HK1036593A1 - Use of oxazolidinones in the manufacture of a medicament for treating non-topical infections. - Google Patents

Use of oxazolidinones in the manufacture of a medicament for treating non-topical infections.

Info

Publication number
HK1036593A1
HK1036593A1 HK01107513A HK01107513A HK1036593A1 HK 1036593 A1 HK1036593 A1 HK 1036593A1 HK 01107513 A HK01107513 A HK 01107513A HK 01107513 A HK01107513 A HK 01107513A HK 1036593 A1 HK1036593 A1 HK 1036593A1
Authority
HK
Hong Kong
Prior art keywords
oxazolidinones
medicament
manufacture
treating non
topical infections
Prior art date
Application number
HK01107513A
Other languages
English (en)
Inventor
Charles W Ford
Jeffrey L Watts
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of HK1036593A1 publication Critical patent/HK1036593A1/xx

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • A61K31/422Oxazoles not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/444Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/53751,4-Oxazines, e.g. morpholine
    • A61K31/53771,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/02Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/16Otologicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Pain & Pain Management (AREA)
  • Cardiology (AREA)
  • Rheumatology (AREA)
  • Dermatology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Medicinal Preparation (AREA)
  • Plural Heterocyclic Compounds (AREA)
HK01107513A 1998-06-05 2001-10-29 Use of oxazolidinones in the manufacture of a medicament for treating non-topical infections. HK1036593A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US8828398P 1998-06-05 1998-06-05
PCT/US1999/010463 WO1999062504A2 (en) 1998-06-05 1999-05-26 Topical administration of oxazolidinones for transdermal delivery

Publications (1)

Publication Number Publication Date
HK1036593A1 true HK1036593A1 (en) 2002-01-11

Family

ID=22210475

Family Applications (1)

Application Number Title Priority Date Filing Date
HK01107513A HK1036593A1 (en) 1998-06-05 2001-10-29 Use of oxazolidinones in the manufacture of a medicament for treating non-topical infections.

Country Status (29)

Country Link
US (2) US6613349B2 (zh)
EP (1) EP1083900B1 (zh)
JP (1) JP2002516852A (zh)
KR (1) KR100626781B1 (zh)
CN (1) CN1168447C (zh)
AT (1) ATE220548T1 (zh)
AU (1) AU749523B2 (zh)
BR (1) BR9910318A (zh)
CA (1) CA2327326A1 (zh)
CO (1) CO5011042A1 (zh)
CZ (1) CZ292420B6 (zh)
DE (1) DE69902170T2 (zh)
DK (1) DK1083900T3 (zh)
EA (1) EA003699B1 (zh)
ES (1) ES2179658T3 (zh)
HK (1) HK1036593A1 (zh)
HU (1) HU225234B1 (zh)
ID (1) ID23775A (zh)
IL (1) IL139843A0 (zh)
MY (1) MY122454A (zh)
NO (1) NO20006161L (zh)
NZ (1) NZ508636A (zh)
PL (1) PL193535B1 (zh)
PT (1) PT1083900E (zh)
SK (1) SK285352B6 (zh)
TR (1) TR200003205T2 (zh)
TW (1) TWI224000B (zh)
WO (1) WO1999062504A2 (zh)
ZA (1) ZA200005886B (zh)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6562820B2 (en) 2000-07-05 2003-05-13 Pharmacia & Upjohn Company Method for treatment and prevention of mastitis
US20030096850A1 (en) * 2001-10-11 2003-05-22 Ford Charles W. Treating infections by administration of oxazolidinones
RU2354372C2 (ru) * 2002-03-29 2009-05-10 Фармация Энд Апджон Компани Ллс Парентеральное, внутривенное и пероральное введение оксазолидинонов для лечения инфекционных поражений стопы при диабете
US20060222692A1 (en) * 2005-03-31 2006-10-05 Fairfield Clinical Trials Llc Method and compositions for transdermal administration of antimicrobial medications
CN112409285A (zh) * 2020-11-30 2021-02-26 山东金城昆仑药业有限公司 噁唑烷酮类化合物的晶型及其制备方法和应用

