FR2282893A1 - Derives de thienothiazine utiles en tant que medicaments et leur procede de preparation - Google Patents

Derives de thienothiazine utiles en tant que medicaments et leur procede de preparation

Info

Publication number
FR2282893A1
FR2282893A1 FR7525999A FR7525999A FR2282893A1 FR 2282893 A1 FR2282893 A1 FR 2282893A1 FR 7525999 A FR7525999 A FR 7525999A FR 7525999 A FR7525999 A FR 7525999A FR 2282893 A1 FR2282893 A1 FR 2282893A1
Authority
FR
France
Prior art keywords
useful
preparation process
medicinal products
thienothiazine derivatives
thienothiazine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7525999A
Other languages
English (en)
French (fr)
Other versions
FR2282893B1 (no
Inventor
Otto Hromatka
Dieter Binder
Rudolf Pfister
Paul Zeller
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
F Hoffmann La Roche AG
Original Assignee
F Hoffmann La Roche AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from CH1158274A external-priority patent/CH608500A5/de
Priority claimed from CH1215774A external-priority patent/CH608501A5/de
Application filed by F Hoffmann La Roche AG filed Critical F Hoffmann La Roche AG
Publication of FR2282893A1 publication Critical patent/FR2282893A1/fr
Application granted granted Critical
Publication of FR2282893B1 publication Critical patent/FR2282893B1/fr
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/30—Hetero atoms other than halogen
    • C07D333/34—Sulfur atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Manufacturing Of Printed Wiring (AREA)
  • Electroplating Methods And Accessories (AREA)
FR7525999A 1974-08-26 1975-08-22 Derives de thienothiazine utiles en tant que medicaments et leur procede de preparation Granted FR2282893A1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH1158274A CH608500A5 (en) 1974-08-26 1974-08-26 Process for the preparation of thiazine derivatives
CH1215774A CH608501A5 (en) 1974-09-09 1974-09-09 Process for the preparation of thiazine derivatives

Publications (2)

Publication Number Publication Date
FR2282893A1 true FR2282893A1 (fr) 1976-03-26
FR2282893B1 FR2282893B1 (no) 1980-05-16

Family

ID=25708582

Family Applications (3)

Application Number Title Priority Date Filing Date
FR7525999A Granted FR2282893A1 (fr) 1974-08-26 1975-08-22 Derives de thienothiazine utiles en tant que medicaments et leur procede de preparation
FR7615425A Granted FR2309558A1 (fr) 1974-08-26 1976-05-21 Derives de thienothiazine et leurs procedes de preparation
FR7615424A Granted FR2303803A1 (fr) 1974-08-26 1976-05-21 Acides sulfothiophene-carboxyliques et leur procede de preparation

Family Applications After (2)

Application Number Title Priority Date Filing Date
FR7615425A Granted FR2309558A1 (fr) 1974-08-26 1976-05-21 Derives de thienothiazine et leurs procedes de preparation
FR7615424A Granted FR2303803A1 (fr) 1974-08-26 1976-05-21 Acides sulfothiophene-carboxyliques et leur procede de preparation

Country Status (20)

Country Link
JP (1) JPS5826758B2 (no)
AR (1) AR216288A1 (no)
AT (1) AT350064B (no)
BR (1) BR7505463A (no)
DD (1) DD124119A5 (no)
DE (1) DE2537070A1 (no)
DK (1) DK137835B (no)
FI (1) FI59253C (no)
FR (3) FR2282893A1 (no)
GB (1) GB1519811A (no)
HU (1) HU173739B (no)
IE (1) IE41457B1 (no)
IL (1) IL47877A (no)
LU (2) LU73257A1 (no)
NL (2) NL183582C (no)
NO (1) NO146096C (no)
PL (1) PL106076B1 (no)
SE (1) SE412066B (no)
SU (1) SU603338A3 (no)
YU (1) YU40266B (no)

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2704485A1 (de) * 1977-02-03 1978-08-10 Thomae Gmbh Dr K Neue 2,5-dihydro-1,2-thiazino eckige klammer auf 5,6-b eckige klammer zu indol-3-carboxamid-1,1-dioxide, verfahren zu ihrer herstellung und diese enthaltende arzneimittel
EP0001113A1 (de) * 1977-09-06 1979-03-21 F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft Thienothiazinderivate, deren Herstellung, sowie diese enthaltende Präparate
FR2401167A1 (fr) * 1977-08-22 1979-03-23 Hoffmann La Roche Derives de thienothiazine utiles comme medicaments
FR2401927A1 (fr) * 1977-09-06 1979-03-30 Hoffmann La Roche Derives de thiazine utiles comme medicaments

