NL7107695A - - Google Patents

Info

Publication number
NL7107695A
NL7107695A NL7107695A NL7107695A NL7107695A NL 7107695 A NL7107695 A NL 7107695A NL 7107695 A NL7107695 A NL 7107695A NL 7107695 A NL7107695 A NL 7107695A NL 7107695 A NL7107695 A NL 7107695A
Authority
NL
Netherlands
Application number
NL7107695A
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of NL7107695A publication Critical patent/NL7107695A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
NL7107695A 1970-06-05 1971-06-04 NL7107695A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19702027645 DE2027645A1 (de) 1970-06-05 1970-06-05 Piperazinylalkyl chinazolon (4) den vate, Verfahren zu deren Herstellung und sie enthaltende Arzneimittel

Publications (1)

Publication Number Publication Date
NL7107695A true NL7107695A (fr) 1971-12-07

Family

ID=5773104

Family Applications (1)

Application Number Title Priority Date Filing Date
NL7107695A NL7107695A (fr) 1970-06-05 1971-06-04

Country Status (10)

Country Link
US (1) US3984555A (fr)
AT (3) AT318628B (fr)
BE (1) BE768137A (fr)
CA (1) CA951319A (fr)
CH (3) CH569732A5 (fr)
DE (1) DE2027645A1 (fr)
FR (1) FR2100726B1 (fr)
GB (1) GB1331522A (fr)
LU (1) LU63267A1 (fr)
NL (1) NL7107695A (fr)