Family Cites Families (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3743727A (en) 1970-11-16 1973-07-03 Crown Zellerbach Corp Enhancing tissue penetration of certain antimicrobial agents with dimethyl sulfoxide
US4507287A (en) 1983-06-20 1985-03-26 Dixon Glen J Preparation and method for the treatment of acne
JP2558107B2 (ja) 1986-12-18 1996-11-27 第一製薬株式会社 外用剤
US4943435A (en) 1987-10-05 1990-07-24 Pharmetrix Corporation Prolonged activity nicotine patch
US4960771A (en) 1988-07-12 1990-10-02 Rajadhyaksha Vithal J Oxazolidinone penetration enhancing compounds
US5254577A (en) * 1988-07-29 1993-10-19 The Du Pont Merck Pharmaceutical Company Aminomethyloxooxazolidinyl arylbenzene derivatives useful as antibacterial agents
US5164510A (en) 1988-09-15 1992-11-17 The Upjohn Company 5'Indolinyl-5β-amidomethyloxazolidin-2-ones
US5231188A (en) 1989-11-17 1993-07-27 The Upjohn Company Tricyclic [6.5.51]-fused oxazolidinone antibacterial agents
US5143928A (en) * 1990-03-27 1992-09-01 Warner-Lambert Company 3,5-di-tertiarybutyl-4-hydroxyphenylmethylene derivatives of 2-substituted thiazolidinones, oxazolidinones, and imidazolidinones as antiinflammatory agents
DK0610265T3 (da) 1991-11-01 1997-06-09 Upjohn Co Substituerede aryl- og heteroarylphenyloxazolidioner, som kan anvendes som antibakterielle midler
TW203552B (en) * 1992-02-18 1993-04-11 J Baroody Lloyd Compositions of clindamycin and benzoyl peroxide for acne treatment
US5457194A (en) * 1993-03-17 1995-10-10 Abbott Laboratories Substituted aliphatic amine-containing macrocyclic immunomodulators
US5688792A (en) * 1994-08-16 1997-11-18 Pharmacia & Upjohn Company Substituted oxazine and thiazine oxazolidinone antimicrobials
WO1995014684A1 (en) * 1993-11-22 1995-06-01 The Upjohn Company Esters of substituted-hydroxyacetyl piperazine phenyl oxazolidinones
DE4425613A1 (de) 1994-07-20 1996-01-25 Bayer Ag 5-gliedrige Heteroaryl-oxazolidinone
DE4425612A1 (de) 1994-07-20 1996-04-04 Bayer Ag 6-gliedrige stickstoffhaltige Heteroaryl-oxazolidinone
DE69517816T2 (de) 1994-09-14 2000-12-28 Minnesota Mining & Mfg Matrix für transdermale wirkstofffreisetzung
US5604262A (en) * 1995-03-22 1997-02-18 Research Corporation Technologies, Inc. Topical antimicrobial agents
ZA968661B (en) * 1995-11-17 1998-04-14 Upjohn Co Oxazolidinone antibacterial agent with tricyclic substituents.
EP0898477B1 (en) * 1996-05-10 2002-12-18 PHARMACIA & UPJOHN COMPANY Topical administration of premafloxacin for the treatment of systemic bacterial diseases
US5929086A (en) 1996-05-10 1999-07-27 Pharmacia & Upjohn Company Topical administration of antimicrobial agents for the treatment of systemic bacterial diseases
US6040306A (en) * 1997-11-18 2000-03-21 Pharmacia & Upjohn Company Method of treating psoriasis, arthritis and reducing the toxicity of cancer chemotherapy
US6312715B1 (en) 1998-05-01 2001-11-06 3M Innovative Properties Company Adhesive microsphere drug delivery composition
US6174878B1 (en) * 1999-08-31 2001-01-16 Alcon Laboratories, Inc. Topical use of kappa opioid agonists to treat otic pain