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2838377A1 (de) * 1978-09-02 1980-03-20 Thomae Gmbh Dr K Neue 4-hydroxy-2h eckige klammer auf 1 eckige klammer zu benzothieno eckige klammer auf 2,3-e eckige klammer zu -1,2- thiazin-3-carboxamid-1,1-dioxide sowie deren salze, deren verwendung und verfahren zu ihrer herstellung
AU5811280A (en) * 1979-06-13 1980-12-18 F. Hoffmann-La Roche Ag Thiazine derivatives
JPS58109492A (ja) * 1981-12-22 1983-06-29 Mitsui Toatsu Chem Inc チエノチアジン誘導体およびそれを含有する医薬組成物
ATE26720T1 (de) * 1982-09-09 1987-05-15 Hoffmann La Roche Thieno(2,3-e)-1,2-thiazin-derivate.
JPS60163533U (ja) * 1984-04-02 1985-10-30 ホシデン株式会社 リ−ル台の制動装置
JPH0318748Y2 (no) * 1985-12-18 1991-04-19
ATA39088A (de) 1988-02-18 1990-06-15 Binder Dieter Dr Basisch substituierte thienoisothiazol-3(2h)-on-1,1-dioxide und ihre pharmazeutisch vertraeglichen salze, verfahren zu ihrer herstellung und ihre verwendung
AT400568B (de) * 1994-05-18 1996-01-25 Chem Pharm Forsch Gmbh Neue n-heterocyclische thienothiazincarboxamide, verfahren zu ihrer herstellung und ihre verwendung
AT400437B (de) * 1993-12-14 1995-12-27 Chem Pharm Forsch Gmbh Neue n-heterocyclische thienothiazincarboxamide, verfahren zu ihrer herstellung und ihre verwendung
EP0658559A1 (de) * 1993-12-14 1995-06-21 Chemisch Pharmazeutische Forschungsgesellschaft m.b.H. Thienothiazinderivate, Verfahren zu ihrer Herstellung und ihre Verwendung als 5-dipoxygenase und Cyclooxygenaseinhibitoren
US5538966A (en) * 1994-01-21 1996-07-23 Alcon Laboratories, Inc. Carbonic anhydrase inhibitors
IT1308633B1 (it) 1999-03-02 2002-01-09 Nicox Sa Nitrossiderivati.
CN1171892C (zh) * 2001-06-25 2004-10-20 李晶 具有抗炎镇痛活性的噻吩并噻嗪化合物及其制备方法和用途

Cited By (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2704485A1 (de) * 1977-02-03 1978-08-10 Thomae Gmbh Dr K Neue 2,5-dihydro-1,2-thiazino eckige klammer auf 5,6-b eckige klammer zu indol-3-carboxamid-1,1-dioxide, verfahren zu ihrer herstellung und diese enthaltende arzneimittel
FR2379542A1 (fr) * 1977-02-03 1978-09-01 Thomae Gmbh Dr K Nouveaux 1,1-dioxydes de 2,5-dihydro-1,2-thiazino (5,6-b) indole-3-carboxamides, procedes pour leur preparation et medicaments les renfermant
FR2401167A1 (fr) * 1977-08-22 1979-03-23 Hoffmann La Roche Derives de thienothiazine utiles comme medicaments
US4187303A (en) 1977-08-22 1980-02-05 Hoffmann-La Roche Inc. Thiazine derivatives
EP0001113A1 (de) * 1977-09-06 1979-03-21 F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft Thienothiazinderivate, deren Herstellung, sowie diese enthaltende Präparate
FR2401927A1 (fr) * 1977-09-06 1979-03-30 Hoffmann La Roche Derives de thiazine utiles comme medicaments

Also Published As

Publication number Publication date
DK381175A (no) 1976-02-27
NO752932L (no) 1976-02-27
DD124119A5 (no) 1977-02-02
AT350064B (de) 1979-05-10
AU8418675A (en) 1977-02-24
FI59253B (fi) 1981-03-31
HU173739B (hu) 1979-08-28
FI752398A (no) 1976-02-27
DK137835C (no) 1978-10-16
SU603338A3 (ru) 1978-04-15
FR2282893B1 (no) 1980-05-16
FI59253C (fi) 1981-07-10
DK137835B (da) 1978-05-16
IL47877A (en) 1978-10-31
LU73257A1 (no) 1977-04-15
FR2303803A1 (fr) 1976-10-08
JPS5826758B2 (ja) 1983-06-04
YU216675A (en) 1982-08-31
IE41457B1 (en) 1980-01-02
LU88312I2 (de) 1994-09-09
NL183582C (nl) 1988-12-01
IE41457L (en) 1976-02-26
IL47877A0 (en) 1975-11-25
FR2303803B1 (no) 1979-07-13
NL183582B (nl) 1988-07-01
ATA655975A (de) 1978-10-15
SE412066B (sv) 1980-02-18
YU40266B (en) 1985-12-31
DE2537070C2 (no) 1987-06-25
NL930080I1 (nl) 1993-09-16
GB1519811A (en) 1978-08-02
FR2309558B1 (no) 1979-05-04
NO146096B (no) 1982-04-19
SE7509446L (sv) 1976-02-27
BR7505463A (pt) 1976-08-03
AR216288A1 (es) 1979-12-14
NO146096C (no) 1982-07-28
JPS5148694A (no) 1976-04-26
NL930080I2 (nl) 1994-01-03
FR2309558A1 (fr) 1976-11-26
PL106076B1 (pl) 1979-11-30
DE2537070A1 (de) 1976-03-18
NL7510057A (nl) 1976-03-01

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Legal Events

Date Code Title Description
TP Transmission of property
CC Supplementary protection certificate (spc) laid open to the public (law of 25 june 1990)

Free format text: 92C0154, 920504

CB Supplementary protection certificate (spc) granted (law of 25 june 1990)

Free format text: 92C0154, 750822

CL Concession to grant licences