CH569732A5 - - Google Patents

Info

Publication number
CH569732A5
CH569732A5 CH450174A CH450174A CH569732A5 CH 569732 A5 CH569732 A5 CH 569732A5 CH 450174 A CH450174 A CH 450174A CH 450174 A CH450174 A CH 450174A CH 569732 A5 CH569732 A5 CH 569732A5
Authority
CH
Switzerland
Application number
CH450174A
Original Assignee
Byk Gulden Lomberg Chem Fab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Byk Gulden Lomberg Chem Fab filed Critical Byk Gulden Lomberg Chem Fab
Publication of CH569732A5 publication Critical patent/CH569732A5/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CH450174A 1970-06-05 1971-06-02 CH569732A5 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19702027645 DE2027645A1 (de) 1970-06-05 1970-06-05 Piperazinylalkyl chinazolon (4) den vate, Verfahren zu deren Herstellung und sie enthaltende Arzneimittel

Publications (1)

Publication Number Publication Date
CH569732A5 true CH569732A5 (fr) 1975-11-28

Family

ID=5773104

Family Applications (3)

Application Number Title Priority Date Filing Date
CH450074A CH558374A (de) 1970-06-05 1971-06-02 Verfahren zur herstellung von arylsubstituierten piperazinylalkyl- bezw. alkenyl- chinazolon-(4)-derivaten.
CH450174A CH569732A5 (fr) 1970-06-05 1971-06-02
CH802071A CH557829A (de) 1970-06-05 1971-06-02 Verfahren zur herstellung von arylsubstituierten piperazinyl-alkyl- bzw. -alkenyl-chinazolon-(4)-derivaten.

Family Applications Before (1)

Application Number Title Priority Date Filing Date
CH450074A CH558374A (de) 1970-06-05 1971-06-02 Verfahren zur herstellung von arylsubstituierten piperazinylalkyl- bezw. alkenyl- chinazolon-(4)-derivaten.

Family Applications After (1)

Application Number Title Priority Date Filing Date
CH802071A CH557829A (de) 1970-06-05 1971-06-02 Verfahren zur herstellung von arylsubstituierten piperazinyl-alkyl- bzw. -alkenyl-chinazolon-(4)-derivaten.

Country Status (10)

Country Link
US (1) US3984555A (fr)
AT (3) AT318615B (fr)
BE (1) BE768137A (fr)
CA (1) CA951319A (fr)
CH (3) CH558374A (fr)
DE (1) DE2027645A1 (fr)
FR (1) FR2100726B1 (fr)
GB (1) GB1331522A (fr)
LU (1) LU63267A1 (fr)
NL (1) NL7107695A (fr)

