HK1028877A1 - Self-emulsifying formulation for lipophilic compounds - Google Patents

Self-emulsifying formulation for lipophilic compounds

Info

Publication number
HK1028877A1
HK1028877A1 HK00108278A HK00108278A HK1028877A1 HK 1028877 A1 HK1028877 A1 HK 1028877A1 HK 00108278 A HK00108278 A HK 00108278A HK 00108278 A HK00108278 A HK 00108278A HK 1028877 A1 HK1028877 A1 HK 1028877A1
Authority
HK
Hong Kong
Prior art keywords
diglyceride
monoglyceride
self
lipophilic compounds
emulsifying formulation
Prior art date
Application number
HK00108278A
Other languages
English (en)
Inventor
Walter Morozowich
Ping Gao
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of HK1028877A1 publication Critical patent/HK1028877A1/xx

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • BPERFORMING OPERATIONS; TRANSPORTING
    • B82NANOTECHNOLOGY
    • B82YSPECIFIC USES OR APPLICATIONS OF NANOSTRUCTURES; MEASUREMENT OR ANALYSIS OF NANOSTRUCTURES; MANUFACTURE OR TREATMENT OF NANOSTRUCTURES
    • B82Y5/00Nanobiotechnology or nanomedicine, e.g. protein engineering or drug delivery
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4433Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with oxygen as a ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/107Emulsions ; Emulsion preconcentrates; Micelles
    • A61K9/1075Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4858Organic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/04Immunostimulants
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
HK00108278A 1997-07-29 2000-12-21 Self-emulsifying formulation for lipophilic compounds HK1028877A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US5407897P 1997-07-29 1997-07-29
PCT/US1998/014816 WO1999006043A1 (en) 1997-07-29 1998-07-27 Self-emulsifying formulation for lipophilic compounds

Publications (1)

Publication Number Publication Date
HK1028877A1 true HK1028877A1 (en) 2001-03-09

Family

ID=21988649

Family Applications (1)

Application Number Title Priority Date Filing Date
HK00108278A HK1028877A1 (en) 1997-07-29 2000-12-21 Self-emulsifying formulation for lipophilic compounds

Country Status (23)

Country Link
US (2) US6531139B1 (xx)
EP (1) EP0999838B1 (xx)
JP (1) JP5005847B2 (xx)
KR (1) KR100509130B1 (xx)
CN (1) CN1113650C (xx)
AT (1) ATE215370T1 (xx)
AU (1) AU728695B2 (xx)
BR (1) BR9810866B1 (xx)
CA (1) CA2294032A1 (xx)
DE (1) DE69804624T2 (xx)
DK (1) DK0999838T3 (xx)
ES (1) ES2174462T3 (xx)
FI (1) FI20000171A (xx)
HK (1) HK1028877A1 (xx)
HU (1) HU225160B1 (xx)
NO (1) NO323773B1 (xx)
NZ (1) NZ502567A (xx)
PL (1) PL192080B1 (xx)
PT (1) PT999838E (xx)
RU (1) RU2203648C2 (xx)
SI (1) SI0999838T1 (xx)
SK (1) SK284579B6 (xx)
WO (1) WO1999006043A1 (xx)

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Also Published As

Publication number Publication date
SK182000A3 (en) 2000-12-11
DE69804624D1 (de) 2002-05-08
HUP0003292A3 (en) 2002-02-28
NO20000465D0 (no) 2000-01-28
ATE215370T1 (de) 2002-04-15
BR9810866B1 (pt) 2010-07-13
SI0999838T1 (en) 2002-08-31
HUP0003292A1 (hu) 2002-01-28
PT999838E (pt) 2002-07-31
AU728695B2 (en) 2001-01-18
BR9810866A (pt) 2000-09-26
US6121313A (en) 2000-09-19
EP0999838A1 (en) 2000-05-17
JP2002510329A (ja) 2002-04-02
ES2174462T3 (es) 2002-11-01
AU8573798A (en) 1999-02-22
EP0999838B1 (en) 2002-04-03
PL338334A1 (en) 2000-10-23
KR100509130B1 (ko) 2005-08-18
NO323773B1 (no) 2007-07-02
CA2294032A1 (en) 1999-02-11
RU2203648C2 (ru) 2003-05-10
DE69804624T2 (de) 2002-09-19
HU225160B1 (en) 2006-07-28
NZ502567A (en) 2002-03-28
WO1999006043A1 (en) 1999-02-11
FI20000171A (fi) 2000-01-28
KR20010022364A (ko) 2001-03-15
JP5005847B2 (ja) 2012-08-22
CN1113650C (zh) 2003-07-09
US6531139B1 (en) 2003-03-11
PL192080B1 (pl) 2006-08-31
SK284579B6 (sk) 2005-07-01
DK0999838T3 (da) 2002-07-08
CN1261797A (zh) 2000-08-02
NO20000465L (no) 2000-03-28

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Effective date: 20150727