HK1192240A1 - 具有噁唑並 嘧啶環的羧酸衍生物 - Google Patents
具有噁唑並 嘧啶環的羧酸衍生物Info
- Publication number
- HK1192240A1 HK1192240A1 HK14105592.5A HK14105592A HK1192240A1 HK 1192240 A1 HK1192240 A1 HK 1192240A1 HK 14105592 A HK14105592 A HK 14105592A HK 1192240 A1 HK1192240 A1 HK 1192240A1
- Authority
- HK
- Hong Kong
- Prior art keywords
- oxazolo
- carboxylic acid
- acid derivatives
- pyrimidine ring
- pyrimidine
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Cardiology (AREA)
- Diabetes (AREA)
- Heart & Thoracic Surgery (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Endocrinology (AREA)
- Hospice & Palliative Care (AREA)
- Emergency Medicine (AREA)
- Dermatology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP11305878 | 2011-07-07 | ||
| EP12305526 | 2012-05-11 | ||
| PCT/EP2012/063298 WO2013004827A1 (de) | 2011-07-07 | 2012-07-06 | Carbonsäurederivate mit einem Oxazolo[5,4-d]Pyrimidinring |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| HK1192240A1 true HK1192240A1 (zh) | 2014-08-15 |
Family
ID=46458547
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HK14105592.5A HK1192240A1 (zh) | 2011-07-07 | 2014-06-13 | 具有噁唑並 嘧啶環的羧酸衍生物 |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US9321787B2 (zh) |
| EP (1) | EP2729471B1 (zh) |
| JP (1) | JP5913585B2 (zh) |
| KR (1) | KR20140061385A (zh) |
| CN (1) | CN103781792B (zh) |
| AU (1) | AU2012280207B2 (zh) |
| BR (1) | BR112014000118A2 (zh) |
| CA (1) | CA2841226C (zh) |
| DK (1) | DK2729471T3 (zh) |
| ES (1) | ES2544620T3 (zh) |
| HK (1) | HK1192240A1 (zh) |
| IL (1) | IL230258A (zh) |
| MX (1) | MX365934B (zh) |
| MY (1) | MY164134A (zh) |
| PT (1) | PT2729471E (zh) |
| RU (1) | RU2609008C2 (zh) |
| WO (1) | WO2013004827A1 (zh) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US9321787B2 (en) | 2011-07-07 | 2016-04-26 | Sanofi | Carboxylic acid derivatives having an oxazolo[5,4-d]pyrimidine ring |
| CN103992279B (zh) * | 2014-06-06 | 2016-06-01 | 重庆华邦胜凯制药有限公司 | 一种制备硫代巴比妥酸化合物的方法 |
| JP6661885B2 (ja) * | 2015-03-09 | 2020-03-11 | セイコーエプソン株式会社 | 画像表示装置 |
Family Cites Families (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3679682A (en) * | 1970-04-23 | 1972-07-25 | Fmc Corp | CERTAIN 5H-ISOXAZOLO{8 5,4-d{9 PYRIMIDIN-4-ONES |
| WO2000021572A2 (en) * | 1998-10-09 | 2000-04-20 | The University Of Michigan | Hydrogels and water soluble polymeric carriers for drug delivery |
| JP2003508127A (ja) * | 1999-08-27 | 2003-03-04 | デパートメント オブ ナショナル ディフェンス | リポソームで被包された治療薬を含むヒドロゲル傷被覆用品 |
| DE102005018389A1 (de) * | 2005-04-20 | 2006-10-26 | Sanofi-Aventis Deutschland Gmbh | Azolderivate als Inhibitoren von Lipasen und Phospholipasen |
| DE602006005242D1 (de) * | 2005-06-27 | 2009-04-02 | Sanofi Aventis | Pyrazolopyridinderivate als inhibitoren der kinase 1 des beta-adrenergen rezeptors |
| EP1964840A1 (en) * | 2007-02-28 | 2008-09-03 | sanofi-aventis | Imidazo[1,2-a]pyridines and their use as pharmaceuticals |
| WO2009155017A2 (en) * | 2008-05-30 | 2009-12-23 | Merck & Co., Inc. | Novel substituted azabenzoxazoles |
| TW201000099A (en) | 2008-06-20 | 2010-01-01 | Amgen Inc | S1P1 receptor agonists and use thereof |
| AU2009270511B2 (en) | 2008-07-15 | 2013-07-18 | Sanofi | Oxazolopyrimidines as Edg-1 receptor agonists |
| AR079981A1 (es) | 2010-01-13 | 2012-03-07 | Sanofi Aventis | Derivados de acido carboxilico que comprenden un anillo de oxoazolopirimidina 2,5,7- sustituido |
