FR2401141A1 - Nouveaux derives halogenes de prostaglandines et medicaments les contenant - Google Patents
Nouveaux derives halogenes de prostaglandines et medicaments les contenantInfo
- Publication number
- FR2401141A1 FR2401141A1 FR7830488A FR7830488A FR2401141A1 FR 2401141 A1 FR2401141 A1 FR 2401141A1 FR 7830488 A FR7830488 A FR 7830488A FR 7830488 A FR7830488 A FR 7830488A FR 2401141 A1 FR2401141 A1 FR 2401141A1
- Authority
- FR
- France
- Prior art keywords
- prostaglandins
- halogen derivatives
- medicines containing
- new halogen
- new
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 229940094443 oxytocics prostaglandins Drugs 0.000 title abstract 2
- 150000003180 prostaglandins Chemical class 0.000 title abstract 2
- 239000003814 drug Chemical class 0.000 title 1
- 229910052736 halogen Inorganic materials 0.000 title 1
- 150000002367 halogens Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/93—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems condensed with a ring other than six-membered
- C07D307/935—Not further condensed cyclopenta [b] furans or hydrogenated cyclopenta [b] furans
- C07D307/937—Not further condensed cyclopenta [b] furans or hydrogenated cyclopenta [b] furans with hydrocarbon or substituted hydrocarbon radicals directly attached in position 2, e.g. prostacyclins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C405/00—Compounds containing a five-membered ring having two side-chains in ortho position to each other, and having oxygen atoms directly attached to the ring in ortho position to one of the side-chains, one side-chain containing, not directly attached to the ring, a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, and the other side-chain having oxygen atoms attached in gamma-position to the ring, e.g. prostaglandins ; Analogues or derivatives thereof
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Furan Compounds (AREA)
- Pyrane Compounds (AREA)
Abstract
L'invention se situe dans le domaine pharmaceutique. Elle concerne de nouveaux dérivés halogénés de prostaglandines ayant comme formule :
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US77500377A | 1977-03-07 | 1977-03-07 |
Publications (1)
Publication Number | Publication Date |
---|---|
FR2401141A1 true FR2401141A1 (fr) | 1979-03-23 |
Family
ID=25103006
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR7806484A Pending FR2401139A2 (fr) | 1977-03-07 | 1978-03-07 | Nouveaux derives d5 de prostaglandines, leur procede de preparation et medicaments les contenant |
FR7830488A Pending FR2401141A1 (fr) | 1977-03-07 | 1978-10-26 | Nouveaux derives halogenes de prostaglandines et medicaments les contenant |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR7806484A Pending FR2401139A2 (fr) | 1977-03-07 | 1978-03-07 | Nouveaux derives d5 de prostaglandines, leur procede de preparation et medicaments les contenant |
Country Status (12)
Country | Link |
---|---|
US (1) | US4150222A (fr) |
JP (1) | JPS53111041A (fr) |
AU (1) | AU524786B2 (fr) |
BE (1) | BE864644A (fr) |
CA (1) | CA1159452A (fr) |
CH (1) | CH636353A5 (fr) |
DE (1) | DE2809452A1 (fr) |
FR (2) | FR2401139A2 (fr) |
GB (1) | GB1576570A (fr) |
IE (1) | IE46570B1 (fr) |
IL (1) | IL54176A0 (fr) |
