FI956236A7 - Uusi menetelmä 17 beta-substituoitujen 4-atsa-androstaanijohdannaisten valmistamiseksi - Google Patents

Uusi menetelmä 17 beta-substituoitujen 4-atsa-androstaanijohdannaisten valmistamiseksi

Info

Publication number
FI956236A7
FI956236A7 FI956236A FI956236A FI956236A7 FI 956236 A7 FI956236 A7 FI 956236A7 FI 956236 A FI956236 A FI 956236A FI 956236 A FI956236 A FI 956236A FI 956236 A7 FI956236 A7 FI 956236A7
Authority
FI
Finland
Prior art keywords
aza
beta
substituted
preparation
new method
Prior art date
Application number
FI956236A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI956236A0 (fi
FI115837B (enExample
Inventor
Zoltan Tuba
Judit Horvath
Janos Szeles
Laszlo Kollar
Gabor Balogh
Original Assignee
Richter Gedeon Vegyeszet
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Richter Gedeon Vegyeszet filed Critical Richter Gedeon Vegyeszet
Publication of FI956236A0 publication Critical patent/FI956236A0/fi
Publication of FI956236A7 publication Critical patent/FI956236A7/fi
Application granted granted Critical
Publication of FI115837B publication Critical patent/FI115837B/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J73/00—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms
    • C07J73/001—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom
    • C07J73/005—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom by nitrogen as hetero atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J73/00—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
FI956236A 1993-06-24 1995-12-22 Uusi menetelmä 17 beta-substituoitujen 4-atsa-androstaanijohdannaisten valmistamiseksi FI956236A7 (fi)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/HU1993/000039 WO1995000531A1 (en) 1993-06-24 1993-06-24 NOVEL PROCESS FOR PREPARING 17β-SUBSTITUTED 4-AZAANDROSTANE DERIVATIVES

Publications (3)

Publication Number Publication Date
FI956236A0 FI956236A0 (fi) 1995-12-22
FI956236A7 true FI956236A7 (fi) 1995-12-22
FI115837B FI115837B (enExample) 2005-07-29

Family

ID=10982846

Family Applications (1)

Application Number Title Priority Date Filing Date
FI956236A FI956236A7 (fi) 1993-06-24 1995-12-22 Uusi menetelmä 17 beta-substituoitujen 4-atsa-androstaanijohdannaisten valmistamiseksi

Country Status (14)

Country Link
EP (1) EP0705272B1 (enExample)
JP (1) JP3253088B2 (enExample)
KR (1) KR100279567B1 (enExample)
AT (1) ATE215092T1 (enExample)
AU (1) AU681585B2 (enExample)
CA (1) CA2166090C (enExample)
DE (1) DE69331763T2 (enExample)
DK (1) DK0705272T3 (enExample)
ES (1) ES2173889T3 (enExample)
FI (1) FI956236A7 (enExample)
PT (1) PT705272E (enExample)
RU (1) RU2109746C1 (enExample)
UA (1) UA41933C2 (enExample)
WO (1) WO1995000531A1 (enExample)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU212459B (en) * 1992-10-02 1996-06-28 Richter Gedeon Vegyeszet Process for producing new 17-beta-substituted 4-aza-androstane-derivatives and pharmaceutical compositions containing them
ES2153789B1 (es) 1999-07-05 2001-10-16 Raga Consultores S L Procedimiento para la obtencion de 178-(n-terc-butlcarbamoil)-3-ona-4-aza-esteroides
US7351698B2 (en) 2003-05-07 2008-04-01 Merck & Co., Inc. Androgen receptor modulators and methods of use thereof

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU527030B2 (en) * 1978-04-13 1983-02-10 Merck & Co., Inc. 4-aza-17-substituted-5a-androstan-3-ones
SU930914A1 (ru) * 1980-03-07 1985-05-30 Институт биоорганической химии АН БССР Способ получени спин-меченых производных 8-аза-16-оксастероидов
IL74365A (en) * 1984-02-27 1990-07-26 Merck & Co Inc 17beta-(n-t.-butylcarbamoyl)-4-aza-5alpha-androst-1-en-3-one and pharmaceutical compositions containing it
US5120847A (en) * 1990-08-27 1992-06-09 Merck & Co., Inc. Process for iodinating or brominating the α-methylenic carbon of a secondary amide
GB9216329D0 (en) * 1992-07-31 1992-09-16 Erba Carlo Spa 17beta-substituted 4-aza-5alpha-androstan-3-one derivatives
GB9216284D0 (en) * 1992-07-31 1992-09-16 Erba Carlo Spa Fluorinated 17beta-substituted 4-aza-5alpha-androstane-3-one derivatives

Also Published As

Publication number Publication date
WO1995000531A1 (en) 1995-01-05
CA2166090C (en) 2006-01-24
DK0705272T3 (da) 2002-05-27
JP3253088B2 (ja) 2002-02-04
FI956236A0 (fi) 1995-12-22
ES2173889T3 (es) 2002-11-01
ATE215092T1 (de) 2002-04-15
JPH08511796A (ja) 1996-12-10
PT705272E (pt) 2002-07-31
EP0705272B1 (en) 2002-03-27
DE69331763D1 (de) 2002-05-02
UA41933C2 (uk) 2001-10-15
EP0705272A1 (en) 1996-04-10
FI115837B (enExample) 2005-07-29
KR100279567B1 (ko) 2001-03-02
RU2109746C1 (ru) 1998-04-27
CA2166090A1 (en) 1995-01-05
KR960703133A (ko) 1996-06-19
DE69331763T2 (de) 2002-10-02
AU4352693A (en) 1995-01-17
AU681585B2 (en) 1997-09-04

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