| AR079982A1 (es) | 2010-01-13 | 2012-03-07 | Sanofi Aventis | Derivados de acido carboxilico heterociclicos que comprenden un anillo de oxazolopirimidina 2,5,7- sustituido., composiciones farmaceuticas y procesos para prepararlos. |
| TWI485153B (zh) | 2010-01-13 | 2015-05-21 | Sanofi Aventis | ２，５，７－經取代唑并嘧啶衍生物 |
| BR112012017437B1 (pt) * | 2010-01-14 | 2022-03-03 | Sanofi | Compostos derivados de ácido carboxílicotendo um anel de oxazolopirimidina 2,5- substituído, seu processo de preparação e composição farmacêutica que os compreende |
| BR112012017484A2 (pt) | 2010-01-14 | 2020-08-25 | Sanofi | "derivados de oxazolopirimidina 2,5-substituídos" |
| UY33180A (es) | 2010-01-14 | 2011-08-31 | Sanofi Aventis | Derivados de ácido carboxílico heterocíclicos que comprenden un anillo de oxazolopirimidina 2,5-sustituida. |
| US8580816B2 (en) | 2011-07-07 | 2013-11-12 | Sanofi | Carboxylic acid derivatives having an oxazolo[5,4-b]pyridine ring |
| US9321787B2 (en) | 2011-07-07 | 2016-04-26 | Sanofi | Carboxylic acid derivatives having an oxazolo[5,4-d]pyrimidine ring |
| US8735402B2 (en) | 2011-07-07 | 2014-05-27 | Sanofi | Cycloalkyloxycarboxylic acid derivatives |
| US8907093B2 (en) | 2011-07-07 | 2014-12-09 | Sanofi | Carboxylic acid derivatives having an oxazolo[4,5-c]pyridine ring |
-
2012
- 2012-06-25 US US13/532,292 patent/US9321787B2/en active Active
- 2012-07-06 MX MX2014000022A patent/MX365934B/es active IP Right Grant
- 2012-07-06 DK DK12732677.5T patent/DK2729471T3/en active
- 2012-07-06 KR KR1020147003227A patent/KR20140061385A/ko not_active Application Discontinuation
- 2012-07-06 EP EP12732677.5A patent/EP2729471B1/de active Active
- 2012-07-06 CN CN201280043698.4A patent/CN103781792B/zh active Active
- 2012-07-06 ES ES12732677.5T patent/ES2544620T3/es active Active
- 2012-07-06 BR BR112014000118A patent/BR112014000118A2/pt not_active IP Right Cessation
- 2012-07-06 WO PCT/EP2012/063298 patent/WO2013004827A1/de active Application Filing
- 2012-07-06 PT PT127326775T patent/PT2729471E/pt unknown
- 2012-07-06 RU RU2014104230A patent/RU2609008C2/ru not_active IP Right Cessation
- 2012-07-06 JP JP2014517830A patent/JP5913585B2/ja active Active
- 2012-07-06 CA CA2841226A patent/CA2841226C/en not_active Expired - Fee Related
- 2012-07-06 MY MYPI2014000007A patent/MY164134A/en unknown
- 2012-07-06 AU AU2012280207A patent/AU2012280207B2/en not_active Ceased
-
2013
- 2013-12-31 IL IL230258A patent/IL230258A/en not_active IP Right Cessation
-
2014
- 2014-06-13 HK HK14105592.5A patent/HK1192240A1/zh not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| ES2544620T3 (es) | 2015-09-02 |
| WO2013004827A1 (de) | 2013-01-10 |
| BR112014000118A2 (pt) | 2017-01-10 |
| RU2014104230A (ru) | 2015-08-20 |
| IL230258A (en) | 2016-08-31 |
| EP2729471A1 (de) | 2014-05-14 |
| DK2729471T3 (en) | 2015-08-10 |
| US20130023544A1 (en) | 2013-01-24 |
| CN103781792B (zh) | 2016-06-29 |
| KR20140061385A (ko) | 2014-05-21 |
| MX365934B (es) | 2019-06-20 |
| MX2014000022A (es) | 2014-02-19 |
| AU2012280207A1 (en) | 2014-01-23 |
| MY164134A (en) | 2017-11-30 |
| CA2841226C (en) | 2019-11-12 |
| AU2012280207B2 (en) | 2017-03-09 |
| CN103781792A (zh) | 2014-05-07 |
| US9321787B2 (en) | 2016-04-26 |
| PT2729471E (pt) | 2015-09-16 |
| JP2014518248A (ja) | 2014-07-28 |
| JP5913585B2 (ja) | 2016-04-27 |
| RU2609008C2 (ru) | 2017-01-30 |
| EP2729471B1 (de) | 2015-05-06 |
| CA2841226A1 (en) | 2013-01-10 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PC | Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee) |
Effective date: 20190704 |