HK1192240A1 - Carboxylic acid derivatives with an oxazolo[5,4-d]pyrimidine ring [54-d] - Google Patents
Carboxylic acid derivatives with an oxazolo[5,4-d]pyrimidine ring [54-d]Info
- Publication number
- HK1192240A1 HK1192240A1 HK14105592.5A HK14105592A HK1192240A1 HK 1192240 A1 HK1192240 A1 HK 1192240A1 HK 14105592 A HK14105592 A HK 14105592A HK 1192240 A1 HK1192240 A1 HK 1192240A1
- Authority
- HK
- Hong Kong
- Prior art keywords
- oxazolo
- carboxylic acid
- acid derivatives
- pyrimidine ring
- pyrimidine
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Diabetes (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Endocrinology (AREA)
- Emergency Medicine (AREA)
- Hospice & Palliative Care (AREA)
- Dermatology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP11305878 | 2011-07-07 | ||
| EP12305526 | 2012-05-11 | ||
| PCT/EP2012/063298 WO2013004827A1 (de) | 2011-07-07 | 2012-07-06 | Carbonsäurederivate mit einem Oxazolo[5,4-d]Pyrimidinring |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| HK1192240A1 true HK1192240A1 (en) | 2014-08-15 |
Family
ID=46458547
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HK14105592.5A HK1192240A1 (en) | 2011-07-07 | 2014-06-13 | Carboxylic acid derivatives with an oxazolo[5,4-d]pyrimidine ring [54-d] |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US9321787B2 (xx) |
| EP (1) | EP2729471B1 (xx) |
| JP (1) | JP5913585B2 (xx) |
| KR (1) | KR20140061385A (xx) |
| CN (1) | CN103781792B (xx) |
| AU (1) | AU2012280207B2 (xx) |
| BR (1) | BR112014000118A2 (xx) |
| CA (1) | CA2841226C (xx) |
| DK (1) | DK2729471T3 (xx) |
| ES (1) | ES2544620T3 (xx) |
| HK (1) | HK1192240A1 (xx) |
| IL (1) | IL230258A (xx) |
| MX (1) | MX365934B (xx) |
| MY (1) | MY164134A (xx) |
| PT (1) | PT2729471E (xx) |
| RU (1) | RU2609008C2 (xx) |
| WO (1) | WO2013004827A1 (xx) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US9321787B2 (en) | 2011-07-07 | 2016-04-26 | Sanofi | Carboxylic acid derivatives having an oxazolo[5,4-d]pyrimidine ring |
| CN103992279B (zh) * | 2014-06-06 | 2016-06-01 | 重庆华邦胜凯制药有限公司 | 一种制备硫代巴比妥酸化合物的方法 |
| JP6661885B2 (ja) * | 2015-03-09 | 2020-03-11 | セイコーエプソン株式会社 | 画像表示装置 |
Family Cites Families (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3679682A (en) * | 1970-04-23 | 1972-07-25 | Fmc Corp | CERTAIN 5H-ISOXAZOLO{8 5,4-d{9 PYRIMIDIN-4-ONES |
| AU6419899A (en) * | 1998-10-09 | 2000-05-01 | Regents Of The University Of Michigan, The | Hydrogels and water soluble polymeric carriers for drug delivery |
| AU6679400A (en) * | 1999-08-27 | 2001-03-26 | Department Of National Defence | Hydrogel wound dressing containing liposome-encapsulated therapeutic agent |
| DE102005018389A1 (de) * | 2005-04-20 | 2006-10-26 | Sanofi-Aventis Deutschland Gmbh | Azolderivate als Inhibitoren von Lipasen und Phospholipasen |
| SI1899333T1 (sl) * | 2005-06-27 | 2009-08-31 | Sanofi Aventis | Pirazolopiridinski derivati kot inhibitorji kinaze 1 betaadrenergičnega receptorja |
| EP1964840A1 (en) * | 2007-02-28 | 2008-09-03 | sanofi-aventis | Imidazo[1,2-a]pyridines and their use as pharmaceuticals |
| EP2300481B1 (en) * | 2008-05-30 | 2015-09-30 | Merck Sharp & Dohme Corp. | Novel substituted azabenzoxazoles |
| TW201000099A (en) | 2008-06-20 | 2010-01-01 | Amgen Inc | S1P1 receptor agonists and use thereof |
| AU2009270511B2 (en) | 2008-07-15 | 2013-07-18 | Sanofi | Oxazolopyrimidines as Edg-1 receptor agonists |
| TWI478929B (zh) | 2010-01-13 | 2015-04-01 | Sanofi Aventis | 含２，５，７－經取代唑并嘧啶環之羧酸衍生物 |
