FI923575A - Foerfarande foer framstaellning av nya 1-acylpiperidinfoereningar - Google Patents

Foerfarande foer framstaellning av nya 1-acylpiperidinfoereningar Download PDF

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Publication number
FI923575A
FI923575A FI923575A FI923575A FI923575A FI 923575 A FI923575 A FI 923575A FI 923575 A FI923575 A FI 923575A FI 923575 A FI923575 A FI 923575A FI 923575 A FI923575 A FI 923575A
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FI
Finland
Prior art keywords
optionally
radical
optionally substituted
alkylene
alkanoyl
Prior art date
Application number
FI923575A
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English (en)
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FI104631B (fi
FI923575A0 (fi
Inventor
Walter Schilling
Silvio Ofner
Siem J Veenstra
Original Assignee
Ciba Geigy
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Application filed by Ciba Geigy filed Critical Ciba Geigy
Publication of FI923575A0 publication Critical patent/FI923575A0/fi
Publication of FI923575A publication Critical patent/FI923575A/fi
Priority to FI964117A priority Critical patent/FI964117A0/fi
Application granted granted Critical
Publication of FI104631B publication Critical patent/FI104631B/fi

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/56—Nitrogen atoms
    • C07D211/58—Nitrogen atoms attached in position 4
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
FI923575A 1991-08-12 1992-08-10 Menetelmä uusien 1-asyyli-2-aralkyyli-4-(alkyyli)-aminopiperidiiniyhdisteiden valmistamiseksi FI104631B (fi)

Priority Applications (1)

Application Number Priority Date Filing Date Title
FI964117A FI964117A0 (fi) 1991-08-12 1996-10-14 Menetelmä uusien 1-asyylipiperidiiniyhdisteiden valmistamiseksi

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH237491 1991-08-12
CH237491 1991-08-12

Publications (3)

Publication Number Publication Date
FI923575A0 FI923575A0 (fi) 1992-08-10
FI923575A true FI923575A (fi) 1993-02-13
FI104631B FI104631B (fi) 2000-03-15

Family

ID=4232283

Family Applications (1)

Application Number Title Priority Date Filing Date
FI923575A FI104631B (fi) 1991-08-12 1992-08-10 Menetelmä uusien 1-asyyli-2-aralkyyli-4-(alkyyli)-aminopiperidiiniyhdisteiden valmistamiseksi

Country Status (23)

Country Link
US (3) US5310743A (fi)
EP (1) EP0532456B1 (fi)
JP (1) JP3118090B2 (fi)
KR (1) KR100261367B1 (fi)
AT (1) ATE120456T1 (fi)
AU (1) AU660180B2 (fi)
CA (1) CA2075684C (fi)
DE (1) DE59201771D1 (fi)
DK (1) DK0532456T3 (fi)
ES (1) ES2070617T3 (fi)
FI (1) FI104631B (fi)
GR (1) GR3015954T3 (fi)
HU (1) HU221305B1 (fi)
IL (2) IL102769A (fi)
MX (1) MX9204627A (fi)
MY (1) MY110227A (fi)
NO (2) NO303448B1 (fi)
NZ (1) NZ243888A (fi)
PH (1) PH29963A (fi)
RU (1) RU2114829C1 (fi)
SA (1) SA94140632A (fi)
TW (1) TW204342B (fi)
ZA (1) ZA926013B (fi)

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NO303448B1 (no) 1998-07-13
ES2070617T3 (es) 1995-06-01
ZA926013B (en) 1993-03-31
JP3118090B2 (ja) 2000-12-18
NO973117L (no) 1993-02-15
US5646144A (en) 1997-07-08
MX9204627A (es) 1993-04-01
AU660180B2 (en) 1995-06-15
AU2096592A (en) 1993-03-04
US5541195A (en) 1996-07-30
RU2114829C1 (ru) 1998-07-10
KR100261367B1 (ko) 2000-07-01
CA2075684C (en) 2003-01-07
CA2075684A1 (en) 1993-02-13
FI104631B (fi) 2000-03-15
US5310743A (en) 1994-05-10
HUT67088A (en) 1995-01-30
NO923123D0 (no) 1992-08-11
SA94140632A (ar) 2005-12-03
NO973117D0 (no) 1997-07-04
HU221305B1 (en) 2002-09-28
MY110227A (en) 1998-03-31
DE59201771D1 (de) 1995-05-04
PH29963A (en) 1996-09-25
KR930004297A (ko) 1993-03-22
ATE120456T1 (de) 1995-04-15
NZ243888A (en) 1996-03-26
TW204342B (fi) 1993-04-21
JPH07196649A (ja) 1995-08-01
IL102769A (en) 1999-01-26
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IL102769A0 (en) 1993-01-31
EP0532456A1 (de) 1993-03-17
DK0532456T3 (da) 1995-06-12
FI923575A0 (fi) 1992-08-10
HU9202615D0 (en) 1992-10-28
NO923123L (no) 1993-02-15
EP0532456B1 (de) 1995-03-29
IL118750A0 (en) 1996-10-16

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