Families Citing this family (32)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4287341A (en) * 1979-11-01 1981-09-01 Pfizer Inc. Alkoxy-substituted-6-chloro-quinazoline-2,4-diones
US6723727B1 (en) * 1996-12-20 2004-04-20 Hoechst Aktiengesellschaft Substituted purine derivatives, processes for their preparation, their use, and compositions comprising them
EP0903344B1 (fr) * 1997-08-21 2011-01-26 Shiseido Co., Ltd. Dérivés de quinazolin-4-one, leur préparation et leur utilisation comme agents favorisant la croissance des cheveux ou dans une composition pour la peau à usage externe
EP1216242A1 (fr) 1999-10-01 2002-06-26 Advanced Medicine, Inc. Quinazolinones macrocycliques et leur utilisation en tant qu'anesthesiques locaux
US6667300B2 (en) * 2000-04-25 2003-12-23 Icos Corporation Inhibitors of human phosphatidylinositol 3-kinase delta
EP1278748B1 (fr) * 2000-04-25 2011-03-23 ICOS Corporation Inhibiteurs de la phosphatidyl-inositol 3-kinase delta humaine
AUPR201600A0 (en) * 2000-12-11 2001-01-11 Fujisawa Pharmaceutical Co., Ltd. Quinazolinone derivative
WO2003020280A2 (fr) * 2001-09-05 2003-03-13 Minerva Biotechnologies Corporation Compositions et methodes de traitement du cancer
EP2329822A1 (fr) 2001-09-05 2011-06-08 Minerva Biotechnologies Corporation Compositions et procédés pour le traitement du cancer
EP1444209A4 (fr) 2001-11-07 2005-02-16 Merck & Co Inc Inhibiteurs de la kinesine mitotique
AUPS019702A0 (en) * 2002-01-29 2002-02-21 Fujisawa Pharmaceutical Co., Ltd. Condensed heterocyclic compounds
JP2005536553A (ja) * 2002-08-21 2005-12-02 サイトキネティクス・インコーポレーテッド 化合物、組成物および方法
JP2006512315A (ja) * 2002-11-04 2006-04-13 エヌピーエス ファーマスーティカルズ インコーポレイテッド カルシリティックとしてのキナゾリノン化合物
EP1646615B1 (fr) * 2003-06-06 2009-08-26 Vertex Pharmaceuticals Incorporated Derives de pyrimidne utilises en tant que modulateurs de transporteurs de cassette de liaison a l'atp
US20050054614A1 (en) * 2003-08-14 2005-03-10 Diacovo Thomas G. Methods of inhibiting leukocyte accumulation
US20050043239A1 (en) * 2003-08-14 2005-02-24 Jason Douangpanya Methods of inhibiting immune responses stimulated by an endogenous factor
EP1761540B1 (fr) * 2004-05-13 2016-09-28 Icos Corporation Quinazolinones utilisees en tant qu'inhibiteurs de la phosphatidylinositol 3-kinase delta humaine
EP1755609A1 (fr) * 2004-05-25 2007-02-28 Icos Corporation Methodes de traitement et/ou de prevention de la proliferation aberrante des cellules hematopoietiques
AU2006214190A1 (en) * 2005-02-17 2006-08-24 Icos Corporation Phosphoinositide 3-kinase inhibitors for inhibiting leukocyte accumulation
EP2233472B1 (fr) * 2006-03-28 2014-01-15 Atir Holding S.A. Composés hétérocycliques et leurs utilisations dans le traitement de troubles sexuels
US9492449B2 (en) 2008-11-13 2016-11-15 Gilead Calistoga Llc Therapies for hematologic malignancies
CA3092449A1 (fr) 2008-11-13 2010-05-20 Gilead Calistoga Llc Therapies pour tumeurs malignes hematologiques
MX2011009955A (es) 2009-03-24 2011-11-18 Gilead Calistoga Llc Atropisomeros de derivados de 2-purinil-3-tolil-quinazolinona y metodos de uso.
CN102458410A (zh) * 2009-04-20 2012-05-16 吉联亚·卡利斯托加有限责任公司 治疗实体瘤的方法
MX2012000817A (es) 2009-07-21 2012-05-08 Gilead Calistoga Llc Tratamiento para desordenes del higado con inhibidores pi3k.
BRPI1003506B1 (pt) 2010-09-24 2019-12-03 Ache Int Bvi Ltd composto alquil-piperazino-fenil-4(3h)quinazolinonas e uso do composto alquil-piperazino-fenil-4(3h)quinazolinonas associado aos receptores serotoninérgicos 5-ht1a e 5-ht2a
US9353067B2 (en) 2011-04-10 2016-05-31 Atir Holding S.A. Heterocyclic compounds and uses thereof in the treatment of sexual disorders
AU2013203620B2 (en) 2012-03-05 2015-11-19 Gilead Calistoga Llc Polymorphic forms of (S)-2-(1-(9H-purin-6-ylamino)propyl)-5-fluoro-3-phenylquinazolin-4(3H)-one
ES2595240T3 (es) 2012-07-09 2016-12-28 Lupin Limited Derivados de tetrahidroquinazolinona como inhibidores de PARP
PL3083630T3 (pl) 2013-12-20 2020-02-28 Gilead Calistoga Llc Sposoby otrzymywania inhibitorów 3-kinazy fosfatydyloinozytolu
JP2017500319A (ja) 2013-12-20 2017-01-05 ギリアード カリストガ エルエルシー (s)−2−(1−(9h−プリン−6−イルアミノ)プロピル)−5−フルオロ−3−フェニルキナゾリン−4(3h)−オンの塩酸塩の多形形態
NZ726360A (en) 2014-06-13 2018-04-27 Gilead Sciences Inc Phosphatidylinositol 3-kinase inhibitors

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1249281B (fr) * 1963-05-18

Also Published As

Publication number Publication date
US3984555A (en) 1976-10-05
DE2027645A1 (de) 1971-12-09
FR2100726B1 (fr) 1975-10-10
BE768137A (fr) 1971-12-06
AT318615B (de) 1974-11-11
FR2100726A1 (fr) 1972-03-24
CH557829A (de) 1975-01-15
CA951319A (en) 1974-07-16
CH569732A5 (fr) 1975-11-28
LU63267A1 (fr) 1972-08-23
AT317899B (de) 1974-09-25
GB1331522A (en) 1973-09-26
CH558374A (de) 1975-01-31
AT318628B (de) 1974-11-11

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