FR2429793A1 - Nouveaux derives de purine et medicament les contenant - Google Patents

Nouveaux derives de purine et medicament les contenant

Info

Publication number
FR2429793A1
FR2429793A1 FR7921304A FR7921304A FR2429793A1 FR 2429793 A1 FR2429793 A1 FR 2429793A1 FR 7921304 A FR7921304 A FR 7921304A FR 7921304 A FR7921304 A FR 7921304A FR 2429793 A1 FR2429793 A1 FR 2429793A1
Authority
FR
France
Prior art keywords
purine derivatives
medicaments containing
novel purine
novel
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7921304A
Other languages
English (en)
Other versions
FR2429793B1 (fr
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bristol Myers Co
Original Assignee
Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Co filed Critical Bristol Myers Co
Publication of FR2429793A1 publication Critical patent/FR2429793A1/fr
Application granted granted Critical
Publication of FR2429793B1 publication Critical patent/FR2429793B1/fr
Granted legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

L'invention a trait au domaine de la chimie médicale et des intermédiaires chimiques. Elle concerne de nouveaux dérivés de purine de formule :
FR7921304A 1978-05-09 1979-08-23 Nouveaux derives de purine et medicament les contenant Granted FR2429793A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/904,146 US4172829A (en) 1978-05-09 1978-05-09 2,9-Disubstituted adenine derivatives and their use as non-adrenergic bronchodilators

Publications (2)

Publication Number Publication Date
FR2429793A1 true FR2429793A1 (fr) 1980-01-25
FR2429793B1 FR2429793B1 (fr) 1983-02-04

Family

ID=25418652

Family Applications (2)

Application Number Title Priority Date Filing Date
FR7911604A Granted FR2432519A1 (fr) 1978-05-09 1979-05-08 Nouveaux derives de purine et medicament les contenant
FR7921304A Granted FR2429793A1 (fr) 1978-05-09 1979-08-23 Nouveaux derives de purine et medicament les contenant

Family Applications Before (1)

Application Number Title Priority Date Filing Date
FR7911604A Granted FR2432519A1 (fr) 1978-05-09 1979-05-08 Nouveaux derives de purine et medicament les contenant

Country Status (19)

Country Link
US (1) US4172829A (fr)
JP (2) JPS55373A (fr)
AU (1) AU532056B2 (fr)
BE (1) BE876122A (fr)
CA (1) CA1109871A (fr)
CH (1) CH640534A5 (fr)
DE (1) DE2918261A1 (fr)
DK (1) DK145698C (fr)
FI (1) FI66615C (fr)
FR (2) FR2432519A1 (fr)
GB (2) GB2097785B (fr)
GR (1) GR73535B (fr)
IE (1) IE48216B1 (fr)
IT (1) IT1116833B (fr)
LU (1) LU81238A1 (fr)
NL (1) NL7903650A (fr)
SE (2) SE436033B (fr)
YU (1) YU41632B (fr)
ZA (1) ZA792186B (fr)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4232155A (en) * 1979-09-13 1980-11-04 Bristol-Myers Company Purine compounds
FI802401A (fi) * 1979-08-06 1981-02-07 Bristol Myers Co Bronkutvidgande purin
US4269839A (en) * 1979-09-13 1981-05-26 Bristol-Myers Company Alkylthio-adenines used as bronchodilators
US4278675A (en) * 1979-09-13 1981-07-14 Bristol-Myers Company Bronchodilating process
US4286093A (en) * 1980-02-25 1981-08-25 Mead Johnson & Company 9-Cyclohexyl-2-alkoxy-9H-adenine process
JPS6237165Y2 (fr) * 1980-05-29 1987-09-22
US4419358A (en) * 1981-11-12 1983-12-06 Mead Johnson & Company Isethionic acid salt of 9-cyclohexyl-2-propoxy-9H-purine-6-amine and compositions containing an effective bronchodilating concentration of it
US5015739A (en) * 1988-04-22 1991-05-14 Schering Corporation Processes for preparation of cyclopentyl purine derivatives
JPH027537A (ja) * 1988-06-27 1990-01-11 Dainippon Printing Co Ltd 移動装置及び形状測定装置
US4999428A (en) * 1989-04-14 1991-03-12 Schering Corporation Process for preparing cyclopentyl purine derivatives
JPH0379236U (fr) * 1990-08-24 1991-08-13
JPH0379235U (fr) * 1990-08-24 1991-08-13
AU4589800A (en) * 1999-05-05 2000-11-21 Darwin Discovery Limited 9-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,9-dihydropurin-6-one derivatives as pde7inhibitors
EP1210347B1 (fr) * 1999-09-10 2004-06-23 Stichting REGA V.Z.W. Nucleosides carbocycliques et procede de production correspondant
AU2877102A (en) * 2000-11-02 2002-05-15 Sloan Kettering Inst Cancer Small molecule compositions for binding to hsp90
WO2015005491A1 (fr) * 2013-07-12 2015-01-15 国立大学法人京都大学 Procédé de criblage d'une substance capable d'inhiber l'épissage anormal provoquant l'apparition ou l'évolution d'une maladie

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5271492A (en) * 1975-12-10 1977-06-14 Kohjin Co Ltd Synthesis of 9-substituted-2-substituted thioadenines

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3930005A (en) * 1973-06-15 1975-12-30 Squibb & Sons Inc Antiinflammatory agents and their use
US3917837A (en) * 1974-10-21 1975-11-04 American Cyanamid Co Method of using trans-2-(6-amino-9H-purin-9-yl)-cyclopentanol
DE2610985A1 (de) 1976-03-16 1977-09-29 Byk Gulden Lomberg Chem Fab Arzneimittel enthaltend beta-d-1 (6-amino-9h-purin-9-yl)-1-deoxyribofuranuronsaeurederivate
US4076711A (en) * 1976-04-05 1978-02-28 Schering Corporation Triazolo [4,5-d]-pyrimidines