Also Published As

Publication number Publication date
NO20006161D0 (no) 2000-12-04
CA2327326A1 (en) 1999-12-09
ATE220548T1 (de) 2002-08-15
JP2002516852A (ja) 2002-06-11
PL193535B1 (pl) 2007-02-28
IL139843A0 (en) 2002-02-10
US20020009483A1 (en) 2002-01-24
EP1083900A2 (en) 2001-03-21
CZ20004432A3 (cs) 2001-03-14
CN1298302A (zh) 2001-06-06
HU225234B1 (en) 2006-08-28
PT1083900E (pt) 2002-12-31
EA200100010A1 (ru) 2001-06-25
ZA200005886B (en) 2002-04-22
US20040072841A1 (en) 2004-04-15
WO1999062504A3 (en) 2000-02-24
CN1168447C (zh) 2004-09-29
TWI224000B (en) 2004-11-21
NO20006161L (no) 2000-12-04
HUP0102191A3 (en) 2003-07-28
SK285352B6 (sk) 2006-11-03
AU4184899A (en) 1999-12-20
BR9910318A (pt) 2001-01-30
DE69902170D1 (de) 2002-08-22
DE69902170T2 (de) 2003-03-13
ID23775A (id) 2000-05-11
US7892574B2 (en) 2011-02-22
SK16262000A3 (sk) 2001-06-11
ES2179658T3 (es) 2003-01-16
DK1083900T3 (da) 2002-11-04
EA003699B1 (ru) 2003-08-28
PL345119A1 (en) 2001-12-03
KR20010052555A (ko) 2001-06-25
CO5011042A1 (es) 2001-02-28
CZ292420B6 (cs) 2003-09-17
HUP0102191A2 (hu) 2002-05-29
MY122454A (en) 2006-04-29
KR100626781B1 (ko) 2006-09-22
NZ508636A (en) 2002-03-01
EP1083900B1 (en) 2002-07-17
WO1999062504A2 (en) 1999-12-09
AU749523B2 (en) 2002-06-27
TR200003205T2 (tr) 2001-05-21
US6613349B2 (en) 2003-09-02

Similar Documents

Publication Publication Date Title
Reyzelman et al. Are antibiotics necessary in the treatment of locally infected ingrown toenails?
AU5056196A (en) Hydrogel-forming, self-solvating absorbable polyester copolymers and methods for use thereof
EP1330221A4 (en) PHARMACEUTICAL COMPOSITIONS, DRESSINGS AND METHODS FOR TREATING MICROBIAL INFECTIONS OF SKIN LESIONS
MXPA02002895A (es) Tratamiento topico de infecciones por estreptococcus.
DK0806941T3 (da) Liposomalt antibakterielt præparat med lav fasthed
US20050181028A1 (en) Topical composition and method for treating occlusive wounds
AU1865100A (en) Hyaluronate lyase used for promoting penetration in topical agents
WO2005007072A3 (en) Methods and pharmaceutical compositions for healing wounds
Nolting Non-traumatic removal of the nail and simultaneous treatment of onychomycosis
Milburn et al. Treatment of scleroderma skin ulcers with a hydrocolloid membrane
HK1036593A1 (en) Use of oxazolidinones in the manufacture of a medicament for treating non-topical infections.
Thomas et al. The current status of maggot therapy in wound healing
DK1135020T3 (da) Bipest-behandlinger
IL140769A0 (en) Oxazolidinones to treat eye infections
TR200401810T4 (tr) Kısırlık tedavisinde fsh'ın kullanılması
BR0014751A (pt) Composto, estereoisÈmero ou mistura de estereoisÈmeros, composição farmacêutica, método de tratamento de um paciente em necessidade de tratamento antimicrobiano, e, uso de um composto
ECSP992967A (es) Aplicación topica de oxazolidinonas para administracion transdermica
Avinash et al. Comparative evaluation of efficacy of controlled release local drug delivery system and local irrigation of chlorhexidine gluconate following scaling and root planing-Clinical study
SE9903499D0 (sv) Antimicrobial agent for treatment and prophylaxis
PT1150981E (pt) Composto nucleosidico terapeutico
TH57851B (th) การให้ออกซาโซลิดิโนนเฉพาะที่สำหรับการส่งผ่านทางผิวหนัง
Wieder Jr et al. Undermining Burrowing Ulcer Complicating Post-traumatic Prepatellar Bursitis
TH57851A3 (th) การให้ออกซาโซลิดิโนนเฉพาะที่สำหรับการส่งผ่านทางผิวหนัง
TNSN03022A1 (en) Method for treatment of inflammation
CA2343471A1 (en) Characterization of an antibiotic impregnated delivery system as an intracanal medicament in endodontic therapy

Legal Events

Date Code Title Description
PC Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee)

Effective date: 20080526