FR2401141A1 - Nouveaux derives halogenes de prostaglandines et medicaments les contenant - Google Patents

Nouveaux derives halogenes de prostaglandines et medicaments les contenant

Info

Publication number
FR2401141A1
FR2401141A1 FR7830488A FR7830488A FR2401141A1 FR 2401141 A1 FR2401141 A1 FR 2401141A1 FR 7830488 A FR7830488 A FR 7830488A FR 7830488 A FR7830488 A FR 7830488A FR 2401141 A1 FR2401141 A1 FR 2401141A1
Authority
FR
France
Prior art keywords
prostaglandins
halogen derivatives
medicines containing
new halogen
new
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
FR7830488A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pharmacia and Upjohn Co
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of FR2401141A1 publication Critical patent/FR2401141A1/fr
Pending legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/93Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems condensed with a ring other than six-membered
    • C07D307/935Not further condensed cyclopenta [b] furans or hydrogenated cyclopenta [b] furans
    • C07D307/937Not further condensed cyclopenta [b] furans or hydrogenated cyclopenta [b] furans with hydrocarbon or substituted hydrocarbon radicals directly attached in position 2, e.g. prostacyclins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C405/00Compounds containing a five-membered ring having two side-chains in ortho position to each other, and having oxygen atoms directly attached to the ring in ortho position to one of the side-chains, one side-chain containing, not directly attached to the ring, a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, and the other side-chain having oxygen atoms attached in gamma-position to the ring, e.g. prostaglandins ; Analogues or derivatives thereof

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Furan Compounds (AREA)
  • Pyrane Compounds (AREA)

Abstract

L'invention se situe dans le domaine pharmaceutique. Elle concerne de nouveaux dérivés halogénés de prostaglandines ayant comme formule :
FR7830488A 1977-03-07 1978-10-26 Nouveaux derives halogenes de prostaglandines et medicaments les contenant Pending FR2401141A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US77500377A 1977-03-07 1977-03-07

Publications (1)

Publication Number Publication Date
FR2401141A1 true FR2401141A1 (fr) 1979-03-23

Family

ID=25103006

Family Applications (2)

Application Number Title Priority Date Filing Date
FR7806484A Pending FR2401139A2 (fr) 1977-03-07 1978-03-07 Nouveaux derives d5 de prostaglandines, leur procede de preparation et medicaments les contenant
FR7830488A Pending FR2401141A1 (fr) 1977-03-07 1978-10-26 Nouveaux derives halogenes de prostaglandines et medicaments les contenant

Family Applications Before (1)

Application Number Title Priority Date Filing Date
FR7806484A Pending FR2401139A2 (fr) 1977-03-07 1978-03-07 Nouveaux derives d5 de prostaglandines, leur procede de preparation et medicaments les contenant

Country Status (12)

Country Link
US (1) US4150222A (fr)
JP (1) JPS53111041A (fr)
AU (1) AU524786B2 (fr)
BE (1) BE864644A (fr)
CA (1) CA1159452A (fr)
CH (1) CH636353A5 (fr)
DE (1) DE2809452A1 (fr)
FR (2) FR2401139A2 (fr)
GB (1) GB1576570A (fr)
IE (1) IE46570B1 (fr)
IL (1) IL54176A0 (fr)
NZ (1) NZ186516A (fr)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2401920A1 (fr) * 1977-07-28 1979-03-30 Upjohn Co Derives de prostaglandines

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4215214A (en) * 1976-08-23 1980-07-29 The Upjohn Company Enlarged-hetero-ring prostacyclin analogs with 5-halo feature
FI71138C (fi) * 1976-12-31 1986-11-24 Erba Farmitalia Foerfarande foer framstaellning av terapeutiskt aktiva bisykliska prostaglandiner
IT1088036B (it) 1977-11-25 1985-06-04 Erba Carlo Spa 15-epi-prostaciclina e prostaciclina analoghi
DE2947526A1 (de) * 1978-11-29 1980-06-12 Ono Pharmaceutical Co Prostacyclin-analoge
DE2902809A1 (de) * 1979-01-25 1980-08-07 Hoechst Ag Neue analoga von prostacyclin
DE3029984C2 (de) * 1980-08-08 1983-12-15 Grünenthal GmbH, 5190 Stolberg 2-Oxabicyclo [3.3.0] octanderivate und diese enthaltende Arzneimittel
DE3035713A1 (de) * 1980-09-22 1982-04-29 F. Hoffmann-La Roche & Co. AG, 4002 Basel Prostacycline

