GB202020191D0 - Pharmaceutical compounds - Google Patents

Pharmaceutical compounds

Info

Publication number
GB202020191D0
GB202020191D0 GBGB2020191.9A GB202020191A GB202020191D0 GB 202020191 D0 GB202020191 D0 GB 202020191D0 GB 202020191 A GB202020191 A GB 202020191A GB 202020191 D0 GB202020191 D0 GB 202020191D0
Authority
GB
United Kingdom
Prior art keywords
pharmaceutical compounds
pharmaceutical
compounds
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
GBGB2020191.9A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Nxera Pharma UK Ltd
Original Assignee
Heptares Therapeutics Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Heptares Therapeutics Ltd filed Critical Heptares Therapeutics Ltd
Priority to GBGB2020191.9A priority Critical patent/GB202020191D0/en
Publication of GB202020191D0 publication Critical patent/GB202020191D0/en
Priority to PCT/GB2021/053372 priority patent/WO2022129951A1/en
Priority to MX2023007140A priority patent/MX2023007140A/es
Priority to EP21836606.0A priority patent/EP4263536A1/en
Priority to CR20230256A priority patent/CR20230256A/es
Priority to AU2021404194A priority patent/AU2021404194A1/en
Priority to JP2023536899A priority patent/JP7730369B2/ja
Priority to KR1020237023911A priority patent/KR20230121830A/ko
Priority to PE2023001903A priority patent/PE20240646A1/es
Priority to IL303484A priority patent/IL303484A/en
Priority to UAA202303458A priority patent/UA130897C2/uk
Priority to CN202180093050.7A priority patent/CN116848109B/zh
Priority to CA3202054A priority patent/CA3202054A1/en
Priority to US17/874,564 priority patent/US11999745B2/en
Priority to JOJO/P/2023/0128A priority patent/JOP20230128A1/ar
Priority to DO2023000125A priority patent/DOP2023000125A/es
Priority to ECSENADI202344370A priority patent/ECSP23044370A/es
Priority to ZA2023/06305A priority patent/ZA202306305B/en
Priority to CL2023001755A priority patent/CL2023001755A1/es
Priority to CONC2023/0007838A priority patent/CO2023007838A2/es
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/10—Spiro-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/46—8-Azabicyclo [3.2.1] octane; Derivatives thereof, e.g. atropine, cocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D271/00—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/06—1,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles
    • C07D271/07—1,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Biomedical Technology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Hospice & Palliative Care (AREA)
  • Emergency Medicine (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
GBGB2020191.9A 2019-04-23 2020-12-18 Pharmaceutical compounds Ceased GB202020191D0 (en)

Priority Applications (20)

Application Number Priority Date Filing Date Title
GBGB2020191.9A GB202020191D0 (en) 2020-12-18 2020-12-18 Pharmaceutical compounds
CA3202054A CA3202054A1 (en) 2020-12-18 2021-12-20 Pharmaceutical compounds
PE2023001903A PE20240646A1 (es) 2020-12-18 2021-12-20 Compuestos farmaceuticos
UAA202303458A UA130897C2 (uk) 2020-12-18 2021-12-20 Фармацевтичні сполуки
EP21836606.0A EP4263536A1 (en) 2020-12-18 2021-12-20 Pharmaceutical compounds
CR20230256A CR20230256A (es) 2020-12-18 2021-12-20 Compuestos farmacéuticos
AU2021404194A AU2021404194A1 (en) 2020-12-18 2021-12-20 Pharmaceutical compounds
JP2023536899A JP7730369B2 (ja) 2020-12-18 2021-12-20 医薬化合物
KR1020237023911A KR20230121830A (ko) 2020-12-18 2021-12-20 제약 화합물
PCT/GB2021/053372 WO2022129951A1 (en) 2020-12-18 2021-12-20 Pharmaceutical compounds
IL303484A IL303484A (en) 2020-12-18 2021-12-20 Pharmaceutical compounds
MX2023007140A MX2023007140A (es) 2020-12-18 2021-12-20 Compuestos farmaceuticos.
CN202180093050.7A CN116848109B (zh) 2020-12-18 2021-12-20 药物化合物
US17/874,564 US11999745B2 (en) 2020-12-18 2022-07-27 Pharmaceutical compounds
JOJO/P/2023/0128A JOP20230128A1 (ar) 2020-12-18 2023-06-06 مركبات صيدلانية
DO2023000125A DOP2023000125A (es) 2020-12-18 2023-06-15 Compuestos farmacéuticos
ECSENADI202344370A ECSP23044370A (es) 2020-12-18 2023-06-15 Compuestos farmacéuticos
ZA2023/06305A ZA202306305B (en) 2019-04-23 2023-06-15 Pharmaceutical compounds
CL2023001755A CL2023001755A1 (es) 2020-12-18 2023-06-15 Compuestos farmacéuticos.
CONC2023/0007838A CO2023007838A2 (es) 2020-12-18 2023-06-15 Compuestos farmacéuticos

