HK1088327A1 - Thiadiazine derivatives and use thereof as positive ampa receptor modulator - Google Patents
Thiadiazine derivatives and use thereof as positive ampa receptor modulatorInfo
- Publication number
- HK1088327A1 HK1088327A1 HK06108870A HK06108870A HK1088327A1 HK 1088327 A1 HK1088327 A1 HK 1088327A1 HK 06108870 A HK06108870 A HK 06108870A HK 06108870 A HK06108870 A HK 06108870A HK 1088327 A1 HK1088327 A1 HK 1088327A1
- Authority
- HK
- Hong Kong
- Prior art keywords
- receptor modulator
- ampa receptor
- thiadiazine derivatives
- positive ampa
- positive
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Psychiatry (AREA)
- Hospice & Palliative Care (AREA)
- Pain & Pain Management (AREA)
- Psychology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0305448A FR2854634B1 (fr) | 2003-05-05 | 2003-05-05 | Nouveaux derives de thiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
PCT/FR2004/001070 WO2004099217A1 (fr) | 2003-05-05 | 2004-05-04 | Derives de thiadiazine et leur utilisation comme modulateurs positifs des recepteurs ampa |
Publications (1)
Publication Number | Publication Date |
---|---|
HK1088327A1 true HK1088327A1 (en) | 2006-11-03 |
Family
ID=33306157
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HK06108870A HK1088327A1 (en) | 2003-05-05 | 2006-08-10 | Thiadiazine derivatives and use thereof as positive ampa receptor modulator |
Country Status (21)
Country | Link |
---|---|
US (1) | US7476668B2 (pt) |
EP (1) | EP1620441A1 (pt) |
JP (1) | JP4461139B2 (pt) |
KR (1) | KR100741235B1 (pt) |
CN (1) | CN100363368C (pt) |
AR (1) | AR044245A1 (pt) |
AU (1) | AU2004236005B2 (pt) |
BR (1) | BRPI0410002A (pt) |
CA (1) | CA2524377C (pt) |
EA (1) | EA009240B1 (pt) |
FR (1) | FR2854634B1 (pt) |
GE (1) | GEP20084318B (pt) |
HK (1) | HK1088327A1 (pt) |
MA (1) | MA27732A1 (pt) |
MX (1) | MXPA05011823A (pt) |
MY (1) | MY136694A (pt) |
NO (1) | NO20055695L (pt) |
NZ (1) | NZ543214A (pt) |
UA (1) | UA80046C2 (pt) |
WO (1) | WO2004099217A1 (pt) |
ZA (1) | ZA200508660B (pt) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DK1781265T3 (da) | 2004-08-25 | 2010-08-02 | Essentialis Inc | Farmaceutiske formuleringer af kalium ATP-kanal-åbnere og anvendelser deraf |
PL1968601T3 (pl) | 2006-01-05 | 2012-03-30 | Essentialis Inc | Sole związków otwierających kanały potasowe ATP i ich zastosowanie |
WO2010054336A2 (en) * | 2008-11-10 | 2010-05-14 | The Regents Of The University Of California | Therapeutic uses of ampa receptor modulators for treatment of motor dysfunction |
PL2603513T3 (pl) | 2010-08-10 | 2020-07-27 | Takeda Pharmaceutical Company Limited | Heterocykliczny związek i jego zastosowanie jako pozytywny modulator allosteryczny receptora AMPA |
JP5901365B2 (ja) * | 2012-03-12 | 2016-04-06 | 株式会社トクヤマ | イミダート化合物の製造方法 |
AU2014277952A1 (en) | 2013-06-13 | 2016-01-28 | Veroscience Llc | Compositions and methods for treating metabolic disorders |
KR101997699B1 (ko) | 2015-07-06 | 2019-07-08 | 고리츠다이가쿠호진 요코하마시리츠다이가쿠 | Ampa 수용체에 특이적으로 결합하는 신규 화합물 |
JP6241974B1 (ja) | 2017-01-11 | 2017-12-06 | 公立大学法人横浜市立大学 | 霊長類生体の脳内ampa受容体のイメージング方法、プログラム、及びスクリーニング方法 |
US10680583B1 (en) * | 2019-02-26 | 2020-06-09 | Xilinx, Inc. | Control circuit for and method of controlling an operation of an integrated circuit device |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3733409A (en) * | 1969-05-20 | 1973-05-15 | Schering Corp | Method of treating hypertension using thieno (1,2,4) thiadiazines |
