CO2023007838A2 - Compuestos farmacéuticos - Google Patents
Compuestos farmacéuticosInfo
- Publication number
- CO2023007838A2 CO2023007838A2 CONC2023/0007838A CO2023007838A CO2023007838A2 CO 2023007838 A2 CO2023007838 A2 CO 2023007838A2 CO 2023007838 A CO2023007838 A CO 2023007838A CO 2023007838 A2 CO2023007838 A2 CO 2023007838A2
- Authority
- CO
- Colombia
- Prior art keywords
- compounds
- pharmaceutical compounds
- agonists
- muscarinic
- salts
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 5
- 102000014415 Muscarinic acetylcholine receptor Human genes 0.000 abstract 2
- 108050003473 Muscarinic acetylcholine receptor Proteins 0.000 abstract 2
- 239000000556 agonist Substances 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 230000001404 mediated effect Effects 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 230000001225 therapeutic effect Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/10—Spiro-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
- C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/46—8-Azabicyclo [3.2.1] octane; Derivatives thereof, e.g. atropine, cocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D271/00—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
- C07D271/02—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
- C07D271/06—1,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles
- C07D271/07—1,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Neurosurgery (AREA)
- Psychiatry (AREA)
- Hospice & Palliative Care (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Emergency Medicine (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Esta invención se refiere a compuestos que son agonistas del receptor muscarínico M1 y M4 y que son útiles en el tratamiento de enfermedades mediadas por los receptores muscarínicos M1 y/o M4. También se proporcionan composiciones farmacéuticas que contienen los compuestos y los usos terapéuticos de los compuestos. Los compuestos proporcionados son de fórmula (1): y sus sales.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB2020191.9A GB202020191D0 (en) | 2020-12-18 | 2020-12-18 | Pharmaceutical compounds |
PCT/GB2021/053372 WO2022129951A1 (en) | 2020-12-18 | 2021-12-20 | Pharmaceutical compounds |
Publications (1)
Publication Number | Publication Date |
---|---|
CO2023007838A2 true CO2023007838A2 (es) | 2023-10-30 |
Family
ID=74221349
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CONC2023/0007838A CO2023007838A2 (es) | 2020-12-18 | 2023-06-15 | Compuestos farmacéuticos |
Country Status (16)
Country | Link |
---|---|
EP (1) | EP4263536A1 (es) |
JP (1) | JP2024504252A (es) |
KR (1) | KR20230121830A (es) |
CN (1) | CN116848109A (es) |
AU (1) | AU2021404194A1 (es) |
CA (1) | CA3202054A1 (es) |
CL (1) | CL2023001755A1 (es) |
CO (1) | CO2023007838A2 (es) |
CR (1) | CR20230256A (es) |
DO (1) | DOP2023000125A (es) |
EC (1) | ECSP23044370A (es) |
GB (1) | GB202020191D0 (es) |
IL (1) | IL303484A (es) |
MX (1) | MX2023007140A (es) |
PE (1) | PE20240646A1 (es) |
WO (1) | WO2022129951A1 (es) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US9187451B2 (en) | 2011-11-18 | 2015-11-17 | Heptares Therapeutics Limited | Muscarinic M1 receptor agonists |
GB201617454D0 (en) | 2016-10-14 | 2016-11-30 | Heptares Therapeutics Limited | Pharmaceutical compounds |
GB201810239D0 (en) | 2018-06-22 | 2018-08-08 | Heptares Therapeutics Ltd | Pharmaceutical compounds |
GB201819960D0 (en) | 2018-12-07 | 2019-01-23 | Heptares Therapeutics Ltd | Pharmaceutical compounds |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB201709652D0 (en) * | 2017-06-16 | 2017-08-02 | Heptares Therapeutics Ltd | Pharmaceutical compounds |
GB201810245D0 (en) * | 2018-06-22 | 2018-08-08 | Heptares Therapeutics Ltd | Pharmaceutical compounds |
-
2020
- 2020-12-18 GB GBGB2020191.9A patent/GB202020191D0/en not_active Ceased
-
2021
- 2021-12-20 CR CR20230256A patent/CR20230256A/es unknown
- 2021-12-20 PE PE2023001903A patent/PE20240646A1/es unknown