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5271492A (en) * 1975-12-10 1977-06-14 Kohjin Co Ltd Synthesis of 9-substituted-2-substituted thioadenines

Non-Patent Citations (3)

* Cited by examiner, † Cited by third party
Title
ABJP/77 *
CA1973 *
EXBK/59 *

Also Published As

Publication number Publication date
GB2020655B (en) 1982-08-25
DK188279A (da) 1979-11-10
AU4689679A (en) 1979-11-15
JPS62116583A (ja) 1987-05-28
CA1109871A (fr) 1981-09-29
IE48216B1 (en) 1984-10-31
ZA792186B (en) 1980-05-28
FR2432519A1 (fr) 1980-02-29
DE2918261A1 (de) 1979-11-15
FR2429793B1 (fr) 1983-02-04
SE436033B (sv) 1984-11-05
IT1116833B (it) 1986-02-10
LU81238A1 (fr) 1979-12-07
FI66615B (fi) 1984-07-31
SE7903976L (sv) 1979-11-10
SE8401493L (sv) 1984-03-16
GB2020655A (en) 1979-11-21
CH640534A5 (de) 1984-01-13
NL7903650A (nl) 1979-11-13
DK145698C (da) 1983-07-25
GB2097785A (en) 1982-11-10
US4172829A (en) 1979-10-30
IT7948986A0 (it) 1979-05-09
AU532056B2 (en) 1983-09-15
DE2918261C2 (fr) 1988-08-04
FI66615C (fi) 1984-11-12
JPS626555B2 (fr) 1987-02-12
IE790878L (en) 1979-11-09
JPS55373A (en) 1980-01-05
DK145698B (da) 1983-01-31
GB2097785B (en) 1983-03-23
BE876122A (fr) 1979-11-08
YU108579A (en) 1983-12-31
FR2432519B1 (fr) 1983-02-04
GR73535B (fr) 1984-03-12
FI791456A (fi) 1979-11-10
SE8401493D0 (sv) 1984-03-16
SE449864B (sv) 1987-05-25
YU41632B (en) 1987-12-31
JPH0146515B2 (fr) 1989-10-09

Similar Documents

Publication Publication Date Title
FR2429793A1 (fr) Nouveaux derives de purine et medicament les contenant
FR2405955A1 (fr) Nouveaux ylides utiles dans la synthese de medicaments
FR2444031A1 (fr) Nouveaux derives d'imidazole, leur procede de production et composition pharmaceutique les contenant
FR2430410A1 (fr) Phenethanolamines et compositions pharmaceutiques en contenant
FR2429593A1 (fr) Medicaments contenant des derives d'imidazole
FR2442851A1 (fr) Nouvelles spiro(4 h-2,3-dihydrovenzopyranne(4,5')oxazolidine)-2',4'-diones et medicament en contenant
FR2371437A1 (fr) Nouveaux derives de pipepidine ou de morpholine utiles comme medicaments et comme fongicides
FR2398748A1 (fr) Nouveaux derives d'imidazoquinazoline, leur preparation et leur application en tant que medicaments
FR2364206A1 (fr) Nouveaux derives d'acides phenoxyvaleriques et compositions herbicides les contenant
FR2432511A1 (fr) Derives triazoliques, leur preparation et leur application en tant que medicaments
FR2446828A1 (fr) N-benzylimidazoles inhibiteurs selectifs de thromboxanne-synthetase, leur procede de production et compositions pharmaceutiques les contenant
FR2402640A1 (fr) Nouveaux phenols a substituant hydroxyalkyle ou oxoalkyle et composition pharmaceutique les contenant
FR2424913A1 (fr) Nouvelles 4-(quinolinylaminobenzoyl) piperazines et composition pharmaceutique les contenant
FR2391215A1 (fr) Nouvelles imidazoazines et imidazodiazines, leur preparation et leur application en tant que medicaments
FR2387229A1 (fr) Dipyrido (4,3-b) (3,4-f) indoles, procede d'obtention, application therapeutique et compositions pharmaceutiques les contenant
FR2394546A1 (fr) Nouveaux derives de 1,2,3,4,6,7-hexahydro-11bah-benzo(a)-quinolizine, leur preparation et leur application en tant que medicaments
FR2446819A1 (fr) Derives 6-alkyles d'acide 1,2-dihydro-2-oxonicotinique et composition pharmaceutique les contenant
FR2422405A1 (fr) Nouveaux medicaments constitues de derives de l'acide p-aminobenzoique
FR2392999A1 (fr) Nouveaux derives de l'acide 6-((aminosulfonyl)-phenyl)-1,2-dihydro-2-oxonicotinique utile comme medicament
FR2453152A1 (fr) Nouveaux derives de prostaglandine et medicament les contenant
FR2426039A1 (fr) Derives de di-o-n-alkylglycerols et medicament immuno-stimulant les contenant
FR2392958A1 (fr) Nouveaux amino-acides fluores utiles comme medicament
FR2430947A1 (fr) Nouveaux composes de 2-amino-octahydro-indolo-(2,3-a)-quinazoline, leur procede de production et medicament les contenant
FR2361361A1 (fr) Nouveaux derives du cyclopentane et medicaments contenant ces substances
FR2401141A1 (fr) Nouveaux derives halogenes de prostaglandines et medicaments les contenant

Legal Events

Date Code Title Description
ST Notification of lapse