Families Citing this family (32)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4287341A (en) * 1979-11-01 1981-09-01 Pfizer Inc. Alkoxy-substituted-6-chloro-quinazoline-2,4-diones
US6723727B1 (en) * 1996-12-20 2004-04-20 Hoechst Aktiengesellschaft Substituted purine derivatives, processes for their preparation, their use, and compositions comprising them
EP0903344B1 (fr) * 1997-08-21 2011-01-26 Shiseido Co., Ltd. Dérivés de quinazolin-4-one, leur préparation et leur utilisation comme agents favorisant la croissance des cheveux ou dans une composition pour la peau à usage externe
WO2001025234A1 (fr) * 1999-10-01 2001-04-12 Advanced Medicine, Inc. Quinazolinones et analogues et leur utilisation comme anesthesiques locaux
US6667300B2 (en) * 2000-04-25 2003-12-23 Icos Corporation Inhibitors of human phosphatidylinositol 3-kinase delta
KR100785363B1 (ko) * 2000-04-25 2007-12-18 이코스 코포레이션 인간 포스파티딜-이노시톨 3-키나제 델타의 억제제
AUPR201600A0 (en) * 2000-12-11 2001-01-11 Fujisawa Pharmaceutical Co., Ltd. Quinazolinone derivative
WO2003020280A2 (fr) * 2001-09-05 2003-03-13 Minerva Biotechnologies Corporation Compositions et methodes de traitement du cancer
ATE469648T1 (de) 2001-09-05 2010-06-15 Minerva Biotechnologies Corp Zusammensetzungen und deren verwendung zur behandlung von krebs
AU2002363429B2 (en) * 2001-11-07 2008-05-08 Merck & Co., Inc. Mitotic kinesin inhibitors
AUPS019702A0 (en) * 2002-01-29 2002-02-21 Fujisawa Pharmaceutical Co., Ltd. Condensed heterocyclic compounds
US20040048853A1 (en) * 2002-08-21 2004-03-11 Gustave Bergnes Compounds, compositions, and methods
WO2004041755A2 (fr) * 2002-11-04 2004-05-21 Nps Pharmaceuticals, Inc. Composes de quinazolinone utilises comme calcilytiques
WO2004111014A1 (fr) * 2003-06-06 2004-12-23 Vertex Pharmaceuticals Incorporated Derives de pyrimidne utilises en tant que modulateurs de transporteurs de cassette de liaison a l'atp
WO2005016348A1 (fr) * 2003-08-14 2005-02-24 Icos Corporation Methodes d'inhibition de reponses immunes stimulees par un facteur endogene
US20050054614A1 (en) * 2003-08-14 2005-03-10 Diacovo Thomas G. Methods of inhibiting leukocyte accumulation
CA2566609C (fr) 2004-05-13 2012-06-26 Icos Corporation Quinazolinones utilisees en tant qu'inhibiteurs de la phosphatidylinositol 3-kinase delta humaine
CA2567883A1 (fr) * 2004-05-25 2005-12-15 Icos Corporation Methodes de traitement et/ou de prevention de la proliferation aberrante des cellules hematopoietiques
EP1885356A2 (fr) * 2005-02-17 2008-02-13 Icos Corporation Inhibiteurs de la phosphoinositide 3-kinase pour inhiber l'accumulation des leucocytes
WO2007110868A2 (fr) * 2006-03-28 2007-10-04 Atir Holding S.A. Composés hétérocycliques et leurs utilisations dans le traitement de troubles sexuels
NZ611764A (en) 2008-11-13 2015-01-30 Gilead Calistoga Llc Therapies for hematologic malignancies
US9492449B2 (en) 2008-11-13 2016-11-15 Gilead Calistoga Llc Therapies for hematologic malignancies
EA019499B1 (ru) 2009-03-24 2014-04-30 ГИЛИЭД КАЛИСТОГА ЭлЭлСи Производные атропоизомеров 2-пуринил-3-толилхиназолинона и способы применения
SG175259A1 (en) * 2009-04-20 2011-11-28 Gilead Calistoga Llc Methods of treatment for solid tumors
WO2011011550A1 (fr) 2009-07-21 2011-01-27 Calistoga Pharmaceuticals Inc. Traitement de troubles du foie par des inhibiteurs de pi3k
BRPI1003506B1 (pt) 2010-09-24 2019-12-03 Ache Int Bvi Ltd composto alquil-piperazino-fenil-4(3h)quinazolinonas e uso do composto alquil-piperazino-fenil-4(3h)quinazolinonas associado aos receptores serotoninérgicos 5-ht1a e 5-ht2a
US9353067B2 (en) 2011-04-10 2016-05-31 Atir Holding S.A. Heterocyclic compounds and uses thereof in the treatment of sexual disorders
WO2013134288A1 (fr) 2012-03-05 2013-09-12 Gilead Calistoga Llc Formes polymorphes de l'acide -2-(1-(9h-purine-6-ylamino)propyl)-5-fluoro-3-phénylquinazolin-4(3h)-one
US9359367B2 (en) 2012-07-09 2016-06-07 Lupin Limited Tetrahydroquinazolinone derivatives as PARP inhibitors
JP2017502021A (ja) 2013-12-20 2017-01-19 ギリアード カリストガ エルエルシー ホスファチジルイノシトール3−キナーゼ阻害剤のためのプロセス方法
JP2017500319A (ja) 2013-12-20 2017-01-05 ギリアード カリストガ エルエルシー (s)−2−(1−(9h−プリン−6−イルアミノ)プロピル)−5−フルオロ−3−フェニルキナゾリン−4(3h)−オンの塩酸塩の多形形態
CA2952012A1 (fr) 2014-06-13 2015-12-17 Gilead Sciences, Inc. Inhibiteurs de la phosphatidylinositol 3-kinase

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1053063A (fr) * 1963-05-18

Also Published As

Publication number Publication date
AT318615B (de) 1974-11-11
FR2100726B1 (fr) 1975-10-10
DE2027645A1 (de) 1971-12-09
US3984555A (en) 1976-10-05
CA951319A (en) 1974-07-16
BE768137A (fr) 1971-12-06
NL7107695A (fr) 1971-12-07
GB1331522A (en) 1973-09-26
CH558374A (de) 1975-01-31
FR2100726A1 (fr) 1972-03-24
AT317899B (de) 1974-09-25
LU63267A1 (fr) 1972-08-23
AT318628B (de) 1974-11-11
CH557829A (de) 1975-01-15

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Legal Events

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