Citations (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2351112A1 (fr) * 1975-10-21 1977-12-09 Wellcome Found Derive de prostaglandine et medicament contenant ce derive
FR2351113A1 (fr) * 1976-05-11 1977-12-09 Wellcome Found Derives de prostaglandines et medicaments contenant ces derives
DE2724555A1 (de) * 1976-06-01 1977-12-15 Upjohn Co 5,6-dihydro-prostacyclin-analoge und verfahren zu deren herstellung
FR2359125A1 (fr) * 1976-02-04 1978-02-17 Upjohn Co Nouveaux derives de prostaglandine, leur procede de preparation et medicament les contenant
FR2376147A1 (fr) * 1976-12-31 1978-07-28 Erba Carlo Spa Prostaglandines bicycliques, utiles notamment comme anti-agglutinants des plaquettes sanguines et leur procede de preparation
FR2381043A1 (fr) * 1977-02-21 1978-09-15 Ono Pharmaceutical Co Nouveaux analogues de prostaglandines, leur preparation et les compositions pharmaceutiques qui les contiennent
FR2387777A1 (fr) * 1977-04-18 1978-11-17 Nixdorf Computer Ag Tete d'impression mosaique
FR2393800A1 (fr) * 1977-06-06 1979-01-05 Univ Chicago Nouvelles prostacyclines et leur procede de preparation et leur application en therapeutique
FR2401919A1 (fr) * 1977-07-28 1979-03-30 Upjohn Co Derives de prostaglandines
FR2404005A1 (fr) * 1977-09-22 1979-04-20 Ono Pharmaceutical Co Analogues de la prostaglandine i2 et compositions pharmaceutiques les contenant
FR2418794A1 (fr) * 1978-03-01 1979-09-28 Ono Pharmaceutical Co Analogues de la prostaglandine i2 et compositions pharmaceutiques les contenant

Patent Citations (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2351112A1 (fr) * 1975-10-21 1977-12-09 Wellcome Found Derive de prostaglandine et medicament contenant ce derive
FR2359125A1 (fr) * 1976-02-04 1978-02-17 Upjohn Co Nouveaux derives de prostaglandine, leur procede de preparation et medicament les contenant
FR2362833A1 (fr) * 1976-02-04 1978-03-24 Upjohn Co Nouveaux derives 5 de prostaglandine, leur procede de preparation et medicament les contenant
FR2362834A1 (fr) * 1976-02-04 1978-03-24 Upjohn Co Nouveaux derives 6-hemicetal ou 6-ceto de prostaglandine, leur procede de preparation et medicament les contenant
FR2351113A1 (fr) * 1976-05-11 1977-12-09 Wellcome Found Derives de prostaglandines et medicaments contenant ces derives
DE2724555A1 (de) * 1976-06-01 1977-12-15 Upjohn Co 5,6-dihydro-prostacyclin-analoge und verfahren zu deren herstellung
FR2376147A1 (fr) * 1976-12-31 1978-07-28 Erba Carlo Spa Prostaglandines bicycliques, utiles notamment comme anti-agglutinants des plaquettes sanguines et leur procede de preparation
FR2381043A1 (fr) * 1977-02-21 1978-09-15 Ono Pharmaceutical Co Nouveaux analogues de prostaglandines, leur preparation et les compositions pharmaceutiques qui les contiennent
FR2387777A1 (fr) * 1977-04-18 1978-11-17 Nixdorf Computer Ag Tete d'impression mosaique
FR2393800A1 (fr) * 1977-06-06 1979-01-05 Univ Chicago Nouvelles prostacyclines et leur procede de preparation et leur application en therapeutique
FR2401919A1 (fr) * 1977-07-28 1979-03-30 Upjohn Co Derives de prostaglandines
FR2401920A1 (fr) * 1977-07-28 1979-03-30 Upjohn Co Derives de prostaglandines
FR2401921A1 (fr) * 1977-07-28 1979-03-30 Upjohn Co Derives de prostaglandines
FR2404005A1 (fr) * 1977-09-22 1979-04-20 Ono Pharmaceutical Co Analogues de la prostaglandine i2 et compositions pharmaceutiques les contenant
FR2418794A1 (fr) * 1978-03-01 1979-09-28 Ono Pharmaceutical Co Analogues de la prostaglandine i2 et compositions pharmaceutiques les contenant

Non-Patent Citations (2)

* Cited by examiner, † Cited by third party
Title
EXBK/77 *
EXBK/78 *

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2401920A1 (fr) * 1977-07-28 1979-03-30 Upjohn Co Derives de prostaglandines

Also Published As

Publication number Publication date
IE780456L (en) 1978-09-07
BE864644A (fr) 1978-09-07
AU524786B2 (en) 1982-10-07
IE46570B1 (en) 1983-07-27
CH636353A5 (de) 1983-05-31
JPS53111041A (en) 1978-09-28
AU3335678A (en) 1979-08-23
GB1576570A (en) 1980-10-08
US4150222A (en) 1979-04-17
FR2401139A2 (fr) 1979-03-23
DE2809452A1 (de) 1978-09-14
NZ186516A (en) 1981-03-16
CA1159452A (fr) 1983-12-27
IL54176A0 (en) 1978-06-15

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