HK1166978A1 - 噁二唑衍生物配體及其作為親代謝性谷氨酸受體 增效劑的用途 - Google Patents
噁二唑衍生物配體及其作為親代謝性谷氨酸受體 增效劑的用途Info
- Publication number
- HK1166978A1 HK1166978A1 HK12106999.4A HK12106999A HK1166978A1 HK 1166978 A1 HK1166978 A1 HK 1166978A1 HK 12106999 A HK12106999 A HK 12106999A HK 1166978 A1 HK1166978 A1 HK 1166978A1
- Authority
- HK
- Hong Kong
- Prior art keywords
- potentiators
- glutamate receptor
- metabotropic glutamate
- oxadiazole derivatives
- oxadiazole
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
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-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/08—Bridged systems
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US94255307P | 2007-06-07 | 2007-06-07 |
Publications (1)
Publication Number | Publication Date |
---|---|
HK1166978A1 true HK1166978A1 (zh) | 2012-11-16 |
Family
ID=40093925
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HK10108742.2A HK1142318A1 (en) | 2007-06-07 | 2010-09-15 | Oxadiazole derivatives and their use as metabotropic glutamate receptor potentiators - 842 |
HK12106999.4A HK1166978A1 (zh) | 2007-06-07 | 2010-09-15 | 噁二唑衍生物配體及其作為親代謝性谷氨酸受體 增效劑的用途 |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HK10108742.2A HK1142318A1 (en) | 2007-06-07 | 2010-09-15 | Oxadiazole derivatives and their use as metabotropic glutamate receptor potentiators - 842 |
Country Status (34)
Country | Link |
---|---|
US (2) | US8377940B2 (zh) |
EP (2) | EP2167502B3 (zh) |
JP (2) | JP5416696B2 (zh) |
KR (2) | KR20100017640A (zh) |
CN (2) | CN102977086B (zh) |
AR (1) | AR066882A1 (zh) |
AU (1) | AU2008260717B2 (zh) |
BR (1) | BRPI0812889A2 (zh) |
CA (1) | CA2690856C (zh) |
CL (1) | CL2008001667A1 (zh) |
CO (1) | CO6251287A2 (zh) |
CY (2) | CY1113422T1 (zh) |
DK (2) | DK2444399T3 (zh) |
EC (1) | ECSP109856A (zh) |
ES (2) | ES2393425T7 (zh) |
HK (2) | HK1142318A1 (zh) |
HR (2) | HRP20120909T4 (zh) |
IL (1) | IL202158A (zh) |
ME (1) | ME01488B (zh) |
MX (1) | MX2009013078A (zh) |
MY (1) | MY158066A (zh) |
NZ (1) | NZ582445A (zh) |
PE (1) | PE20090328A1 (zh) |
PL (2) | PL2167502T6 (zh) |
PT (2) | PT2167502E (zh) |
RS (2) | RS53845B1 (zh) |
RU (2) | RU2470931C2 (zh) |
SA (1) | SA08290344B1 (zh) |
SI (2) | SI2444399T1 (zh) |
TW (1) | TWI417100B (zh) |
UA (1) | UA99129C2 (zh) |
UY (1) | UY31124A1 (zh) |
WO (1) | WO2008150233A1 (zh) |
ZA (1) | ZA200908285B (zh) |
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TW200804281A (en) * | 2006-02-16 | 2008-01-16 | Astrazeneca Ab | New metabotropic glutamate receptor-potentiating isoindolones |
AR059898A1 (es) | 2006-03-15 | 2008-05-07 | Janssen Pharmaceutica Nv | Derivados de 3-ciano-piridona 1,4-disustituida y su uso como moduladores alostericos de los receptores mglur2 |
TW200845978A (en) | 2007-03-07 | 2008-12-01 | Janssen Pharmaceutica Nv | 3-cyano-4-(4-tetrahydropyran-phenyl)-pyridin-2-one derivatives |
TW200900065A (en) | 2007-03-07 | 2009-01-01 | Janssen Pharmaceutica Nv | 3-cyano-4-(4-pyridinyloxy-phenyl)-pyridin-2-one derivatives |
TWI417100B (zh) | 2007-06-07 | 2013-12-01 | Astrazeneca Ab | 二唑衍生物及其作為代謝型麩胺酸受體增效劑-842之用途 |
TW200911255A (en) | 2007-06-07 | 2009-03-16 | Astrazeneca Ab | Metabotropic glutamate receptor oxadiazole ligands and their use as potentiators-841 |
KR20100065191A (ko) | 2007-09-14 | 2010-06-15 | 오르토-맥닐-얀센 파마슈티칼스 인코포레이티드 | 1,3-이치환된 4-(아릴-x-페닐)-1h-피리딘-2-온 |
TW200927731A (en) | 2007-09-14 | 2009-07-01 | Ortho Mcneil Janssen Pharm | 1,3-disubstituted-4-phenyl-1H-pyridin-2-ones |
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JP5707390B2 (ja) | 2009-05-12 | 2015-04-30 | ジャンセン ファーマシューティカルズ, インコーポレイテッド | 1,2,4−トリアゾロ[4,3−a]ピリジン誘導体およびmGluR2受容体の正のアロステリック調節因子としてのその使用 |
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RU2012134329A (ru) | 2010-01-07 | 2014-02-20 | Астразенека Аб | Способ получения позитивного аллостерического модулятора метаботропных глутаматных рецепторов-874 |
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JO3367B1 (ar) | 2013-09-06 | 2019-03-13 | Janssen Pharmaceutica Nv | مركبات 2،1، 4- ثلاثي زولو [3،4-a] بيريدين واستخدامها بصفة منظمات تفارغية موجبة لمستقبلات ميجلور 2 |
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