BE768137A - Derives de piperazinyl-alcoyl-quinazolone-(4), leur procede de preparation et medicaments en contenant - Google Patents
Derives de piperazinyl-alcoyl-quinazolone-(4), leur procede de preparation et medicaments en contenantInfo
- Publication number
- BE768137A BE768137A BE768137A BE768137A BE768137A BE 768137 A BE768137 A BE 768137A BE 768137 A BE768137 A BE 768137A BE 768137 A BE768137 A BE 768137A BE 768137 A BE768137 A BE 768137A
- Authority
- BE
- Belgium
- Prior art keywords
- alcoyl
- quinazolone
- piperazinyl
- derivatives
- preparation process
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19702027645 DE2027645A1 (de) | 1970-06-05 | 1970-06-05 | Piperazinylalkyl chinazolon (4) den vate, Verfahren zu deren Herstellung und sie enthaltende Arzneimittel |
Publications (1)
Publication Number | Publication Date |
---|---|
BE768137A true BE768137A (fr) | 1971-12-06 |
Family
ID=5773104
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BE768137A BE768137A (fr) | 1970-06-05 | 1971-06-04 | Derives de piperazinyl-alcoyl-quinazolone-(4), leur procede de preparation et medicaments en contenant |
Country Status (10)
Country | Link |
---|---|
US (1) | US3984555A (fr) |
AT (3) | AT318628B (fr) |
BE (1) | BE768137A (fr) |
CA (1) | CA951319A (fr) |
CH (3) | CH558374A (fr) |
DE (1) | DE2027645A1 (fr) |
FR (1) | FR2100726B1 (fr) |
GB (1) | GB1331522A (fr) |
LU (1) | LU63267A1 (fr) |
NL (1) | NL7107695A (fr) |
Families Citing this family (32)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4287341A (en) * | 1979-11-01 | 1981-09-01 | Pfizer Inc. | Alkoxy-substituted-6-chloro-quinazoline-2,4-diones |
US6723727B1 (en) * | 1996-12-20 | 2004-04-20 | Hoechst Aktiengesellschaft | Substituted purine derivatives, processes for their preparation, their use, and compositions comprising them |
DE69842109D1 (de) * | 1997-08-21 | 2011-03-10 | Shiseido Co Ltd | Chinazolin-4-on Derivate, deren Herstellung und deren Verwendung als Haarwuchsmittel oder in äusserlich anzuwendenden Hautpflegemitteln |
EP1216243A1 (fr) * | 1999-10-01 | 2002-06-26 | Advanced Medicine, Inc. | Quinazolinones et analogues et leur utilisation comme anesthesiques locaux |
WO2001081346A2 (fr) * | 2000-04-25 | 2001-11-01 | Icos Corporation | Inhibiteurs de la phosphatidyl-inositol 3-kinase delta humaine |
US6667300B2 (en) | 2000-04-25 | 2003-12-23 | Icos Corporation | Inhibitors of human phosphatidylinositol 3-kinase delta |
AUPR201600A0 (en) * | 2000-12-11 | 2001-01-11 | Fujisawa Pharmaceutical Co., Ltd. | Quinazolinone derivative |
EP2116248A1 (fr) | 2001-09-05 | 2009-11-11 | Minerva Biotechnologies Corporation | Compositions et procédés pour le traitement du cancer |
US20030119834A1 (en) * | 2001-09-05 | 2003-06-26 | Bamdad Cynthia C. | Compositions and methods of treatment of cancer |
AU2002363429B2 (en) * | 2001-11-07 | 2008-05-08 | Merck & Co., Inc. | Mitotic kinesin inhibitors |
AUPS019702A0 (en) * | 2002-01-29 | 2002-02-21 | Fujisawa Pharmaceutical Co., Ltd. | Condensed heterocyclic compounds |
JP2005536553A (ja) * | 2002-08-21 | 2005-12-02 | サイトキネティクス・インコーポレーテッド | 化合物、組成物および方法 |
CA2502302A1 (fr) * | 2002-11-04 | 2004-05-21 | Nps Pharmaceuticals, Inc. | Composes de quinazolinone utilises comme calcilytiques |
DE602004022819D1 (de) * | 2003-06-06 | 2009-10-08 | Vertex Pharma | Von atp-bindende kassette transportern |
WO2005016348A1 (fr) * | 2003-08-14 | 2005-02-24 | Icos Corporation | Methodes d'inhibition de reponses immunes stimulees par un facteur endogene |
US20050054614A1 (en) * | 2003-08-14 | 2005-03-10 | Diacovo Thomas G. | Methods of inhibiting leukocyte accumulation |
US7932260B2 (en) | 2004-05-13 | 2011-04-26 | Icos Corporation | Quinazolinones as inhibitors of human phosphatidylinositol 3-kinase delta |