NZ (1) | NZ186516A (fr) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2401920A1 (fr) * | 1977-07-28 | 1979-03-30 | Upjohn Co | Derives de prostaglandines |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4215214A (en) * | 1976-08-23 | 1980-07-29 | The Upjohn Company | Enlarged-hetero-ring prostacyclin analogs with 5-halo feature |
FI71138C (fi) * | 1976-12-31 | 1986-11-24 | Erba Farmitalia | Foerfarande foer framstaellning av terapeutiskt aktiva bisykliska prostaglandiner |
IT1088036B (it) | 1977-11-25 | 1985-06-04 | Erba Carlo Spa | 15-epi-prostaciclina e prostaciclina analoghi |
DE2947526A1 (de) * | 1978-11-29 | 1980-06-12 | Ono Pharmaceutical Co | Prostacyclin-analoge |
DE2902809A1 (de) * | 1979-01-25 | 1980-08-07 | Hoechst Ag | Neue analoga von prostacyclin |
DE3029984C2 (de) * | 1980-08-08 | 1983-12-15 | Grünenthal GmbH, 5190 Stolberg | 2-Oxabicyclo [3.3.0] octanderivate und diese enthaltende Arzneimittel |
DE3035713A1 (de) * | 1980-09-22 | 1982-04-29 | F. Hoffmann-La Roche & Co. AG, 4002 Basel | Prostacycline |
Citations (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2351112A1 (fr) * | 1975-10-21 | 1977-12-09 | Wellcome Found | Derive de prostaglandine et medicament contenant ce derive |
FR2351113A1 (fr) * | 1976-05-11 | 1977-12-09 | Wellcome Found | Derives de prostaglandines et medicaments contenant ces derives |
DE2724555A1 (de) * | 1976-06-01 | 1977-12-15 | Upjohn Co | 5,6-dihydro-prostacyclin-analoge und verfahren zu deren herstellung |
FR2359125A1 (fr) * | 1976-02-04 | 1978-02-17 | Upjohn Co | Nouveaux derives de prostaglandine, leur procede de preparation et medicament les contenant |
FR2376147A1 (fr) * | 1976-12-31 | 1978-07-28 | Erba Carlo Spa | Prostaglandines bicycliques, utiles notamment comme anti-agglutinants des plaquettes sanguines et leur procede de preparation |
FR2381043A1 (fr) * | 1977-02-21 | 1978-09-15 | Ono Pharmaceutical Co | Nouveaux analogues de prostaglandines, leur preparation et les compositions pharmaceutiques qui les contiennent |
FR2387777A1 (fr) * | 1977-04-18 | 1978-11-17 | Nixdorf Computer Ag | Tete d'impression mosaique |
FR2393800A1 (fr) * | 1977-06-06 | 1979-01-05 | Univ Chicago | Nouvelles prostacyclines et leur procede de preparation et leur application en therapeutique |
FR2401919A1 (fr) * | 1977-07-28 | 1979-03-30 | Upjohn Co | Derives de prostaglandines |
FR2404005A1 (fr) * | 1977-09-22 | 1979-04-20 | Ono Pharmaceutical Co | Analogues de la prostaglandine i2 et compositions pharmaceutiques les contenant |
FR2418794A1 (fr) * | 1978-03-01 | 1979-09-28 | Ono Pharmaceutical Co | Analogues de la prostaglandine i2 et compositions pharmaceutiques les contenant |
-
1978
- 1978-02-16 AU AU33356/78A patent/AU524786B2/en not_active Expired
- 1978-02-20 NZ NZ186516A patent/NZ186516A/xx unknown
- 1978-03-01 CH CH223778A patent/CH636353A5/de not_active IP Right Cessation
- 1978-03-02 JP JP2289978A patent/JPS53111041A/ja active Pending
- 1978-03-02 GB GB8270/78A patent/GB1576570A/en not_active Expired
- 1978-03-02 IL IL54176A patent/IL54176A0/xx unknown
- 1978-03-04 DE DE19782809452 patent/DE2809452A1/de not_active Withdrawn
- 1978-03-06 IE IE456/78A patent/IE46570B1/en not_active IP Right Cessation