- 2021-12-20 IL IL303484A patent/IL303484A/en unknown
- 2021-12-20 AU AU2021404194A patent/AU2021404194A1/en active Pending
- 2021-12-20 MX MX2023007140A patent/MX2023007140A/es unknown
- 2021-12-20 KR KR1020237023911A patent/KR20230121830A/ko unknown
- 2021-12-20 EP EP21836606.0A patent/EP4263536A1/en active Pending
- 2021-12-20 JP JP2023536899A patent/JP2024504252A/ja active Pending
- 2021-12-20 WO PCT/GB2021/053372 patent/WO2022129951A1/en active Application Filing
- 2021-12-20 CN CN202180093050.7A patent/CN116848109A/zh active Pending
- 2021-12-20 CA CA3202054A patent/CA3202054A1/en active Pending
-
2023
- 2023-06-15 EC ECSENADI202344370A patent/ECSP23044370A/es unknown
- 2023-06-15 CO CONC2023/0007838A patent/CO2023007838A2/es unknown
- 2023-06-15 DO DO2023000125A patent/DOP2023000125A/es unknown
- 2023-06-15 CL CL2023001755A patent/CL2023001755A1/es unknown
Also Published As
Publication number | Publication date |
---|---|
JP2024504252A (ja) | 2024-01-31 |
AU2021404194A1 (en) | 2023-08-03 |
WO2022129951A1 (en) | 2022-06-23 |
IL303484A (en) | 2023-08-01 |
CN116848109A (zh) | 2023-10-03 |
GB202020191D0 (en) | 2021-02-03 |
CL2023001755A1 (es) | 2024-01-05 |
PE20240646A1 (es) | 2024-04-04 |
CR20230256A (es) | 2023-09-29 |
US20220380379A1 (en) | 2022-12-01 |
CA3202054A1 (en) | 2022-06-23 |
KR20230121830A (ko) | 2023-08-21 |
ECSP23044370A (es) | 2023-08-31 |
EP4263536A1 (en) | 2023-10-25 |
MX2023007140A (es) | 2023-08-25 |
DOP2023000125A (es) | 2023-08-31 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
DOP2023000125A (es) | Compuestos farmacéuticos | |
CO2018002060A2 (es) | Compuestos farmacéuticos | |
CL2021000907A1 (es) | Nuevas piridopirimidinonas sustituidas con bencilamino y derivados como inhibidores de sos1 (divisional de solicitud n° 01501-2020) | |
ECSP21004787A (es) | Inhibidores de inflamasoma nlrp3 | |
PE20191474A1 (es) | Compuestos de amino-triazolopiridina y su uso en el tratamiento del cancer | |
CO6470866A2 (es) | Enantiómeros de compuestos de espirooxindol y sus usos como agentes terapéuticos. | |
CR9098A (es) | 3-phenyl-pyrazole derivatives as modulators of the 5-ht2a serotonin receptor useful for the treatment of disorders related thereto | |
CL2008002768A1 (es) | Compuestos derivados de carboxiciclopropil-(bis-fenil-oxamidas); composicion farmaceutica que los contiene; procedimiento para la elaboracion de las composiciones y el uso de los compuestos en el tratamiento de diabetes y trastornos del sncentre otras enfermedades. | |
CO2024001922A2 (es) | Inhibidores de nlrp3 | |
MX2020014156A (es) | Oxadiazoles como agonistas de los receptores muscarinicos m1 y/o m4. | |
UY38625A (es) | Compuestos y su uso en el tratamiento del cáncer | |
ECSP23030959A (es) | Compuestos y su uso en el tratamiento del cáncer | |
CL2021001388A1 (es) | Compuestos útiles en la terapia para el vih | |
CO2022015930A2 (es) | Compuestos heterocíclicos como agonistas del receptor de activación expresado en las células mieloides 2 | |
UY38228A (es) | Compuestos de triazolopirimidina y su uso en el tratamiento del cáncer | |
CL2022003041A1 (es) | Compuestos heterocíclicos como agonistas del receptor de activación expresado en las células mieloides 2 | |
CL2022002386A1 (es) | Compuestos de amino pirimidina fusionados | |
CL2019003467A1 (es) | Compuestos bicíclicos 5,6-fusionados y composiciones para el tratamiento de enfermedades parasitarias. | |
CL2022001307A1 (es) | Compuestos antagonistas de receptores de adenosina. | |
UY30880A1 (es) | 7-alcoxicinolin-3-carboxamidas sustituidas y sales farmacéuticamente aceptables de las mismas, procedimientos de preparacion y aplicaciones | |
CO2021001925A2 (es) | Piridopirimidinas como inhibidores del receptor de histamina h4 | |
UY39681A (es) | Derivados de ciclobutilo 1,3–sustituidos y sus usos | |
AR123685A1 (es) | Antagonistas del mrgx2 | |
AR072535A1 (es) | Compuestos de fenantrenona y composiciones farmaceuticas que los contienen | |
CL2021000282A1 (es) | Inhibidores de ckd8/19 |