HK52580A - 3-amino-indazolecarboxylic acid derivatives,process for their preparation and their use as medicaments - Google Patents

3-amino-indazolecarboxylic acid derivatives,process for their preparation and their use as medicaments

Info

Publication number
HK52580A
HK52580A HK525/80A HK52580A HK52580A HK 52580 A HK52580 A HK 52580A HK 525/80 A HK525/80 A HK 525/80A HK 52580 A HK52580 A HK 52580A HK 52580 A HK52580 A HK 52580A
Authority
HK
Hong Kong
Prior art keywords
medicaments
amino
preparation
acid derivatives
indazolecarboxylic acid
Prior art date
Application number
HK525/80A
Other languages
English (en)
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of HK52580A publication Critical patent/HK52580A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56Benzopyrazoles; Hydrogenated benzopyrazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
HK525/80A 1974-12-13 1980-09-18 3-amino-indazolecarboxylic acid derivatives,process for their preparation and their use as medicaments HK52580A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE2458965A DE2458965C3 (de) 1974-12-13 1974-12-13 3-Amino-indazol-N-carbonsäure-Derivate, Verfahren zu ihrer Herstellung sowie sie enthaltende Arzneimittel

Publications (1)

Publication Number Publication Date
HK52580A true HK52580A (en) 1980-09-26

Family

ID=5933305

Family Applications (1)

Application Number Title Priority Date Filing Date
HK525/80A HK52580A (en) 1974-12-13 1980-09-18 3-amino-indazolecarboxylic acid derivatives,process for their preparation and their use as medicaments

Country Status (27)

Country Link
US (1) US4051252A (forum.php)
JP (1) JPS5182266A (forum.php)
AT (1) AT343653B (forum.php)
BE (1) BE836528A (forum.php)
CA (1) CA1059523A (forum.php)
CH (1) CH622250A5 (forum.php)
CS (1) CS189731B2 (forum.php)
DD (1) DD125484A5 (forum.php)
DE (1) DE2458965C3 (forum.php)
DK (1) DK137082C (forum.php)
ES (1) ES443429A1 (forum.php)
FI (1) FI753493A7 (forum.php)
FR (1) FR2293928A1 (forum.php)
GB (1) GB1490306A (forum.php)
HK (1) HK52580A (forum.php)
HU (1) HU173557B (forum.php)
IE (1) IE42208B1 (forum.php)
IL (1) IL48642A (forum.php)
KE (1) KE3078A (forum.php)
LU (1) LU73993A1 (forum.php)
NL (1) NL7514521A (forum.php)
NO (1) NO145382C (forum.php)
PL (1) PL99858B1 (forum.php)
SE (1) SE419645B (forum.php)
SU (1) SU604487A3 (forum.php)
YU (1) YU315275A (forum.php)
ZA (1) ZA757777B (forum.php)