EP1755609A1 (fr) * | 2004-05-25 | 2007-02-28 | Icos Corporation | Methodes de traitement et/ou de prevention de la proliferation aberrante des cellules hematopoietiques |
CA2598409A1 (fr) * | 2005-02-17 | 2006-08-24 | Icos Corporation | Procede d'inhibition d'accumulation de leucocytes |
WO2007110868A2 (fr) * | 2006-03-28 | 2007-10-04 | Atir Holding S.A. | Composés hétérocycliques et leurs utilisations dans le traitement de troubles sexuels |
CA2975473C (fr) | 2008-11-13 | 2021-01-19 | Gilead Calistoga Llc | Therapies pour tumeurs malignes hematologiques |
US9492449B2 (en) | 2008-11-13 | 2016-11-15 | Gilead Calistoga Llc | Therapies for hematologic malignancies |
JP2012521994A (ja) | 2009-03-24 | 2012-09-20 | ギリアード カリストガ エルエルシー | 2−プリニル−3−トリル−キナゾリノン誘導体のアトロプ異性体および使用方法 |
ES2548253T3 (es) * | 2009-04-20 | 2015-10-15 | Gilead Calistoga Llc | Métodos para el tratamiento de tumores sólidos |
CA2768843A1 (fr) | 2009-07-21 | 2011-01-27 | Gilead Calistoga Llc | Traitement de troubles du foie par des inhibiteurs de pi3k |
BRPI1003506B1 (pt) | 2010-09-24 | 2019-12-03 | Ache Int Bvi Ltd | composto alquil-piperazino-fenil-4(3h)quinazolinonas e uso do composto alquil-piperazino-fenil-4(3h)quinazolinonas associado aos receptores serotoninérgicos 5-ht1a e 5-ht2a |
EP3581567A1 (fr) * | 2011-04-10 | 2019-12-18 | Atir Holding S.A. | Composés hétérocycliques et leurs utilisations dans le traitement de troubles sexuels |
WO2013134288A1 (fr) | 2012-03-05 | 2013-09-12 | Gilead Calistoga Llc | Formes polymorphes de l'acide -2-(1-(9h-purine-6-ylamino)propyl)-5-fluoro-3-phénylquinazolin-4(3h)-one |
US9359367B2 (en) | 2012-07-09 | 2016-06-07 | Lupin Limited | Tetrahydroquinazolinone derivatives as PARP inhibitors |
JP2017502021A (ja) | 2013-12-20 | 2017-01-19 | ギリアード カリストガ エルエルシー | ホスファチジルイノシトール3−キナーゼ阻害剤のためのプロセス方法 |
AU2014364414A1 (en) | 2013-12-20 | 2016-06-30 | Gilead Calistoga Llc | Polymorphic forms of a hydrochloride salt of (S) -2-(1-(9H-purin-6-ylamino) propyl) -5-fluoro-3-phenylquinazolin-4 (3H) -one |
EP3154960A1 (fr) | 2014-06-13 | 2017-04-19 | Gilead Sciences, Inc. | Inhibiteurs de la phosphatidylinositol 3-kinase |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1053063A (fr) * | 1963-05-18 |
-
1970
- 1970-06-05 DE DE19702027645 patent/DE2027645A1/de active Pending
-
1971
- 1971-05-28 US US05/148,100 patent/US3984555A/en not_active Expired - Lifetime
- 1971-06-01 AT AT244173A patent/AT318628B/de not_active IP Right Cessation
- 1971-06-01 AT AT244273A patent/AT317899B/de not_active IP Right Cessation
- 1971-06-01 AT AT470571A patent/AT318615B/de not_active IP Right Cessation
- 1971-06-02 LU LU63267D patent/LU63267A1/xx unknown
- 1971-06-02 CH CH450074A patent/CH558374A/xx not_active IP Right Cessation
- 1971-06-02 CH CH450174A patent/CH569732A5/xx not_active IP Right Cessation
- 1971-06-02 CH CH802071A patent/CH557829A/xx not_active IP Right Cessation
- 1971-06-03 GB GB1880371*[A patent/GB1331522A/en not_active Expired
- 1971-06-03 CA CA114,709,A patent/CA951319A/en not_active Expired
- 1971-06-04 FR FR7120368A patent/FR2100726B1/fr not_active Expired
- 1971-06-04 BE BE768137A patent/BE768137A/fr unknown
- 1971-06-04 NL NL7107695A patent/NL7107695A/xx unknown
Also Published As
Publication number | Publication date |
---|---|
AT317899B (de) | 1974-09-25 |
CH557829A (de) | 1975-01-15 |
US3984555A (en) | 1976-10-05 |
CH558374A (de) | 1975-01-31 |
AT318628B (de) | 1974-11-11 |
LU63267A1 (fr) | 1972-08-23 |
CA951319A (en) | 1974-07-16 |
NL7107695A (fr) | 1971-12-07 |
AT318615B (de) | 1974-11-11 |
FR2100726B1 (fr) | 1975-10-10 |
FR2100726A1 (fr) | 1972-03-24 |
DE2027645A1 (de) | 1971-12-09 |
CH569732A5 (fr) | 1975-11-28 |
GB1331522A (en) | 1973-09-26 |
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