| TWI517851B (zh) | 2010-01-13 | 2016-01-21 | 賽諾菲阿凡提斯公司 | 含２，５，７－經取代唑并嘧啶環之雜環羧酸衍生物 |
| UY33176A (es) | 2010-01-13 | 2011-08-31 | Sanofi Aventis | Derivados de oxazolopirimidina sustituida en 2, 5, 7. |
| WO2011086081A1 (de) | 2010-01-14 | 2011-07-21 | Sanofi-Aventis | 2,5-substituierte oxazolopyrimidinderivate |
| AR079997A1 (es) * | 2010-01-14 | 2012-03-07 | Sanofi Aventis | Derivados de acido carboxilico de oxazolo[5,4-d]pirimidinas utiles en el tratamiento del sindrome del pie diabetico(dfs), composiciones farmaceuticas que los contienen y metodo de preparacion de los mismos. |
| JP5841068B2 (ja) | 2010-01-14 | 2016-01-06 | サノフイ | ２，５−置換されたオキサゾロピリミジン環を有する複素環式カルボン酸誘導体 |
| US8735402B2 (en) | 2011-07-07 | 2014-05-27 | Sanofi | Cycloalkyloxycarboxylic acid derivatives |
| US8907093B2 (en) * | 2011-07-07 | 2014-12-09 | Sanofi | Carboxylic acid derivatives having an oxazolo[4,5-c]pyridine ring |
| US9321787B2 (en) | 2011-07-07 | 2016-04-26 | Sanofi | Carboxylic acid derivatives having an oxazolo[5,4-d]pyrimidine ring |
| US8580816B2 (en) | 2011-07-07 | 2013-11-12 | Sanofi | Carboxylic acid derivatives having an oxazolo[5,4-b]pyridine ring |
-
2012
- 2012-06-25 US US13/532,292 patent/US9321787B2/en active Active
- 2012-07-06 MX MX2014000022A patent/MX365934B/es active IP Right Grant
- 2012-07-06 RU RU2014104230A patent/RU2609008C2/ru not_active IP Right Cessation
- 2012-07-06 MY MYPI2014000007A patent/MY164134A/en unknown
- 2012-07-06 DK DK12732677.5T patent/DK2729471T3/en active
- 2012-07-06 WO PCT/EP2012/063298 patent/WO2013004827A1/de active Application Filing
- 2012-07-06 KR KR1020147003227A patent/KR20140061385A/ko not_active Application Discontinuation
- 2012-07-06 CA CA2841226A patent/CA2841226C/en not_active Expired - Fee Related
- 2012-07-06 AU AU2012280207A patent/AU2012280207B2/en not_active Ceased
- 2012-07-06 BR BR112014000118A patent/BR112014000118A2/pt not_active IP Right Cessation
- 2012-07-06 PT PT127326775T patent/PT2729471E/pt unknown
- 2012-07-06 CN CN201280043698.4A patent/CN103781792B/zh active Active
- 2012-07-06 EP EP12732677.5A patent/EP2729471B1/de active Active
- 2012-07-06 JP JP2014517830A patent/JP5913585B2/ja active Active
- 2012-07-06 ES ES12732677.5T patent/ES2544620T3/es active Active
-
2013
- 2013-12-31 IL IL230258A patent/IL230258A/en not_active IP Right Cessation
-
2014
- 2014-06-13 HK HK14105592.5A patent/HK1192240A1/xx not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| PT2729471E (pt) | 2015-09-16 |
| DK2729471T3 (en) | 2015-08-10 |
| AU2012280207B2 (en) | 2017-03-09 |
| IL230258A (en) | 2016-08-31 |
| JP5913585B2 (ja) | 2016-04-27 |
| CN103781792B (zh) | 2016-06-29 |
| MY164134A (en) | 2017-11-30 |
| CN103781792A (zh) | 2014-05-07 |
| RU2014104230A (ru) | 2015-08-20 |
| BR112014000118A2 (pt) | 2017-01-10 |
| WO2013004827A1 (de) | 2013-01-10 |
| MX365934B (es) | 2019-06-20 |
| MX2014000022A (es) | 2014-02-19 |
| JP2014518248A (ja) | 2014-07-28 |
| EP2729471A1 (de) | 2014-05-14 |
| KR20140061385A (ko) | 2014-05-21 |
| US20130023544A1 (en) | 2013-01-24 |
| RU2609008C2 (ru) | 2017-01-30 |
| ES2544620T3 (es) | 2015-09-02 |
| US9321787B2 (en) | 2016-04-26 |
| EP2729471B1 (de) | 2015-05-06 |
| CA2841226A1 (en) | 2013-01-10 |
| CA2841226C (en) | 2019-11-12 |
| AU2012280207A1 (en) | 2014-01-23 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PC | Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee) |
Effective date: 20190704 |