Families Citing this family (39)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4431657A (en) * 1982-05-24 1984-02-14 Ayerst, Mckenna & Harrison Inc. Analgesic compositions consisting of 2H-benzothieno[3,2-c]pyrazol-3-amine derivatives
KR20010086657A (ko) * 2000-03-02 2001-09-15 성재갑 아미노인다졸 유도체 및 이를 함유하는 싸이클린 의존키나아제 저해제 조성물
NZ525014A (en) * 2000-09-15 2005-09-30 Vertex Pharma Pyrazole compounds useful as protein kinase inhibitors
ZA200301701B (en) * 2000-09-15 2004-03-01 Vertex Pharma Pyrazole compounds useful as protein kinase inhibitors.
SI1318997T1 (sl) * 2000-09-15 2006-12-31 Vertex Pharma Pirazolne spojine, uporabne kot inhibitorji protein-kinaze
US6660731B2 (en) 2000-09-15 2003-12-09 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
US7473691B2 (en) * 2000-09-15 2009-01-06 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
WO2002057259A2 (en) 2000-12-21 2002-07-25 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
KR100406634B1 (ko) * 2001-03-12 2003-11-20 주식회사 엘지생명과학 3,5-디아미노인다졸 유도체, 그의 제조방법 및 사이클린의존성 키나아제 저해제로서의 그의 용도
CA2460145C (en) 2001-09-26 2011-04-26 Pharmacia Italia S.P.A. Aminoindazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions containing them
EP1472245A2 (en) * 2002-02-06 2004-11-03 Vertex Pharmaceuticals Incorporated Heteroaryl compounds useful as inhibitors of gsk-3
FR2836915B1 (fr) * 2002-03-11 2008-01-11 Aventis Pharma Sa Derives d'aminoindazoles, procede de preparation et intermediaires de ce procede a titre de medicaments et compositions pharmaceutiques les renfermant
DE60332604D1 (de) 2002-03-15 2010-07-01 Vertex Pharma Azolylaminoazine als proteinkinasehemmer
AU2003227741A1 (en) 2002-05-17 2003-12-02 Pharmacia Italia S.P.A. Aminoindazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them
MY141867A (en) * 2002-06-20 2010-07-16 Vertex Pharma Substituted pyrimidines useful as protein kinase inhibitors
DK1532145T3 (da) 2002-08-02 2007-01-15 Vertex Pharma Pyrazolpræparater der er anvendelige som inhibitorer af GSK-3
WO2004041285A1 (en) * 2002-10-31 2004-05-21 Amgen Inc. Antiinflammation agents
US7601718B2 (en) 2003-02-06 2009-10-13 Vertex Pharmaceuticals Incorporated Compositions useful as inhibitors of protein kinases
US7592340B2 (en) * 2003-12-04 2009-09-22 Vertex Pharmaceuticals Incorporated Quinoxalines useful as inhibitors of protein kinases
DE102004005172A1 (de) * 2004-02-02 2005-08-18 Aventis Pharma Deutschland Gmbh Indazolderivate als Inhibitoren der Hormon Sensitiven Lipase
WO2007022384A2 (en) 2005-08-18 2007-02-22 Vertex Pharmaceuticals Incorporated Pyrazine kinase inhibitors
SG166828A1 (en) * 2005-11-03 2010-12-29 Vertex Pharma Aminopyrimidines useful as kinase inhibitors
AU2007238019B2 (en) * 2006-04-14 2013-03-14 Abbvie Inc. Process for the preparation of indazolyl ureas that inhibit vanilloid subtype 1 (VR1) receptors
MX2009004807A (es) 2006-11-02 2009-06-15 Vertex Pharma Aminopiridinas y aminopirimidinas utiles como inhibidores de proteina cinasa.
CA2673353A1 (en) 2006-12-19 2008-06-26 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as inhibitors of protein kinases
ATE526328T1 (de) 2007-03-09 2011-10-15 Vertex Pharma Als inhibitoren von proteinkinasen geeignete aminopyrimidine
EP2134709A1 (en) 2007-03-09 2009-12-23 Vertex Pharmaceuticals, Inc. Aminopyridines useful as inhibitors of protein kinases
MX2009009590A (es) 2007-03-09 2009-11-10 Vertex Pharma Aminopirimidinas utiles como inhibidores de proteinas cinasas.
MX2009011059A (es) 2007-04-13 2009-11-26 Vertex Pharma Aminopirimidinas utiles como inhibidores de cinasas.
JP5572087B2 (ja) * 2007-05-02 2014-08-13 バーテックス ファーマシューティカルズ インコーポレイテッド キナーゼ阻害として有用なアミノピリミジン
CA2694381A1 (en) 2007-05-02 2008-11-13 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as kinase inhibitors
CA2685876A1 (en) * 2007-05-02 2008-11-13 Vertex Pharmaceuticals Incorporated Thiazoles and pyrazoles useful as kinase inhibitors
AU2008257044A1 (en) * 2007-05-24 2008-12-04 Vertex Pharmaceuticals Incorporated Thiazoles and pyrazoles useful as kinase inhibitors
MX2010001137A (es) * 2007-07-31 2010-03-31 Vertex Pharma Procesopara preparar 5-fluoro-1h-pirazol[3,4-b]piridin-3-amina y derivados del mismo.
RU2011112802A (ru) * 2008-09-03 2012-10-10 Вертекс Фармасьютикалз Инкорпорейтед (Us) Сокристаллы и содержащие их фармацевтические композиции
DE102009004245A1 (de) 2009-01-09 2010-07-15 Bayer Schering Pharma Aktiengesellschaft Neue anellierte, Heteroatom-verbrückte Pyrazol- und Imidazol-Derivate und ihre Verwendung
JP6317345B2 (ja) 2012-07-24 2018-04-25 ビアル−ポルテラ エ コンパニア,ソシエダッド アノニマ ウレア化合物および酵素阻害剤としてのそれらの使用
CA2880299A1 (en) * 2012-07-27 2014-01-30 Bial - Portela & Ca, S.A. Process for the synthesis of substituted urea compounds
AU2014293731B2 (en) 2013-07-24 2018-03-08 Bial - Portela & Ca, S.A. Imidazolecarboxamides and their use as FAAH inhibitors

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3133081A (en) * 1964-05-12 J-aminoindazole derivatives
CH397698A (de) * 1961-09-08 1965-08-31 Siegfried Ag Verfahren zur Herstellung neuer 1-Carbamyl-indazole
US3274203A (en) * 1963-05-31 1966-09-20 Du Pont 1-carbamyl and thiocarbamyl-3-amino-4-nonsubstituted and substituted pyrazoles
NL6707299A (forum.php) * 1966-07-16 1968-01-17
DE1770649A1 (de) * 1968-06-15 1971-11-11 Bayer Ag Substituierte 3-Amino-indazole

Also Published As

Publication number Publication date
SE7513990L (sv) 1976-06-14
SE419645B (sv) 1981-08-17
AT343653B (de) 1978-06-12
DK137082B (da) 1978-01-16
ATA939775A (de) 1977-10-15
PL99858B1 (pl) 1978-08-31
US4051252A (en) 1977-09-27
CS189731B2 (en) 1979-04-30
NO145382B (no) 1981-11-30
AU8717075A (en) 1977-06-09
ZA757777B (en) 1976-11-24
FR2293928B1 (forum.php) 1979-09-21
DE2458965A1 (de) 1976-06-16
DK567275A (da) 1976-06-14
IL48642A (en) 1979-12-30
FR2293928A1 (fr) 1976-07-09
IE42208B1 (en) 1980-06-18
NO754024L (forum.php) 1976-06-15
SU604487A3 (ru) 1978-04-25
NL7514521A (nl) 1976-06-15
CH622250A5 (forum.php) 1981-03-31
YU315275A (en) 1982-02-28
IE42208L (en) 1976-06-13
GB1490306A (en) 1977-11-02
BE836528A (fr) 1976-06-11
JPS5182266A (en) 1976-07-19
HU173557B (hu) 1979-06-28
ES443429A1 (es) 1977-04-16
DE2458965B2 (de) 1979-02-22
IL48642A0 (en) 1976-02-29
DK137082C (da) 1978-06-19
KE3078A (en) 1980-10-03
DE2458965C3 (de) 1979-10-11
LU73993A1 (forum.php) 1976-11-11
FI753493A7 (forum.php) 1976-06-14
CA1059523A (en) 1979-07-31
DD125484A5 (forum.php) 1977-04-20
NO145382C (no) 1982-03-10

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