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB2020191.9A GB202020191D0 (en) 2020-12-18 2020-12-18 Pharmaceutical compounds

Publications (1)

Publication Number Publication Date
GB202020191D0 true GB202020191D0 (en) 2021-02-03

Family

ID=74221349

Family Applications (1)

Application Number Title Priority Date Filing Date
GBGB2020191.9A Ceased GB202020191D0 (en) 2019-04-23 2020-12-18 Pharmaceutical compounds

Country Status (19)

Country Link
US (1) US11999745B2 (enExample)
EP (1) EP4263536A1 (enExample)
JP (1) JP7730369B2 (enExample)
KR (1) KR20230121830A (enExample)
CN (1) CN116848109B (enExample)
AU (1) AU2021404194A1 (enExample)
CA (1) CA3202054A1 (enExample)
CL (1) CL2023001755A1 (enExample)
CO (1) CO2023007838A2 (enExample)
CR (1) CR20230256A (enExample)
DO (1) DOP2023000125A (enExample)
EC (1) ECSP23044370A (enExample)
GB (1) GB202020191D0 (enExample)
IL (1) IL303484A (enExample)
JO (1) JOP20230128A1 (enExample)
MX (1) MX2023007140A (enExample)
PE (1) PE20240646A1 (enExample)
UA (1) UA130897C2 (enExample)
WO (1) WO2022129951A1 (enExample)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2619829T3 (es) 2011-11-18 2017-06-27 Heptares Therapeutics Limited Agonistas del receptor muscarínico M1
GB201404922D0 (en) 2014-03-19 2014-04-30 Heptares Therapeutics Ltd Pharmaceutical compounds
GB201513743D0 (en) 2015-08-03 2015-09-16 Heptares Therapeutics Ltd Muscarinic agonists
GB201519352D0 (en) 2015-11-02 2015-12-16 Heptares Therapeutics Ltd Pharmaceutical compounds
GB201617454D0 (en) 2016-10-14 2016-11-30 Heptares Therapeutics Limited Pharmaceutical compounds
GB201810239D0 (en) 2018-06-22 2018-08-08 Heptares Therapeutics Ltd Pharmaceutical compounds
GB201819961D0 (en) 2018-12-07 2019-01-23 Heptares Therapeutics Ltd Pharmaceutical compounds
GB201819960D0 (en) 2018-12-07 2019-01-23 Heptares Therapeutics Ltd Pharmaceutical compounds
GB202020191D0 (en) 2020-12-18 2021-02-03 Heptares Therapeutics Ltd Pharmaceutical compounds

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GB201810245D0 (en) 2018-06-22 2018-08-08 Heptares Therapeutics Ltd Pharmaceutical compounds
GB201819961D0 (en) 2018-12-07 2019-01-23 Heptares Therapeutics Ltd Pharmaceutical compounds
GB201819960D0 (en) 2018-12-07 2019-01-23 Heptares Therapeutics Ltd Pharmaceutical compounds
GB202020191D0 (en) 2020-12-18 2021-02-03 Heptares Therapeutics Ltd Pharmaceutical compounds
GB202103211D0 (en) 2021-03-08 2021-04-21 Heptares Therapeutics Ltd Pharmaceutical compounds for use in therapy

Also Published As

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US11999745B2 (en) 2024-06-04
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DOP2023000125A (es) 2023-08-31
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CN116848109B (zh) 2026-02-10
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AU2021404194A9 (en) 2024-10-17
CL2023001755A1 (es) 2024-01-05
PE20240646A1 (es) 2024-04-04
KR20230121830A (ko) 2023-08-21
US20220380379A1 (en) 2022-12-01

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