- 1978-03-06 CA CA000298279A patent/CA1159452A/fr not_active Expired
- 1978-03-07 FR FR7806484A patent/FR2401139A2/fr active Pending
- 1978-03-07 BE BE185731A patent/BE864644A/fr not_active IP Right Cessation
- 1978-06-05 US US05/912,552 patent/US4150222A/en not_active Expired - Lifetime
- 1978-10-26 FR FR7830488A patent/FR2401141A1/fr active Pending
Patent Citations (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2351112A1 (fr) * | 1975-10-21 | 1977-12-09 | Wellcome Found | Derive de prostaglandine et medicament contenant ce derive |
FR2359125A1 (fr) * | 1976-02-04 | 1978-02-17 | Upjohn Co | Nouveaux derives de prostaglandine, leur procede de preparation et medicament les contenant |
FR2362833A1 (fr) * | 1976-02-04 | 1978-03-24 | Upjohn Co | Nouveaux derives 5 de prostaglandine, leur procede de preparation et medicament les contenant |
FR2362834A1 (fr) * | 1976-02-04 | 1978-03-24 | Upjohn Co | Nouveaux derives 6-hemicetal ou 6-ceto de prostaglandine, leur procede de preparation et medicament les contenant |
FR2351113A1 (fr) * | 1976-05-11 | 1977-12-09 | Wellcome Found | Derives de prostaglandines et medicaments contenant ces derives |
DE2724555A1 (de) * | 1976-06-01 | 1977-12-15 | Upjohn Co | 5,6-dihydro-prostacyclin-analoge und verfahren zu deren herstellung |
FR2376147A1 (fr) * | 1976-12-31 | 1978-07-28 | Erba Carlo Spa | Prostaglandines bicycliques, utiles notamment comme anti-agglutinants des plaquettes sanguines et leur procede de preparation |
FR2381043A1 (fr) * | 1977-02-21 | 1978-09-15 | Ono Pharmaceutical Co | Nouveaux analogues de prostaglandines, leur preparation et les compositions pharmaceutiques qui les contiennent |
FR2387777A1 (fr) * | 1977-04-18 | 1978-11-17 | Nixdorf Computer Ag | Tete d'impression mosaique |
FR2393800A1 (fr) * | 1977-06-06 | 1979-01-05 | Univ Chicago | Nouvelles prostacyclines et leur procede de preparation et leur application en therapeutique |
FR2401919A1 (fr) * | 1977-07-28 | 1979-03-30 | Upjohn Co | Derives de prostaglandines |
FR2401920A1 (fr) * | 1977-07-28 | 1979-03-30 | Upjohn Co | Derives de prostaglandines |
FR2401921A1 (fr) * | 1977-07-28 | 1979-03-30 | Upjohn Co | Derives de prostaglandines |
FR2404005A1 (fr) * | 1977-09-22 | 1979-04-20 | Ono Pharmaceutical Co | Analogues de la prostaglandine i2 et compositions pharmaceutiques les contenant |
FR2418794A1 (fr) * | 1978-03-01 | 1979-09-28 | Ono Pharmaceutical Co | Analogues de la prostaglandine i2 et compositions pharmaceutiques les contenant |
Non-Patent Citations (2)
Title |
---|
EXBK/77 * |
EXBK/78 * |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2401920A1 (fr) * | 1977-07-28 | 1979-03-30 | Upjohn Co | Derives de prostaglandines |
Also Published As
Publication number | Publication date |
---|---|
IE780456L (en) | 1978-09-07 |
BE864644A (fr) | 1978-09-07 |
AU524786B2 (en) | 1982-10-07 |
IE46570B1 (en) | 1983-07-27 |
CH636353A5 (de) | 1983-05-31 |
JPS53111041A (en) | 1978-09-28 |
AU3335678A (en) | 1979-08-23 |
GB1576570A (en) | 1980-10-08 |
US4150222A (en) | 1979-04-17 |
FR2401139A2 (fr) | 1979-03-23 |
DE2809452A1 (de) | 1978-09-14 |
NZ186516A (en) | 1981-03-16 |
CA1159452A (fr) | 1983-12-27 |
IL54176A0 (en) | 1978-06-15 |
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