19 2008-01-30 Janssen Pharmaceutica Nv Uso de derivados heterociclicos benzo-fusionados de sulfamida para el tratamiento de la obesidad
US8691867B2 (en) 2005-12-19 2014-04-08 Janssen Pharmaceutica Nv Use of benzo-fused heterocycle sulfamide derivatives for the treatment of substance abuse and addiction
US8497298B2 (en) 2005-12-19 2013-07-30 Janssen Pharmaceutica Nv Use of benzo-fused heterocycle sulfamide derivatives for lowering lipids and lowering blood glucose levels
US20070191461A1 (en) * 2006-02-15 2007-08-16 Smith-Swintosky Virginia L Use of benzo-heteroaryl sulfamide derivatives for the treatment of migraine
JP2009537635A (ja) 2006-05-19 2009-10-29 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ 癲癇の処置のための共同−療法
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US20080275030A1 (en) 2007-01-19 2008-11-06 Sveinbjorn Gizurarson Methods and Compositions for the Delivery of a Therapeutic Agent
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US20090252791A1 (en) * 2008-04-02 2009-10-08 Venkata Nookaraju Sreedharala Pharmaceutical compositions comprising a triptan and a nonsteroidal anti-inflammatory drug
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US11337962B2 (en) 2009-09-25 2022-05-24 Upsher-Smith Laboratories, Llc Formulations comprising triptan compounds
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US10383816B2 (en) 2015-03-02 2019-08-20 Afgin Pharma, Llc Topical regional neuro-affective therapy with cannabinoid combination products
CN107530318A (zh) 2015-03-02 2018-01-02 阿福金制药有限责任公司 用大麻素的局部区域神经影响性疗法
JP6897971B2 (ja) 2015-05-15 2021-07-07 ザ リージェンツ オブ ザ ユニバーシティ オブ ミシガン 関節炎を処置するための、方法および組成物
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US20180049994A1 (en) 2016-08-16 2018-02-22 Afgin Pharma, Llc Topical regional neuro-affective therapy with caryophyllene
KR20200085278A (ko) 2017-11-07 2020-07-14 더 리젠츠 오브 더 유니버시티 오브 미시건 공유 에피토프-칼레티쿨린 상호 작용의 소분자 억제제　및 사용 방법
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US11364225B2 (en) * 2019-08-21 2022-06-21 Bn Intellectual Properties, Inc. Pharmaceutical formulation for treating symptoms of migraine and cluster headaches, and method of using the same
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GB8928208D0 (en) * 1989-12-13 1990-02-14 Glaxo Group Ltd Medicaments

Also Published As

Publication number Publication date
IS3790A7 (is) 1992-06-13
PT99757B (pt) 1999-05-31
GB9126297D0 (en) 1992-02-12
ES2069836T3 (es) 1995-05-16
JPH06503560A (ja) 1994-04-21
HU211937A9 (en) 1996-01-29
ZA919750B (en) 1992-10-28
GB2251614B (en) 1994-12-14
IE62894B1 (en) 1995-03-08
TW205035B (el) 1993-05-01
NL9102071A (nl) 1992-07-01
IT1252868B (it) 1995-06-28
YU191491A (sh) 1994-04-05
TW300886B (el) 1997-03-21
YU48926B (sh) 2002-12-10
PT99757A (pt) 1992-12-31
ITRM910922A0 (it) 1991-12-11
AP230A (en) 1993-01-27
FR2670487B1 (fr) 1993-08-20
CN1128259A (zh) 1996-08-07
WO1992010477A1 (en) 1992-06-25
IL100330A (en) 1996-06-18
CN1050831C (zh) 2000-03-29
CN1063099A (zh) 1992-07-29
GB2251614A (en) 1992-07-15
IS1706B (is) 1998-12-10
IE914317A1 (en) 1992-06-17
EP0490689A1 (en) 1992-06-17
CZ281931B6 (cs) 1997-04-16
EP0490689B1 (en) 1995-03-15
MX9102501A (es) 1992-09-01
ITRM910922A1 (it) 1993-06-11
KR100211479B1 (ko) 1999-08-02
CA2098302C (en) 2001-10-16
AU650706B2 (en) 1994-06-30
CY2005A (en) 1997-12-05
CA2098302A1 (en) 1992-06-13
US5705520A (en) 1998-01-06
ATE119881T1 (de) 1995-04-15
AU9072091A (en) 1992-07-08
GR3015430T3 (en) 1995-06-30
BE1005085A3 (fr) 1993-04-13
MY109265A (en) 1996-12-31
NZ240942A (en) 1994-03-25
CH684192A5 (fr) 1994-07-29
CZ114093A3 (en) 1994-02-16
DE69108200T2 (de) 1995-07-20
RU2108328C1 (ru) 1998-04-10
AP9100339A0 (en) 1992-01-31
CN1030890C (zh) 1996-02-07
EG20219A (en) 1997-11-30
DE69108200D1 (de) 1995-04-20
GB9026998D0 (en) 1991-01-30
IL100330A0 (en) 1992-09-06
DK0490689T3 (da) 1995-05-22
US5554639A (en) 1996-09-10
JP2994037B2 (ja) 1999-12-27
FR2670487A1 (fr) 1992-06-19

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Legal Events

Date Code Title Description
PF Patent in force
PC Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee)

Effective date: 20091212