HK1094582A1 - Process for producing pentacyclic taxane - Google Patents
Process for producing pentacyclic taxaneInfo
- Publication number
- HK1094582A1 HK1094582A1 HK07101873.3A HK07101873A HK1094582A1 HK 1094582 A1 HK1094582 A1 HK 1094582A1 HK 07101873 A HK07101873 A HK 07101873A HK 1094582 A1 HK1094582 A1 HK 1094582A1
- Authority
- HK
- Hong Kong
- Prior art keywords
- group
- oral
- compound
- formula
- antitumor compounds
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
- C07D493/02—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
- C07D493/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/61—Halogen atoms or nitro radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
- C07D493/02—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
- C07D493/08—Bridged systems
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- General Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Plural Heterocyclic Compounds (AREA)
- Epoxy Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2004136359 | 2004-04-30 | ||
| PCT/JP2005/008034 WO2005105807A1 (ja) | 2004-04-30 | 2005-04-27 | 五環性タキサンの製造方法 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| HK1094582A1 true HK1094582A1 (en) | 2007-04-04 |
Family
ID=35241616
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HK07101873.3A HK1094582A1 (en) | 2004-04-30 | 2007-02-15 | Process for producing pentacyclic taxane |
Country Status (14)
| Country | Link |
|---|---|
| US (2) | US7456302B2 (es) |
| EP (1) | EP1741716B8 (es) |
| JP (1) | JP4800205B2 (es) |
| KR (1) | KR101186475B1 (es) |
| CN (1) | CN1942473B (es) |
| AT (1) | ATE526332T1 (es) |
| CA (1) | CA2565013C (es) |
| DK (1) | DK1741716T3 (es) |
| ES (1) | ES2371947T3 (es) |
| HK (1) | HK1094582A1 (es) |
| IL (1) | IL178918A (es) |
| MX (1) | MXPA06012588A (es) |
| PT (1) | PT1741716E (es) |
| WO (1) | WO2005105807A1 (es) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2007307057B2 (en) * | 2006-10-10 | 2011-09-15 | F. Hoffmann La-Roche Ag | Preparation of nucleosides ribofuranosyl pyrimidines |
| WO2008121476A1 (en) * | 2007-03-28 | 2008-10-09 | Tapestry Pharmaceuticals, Inc. | Biologically active taxane analogs and methods of treatment by oral administration |
| US8785669B2 (en) | 2010-06-30 | 2014-07-22 | Gfv, Llc | Taxane compounds, compositions and methods |
| US8697892B2 (en) | 2010-06-30 | 2014-04-15 | Gfv, Llc | Taxane compounds, compositions and methods |
| FR2986526A1 (fr) | 2012-02-03 | 2013-08-09 | Sanofi Sa | Procede de preparation de derives du taxol et certains composes intermediaires |
| WO2013162922A1 (en) * | 2012-04-25 | 2013-10-31 | Genta Incorporated | Taxane compounds, compositions and methods |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP3746563B2 (ja) * | 1995-04-28 | 2006-02-15 | 第一製薬株式会社 | 五環性化合物 |
| TW480262B (en) * | 1995-04-28 | 2002-03-21 | Daiichi Seiyaku Co | A taxol derivative having an antitumor activity and a pharmaceutical composition comprising the same |
| US6008417A (en) * | 1997-10-20 | 1999-12-28 | Roche Vitamins Inc. | Process for making metabolites of lycopene |
| US6677456B2 (en) * | 1999-10-15 | 2004-01-13 | Daiichi Pharmaceutical Co., Ltd. | Pentacyclic taxan compound |
| DE60039998D1 (de) * | 1999-10-15 | 2008-10-02 | Daiichi Sankyo Co Ltd | Pentacyclische taxan-verbindungen |
| JP3776818B2 (ja) * | 2001-03-07 | 2006-05-17 | 第一製薬株式会社 | 五環性タキサン化合物およびその製造方法 |
| CN1295229C (zh) | 2001-11-29 | 2007-01-17 | 第一制药株式会社 | 紫杉烷衍生物的结晶及其制备方法 |
-
2005
- 2005-04-27 KR KR1020067025289A patent/KR101186475B1/ko not_active IP Right Cessation
- 2005-04-27 DK DK05737233.6T patent/DK1741716T3/da active
- 2005-04-27 US US11/579,140 patent/US7456302B2/en active Active
- 2005-04-27 ES ES05737233T patent/ES2371947T3/es active Active
- 2005-04-27 AT AT05737233T patent/ATE526332T1/de active
- 2005-04-27 EP EP05737233A patent/EP1741716B8/en not_active Not-in-force
- 2005-04-27 CA CA2565013A patent/CA2565013C/en not_active Expired - Fee Related
- 2005-04-27 CN CN2005800117870A patent/CN1942473B/zh not_active Expired - Fee Related
- 2005-04-27 PT PT05737233T patent/PT1741716E/pt unknown
- 2005-04-27 JP JP2006512820A patent/JP4800205B2/ja not_active Expired - Fee Related
- 2005-04-27 MX MXPA06012588A patent/MXPA06012588A/es active IP Right Grant
- 2005-04-27 WO PCT/JP2005/008034 patent/WO2005105807A1/ja active Application Filing
-
2006
- 2006-10-29 IL IL178918A patent/IL178918A/en not_active IP Right Cessation
-
2007
- 2007-02-15 HK HK07101873.3A patent/HK1094582A1/xx not_active IP Right Cessation
-
2008
- 2008-09-25 US US12/238,070 patent/US7678919B2/en active Active
Also Published As
| Publication number | Publication date |
|---|---|
| ES2371947T3 (es) | 2012-01-11 |
| US7456302B2 (en) | 2008-11-25 |
| EP1741716A1 (en) | 2007-01-10 |
| DK1741716T3 (da) | 2011-11-28 |
| EP1741716B1 (en) | 2011-09-28 |
| IL178918A0 (en) | 2007-03-08 |
| CA2565013A1 (en) | 2005-11-10 |
| US20070167630A1 (en) | 2007-07-19 |
| CN1942473A (zh) | 2007-04-04 |
| US7678919B2 (en) | 2010-03-16 |
| IL178918A (en) | 2011-06-30 |
| ATE526332T1 (de) | 2011-10-15 |
| KR20070026553A (ko) | 2007-03-08 |
| US20090030209A1 (en) | 2009-01-29 |
| EP1741716A4 (en) | 2009-03-04 |
| JPWO2005105807A1 (ja) | 2008-03-13 |
| WO2005105807A1 (ja) | 2005-11-10 |
| CN1942473B (zh) | 2011-02-02 |
| EP1741716B8 (en) | 2012-02-22 |
| MXPA06012588A (es) | 2007-01-31 |
| JP4800205B2 (ja) | 2011-10-26 |
| PT1741716E (pt) | 2011-12-21 |
| KR101186475B1 (ko) | 2012-09-27 |
| CA2565013C (en) | 2013-01-08 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PC | Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee) |
Effective date: 20160427 |