WO1998012185A1 (en) * | 1996-09-17 | 1998-03-26 | The Regents Of The University Of California | Benzothiadiazide derivatives and their use as allosteric up-modulators of the ampa receptor |
KR20010021936A (ko) * | 1997-07-16 | 2001-03-15 | 한센 핀 베네드, 안네 제헤르, 웨이콥 마리안느 | 융합된 1,2,4-티아디아진 유도체, 그의 제조와 사용 |
JP2002504481A (ja) * | 1998-02-18 | 2002-02-12 | ニューロサーチ、アクティーゼルスカブ | 新規化合物及び陽性ampaレセプターモジュレーターとしてこれを使用する方法 |
FR2801587B1 (fr) * | 1999-11-30 | 2002-01-11 | Adir | Nouveaux derives de benzothiadiazines, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
-
2003
- 2003-05-05 FR FR0305448A patent/FR2854634B1/fr not_active Expired - Fee Related
-
2004
- 2004-04-05 UA UAA200511454A patent/UA80046C2/uk unknown
- 2004-04-30 MY MYPI20041647A patent/MY136694A/en unknown
- 2004-05-04 AU AU2004236005A patent/AU2004236005B2/en not_active Ceased
- 2004-05-04 ZA ZA200508660A patent/ZA200508660B/en unknown
- 2004-05-04 KR KR1020057020817A patent/KR100741235B1/ko not_active IP Right Cessation
- 2004-05-04 MX MXPA05011823A patent/MXPA05011823A/es active IP Right Grant
- 2004-05-04 CA CA2524377A patent/CA2524377C/fr not_active Expired - Fee Related
- 2004-05-04 NZ NZ543214A patent/NZ543214A/en not_active IP Right Cessation
- 2004-05-04 GE GEAP20049092A patent/GEP20084318B/en unknown
- 2004-05-04 EA EA200501696A patent/EA009240B1/ru not_active IP Right Cessation
- 2004-05-04 JP JP2006505830A patent/JP4461139B2/ja not_active Expired - Fee Related
- 2004-05-04 AR ARP040101515A patent/AR044245A1/es unknown
- 2004-05-04 CN CNB200480014886XA patent/CN100363368C/zh not_active Expired - Fee Related
- 2004-05-04 EP EP04742632A patent/EP1620441A1/fr not_active Withdrawn
- 2004-05-04 WO PCT/FR2004/001070 patent/WO2004099217A1/fr active Application Filing
- 2004-05-04 US US10/555,743 patent/US7476668B2/en not_active Expired - Fee Related
- 2004-05-04 BR BRPI0410002-6A patent/BRPI0410002A/pt not_active IP Right Cessation
-
2005
- 2005-10-21 MA MA28567A patent/MA27732A1/fr unknown
- 2005-12-01 NO NO20055695A patent/NO20055695L/no not_active Application Discontinuation
-
2006
- 2006-08-10 HK HK06108870A patent/HK1088327A1/xx not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
EA200501696A1 (ru) | 2006-06-30 |
MA27732A1 (fr) | 2006-01-02 |
US20070004709A1 (en) | 2007-01-04 |
CN100363368C (zh) | 2008-01-23 |
UA80046C2 (en) | 2007-08-10 |
JP4461139B2 (ja) | 2010-05-12 |
NO20055695L (no) | 2005-12-01 |
BRPI0410002A (pt) | 2006-04-25 |
MY136694A (en) | 2008-11-28 |
FR2854634A1 (fr) | 2004-11-12 |
NZ543214A (en) | 2009-02-28 |
US7476668B2 (en) | 2009-01-13 |
EP1620441A1 (fr) | 2006-02-01 |
CA2524377A1 (fr) | 2004-11-18 |
CA2524377C (fr) | 2010-08-24 |
ZA200508660B (en) | 2007-01-31 |
AU2004236005A1 (en) | 2004-11-18 |
CN1798750A (zh) | 2006-07-05 |
FR2854634B1 (fr) | 2005-07-08 |
KR20060006830A (ko) | 2006-01-19 |
MXPA05011823A (es) | 2006-05-25 |
AU2004236005B2 (en) | 2010-01-21 |
GEP20084318B (en) | 2008-03-10 |
KR100741235B1 (ko) | 2007-07-19 |
EA009240B1 (ru) | 2007-12-28 |
AR044245A1 (es) | 2005-09-07 |
JP2006525292A (ja) | 2006-11-09 |
WO2004099217A1 (fr) | 2004-11-18 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
PC | Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee) |
Effective date: 20120504 |