FI880265A - 1-substituoitujen (S)- ja (R)-2-aminometyylipyrrolidiinien tehokas, stereorakenteen säilyttävä synteesi sekä synteesin välituotteet - Google Patents
1-substituoitujen (S)- ja (R)-2-aminometyylipyrrolidiinien tehokas, stereorakenteen säilyttävä synteesi sekä synteesin välituotteet Download PDFInfo
- Publication number
- FI880265A FI880265A FI880265A FI880265A FI880265A FI 880265 A FI880265 A FI 880265A FI 880265 A FI880265 A FI 880265A FI 880265 A FI880265 A FI 880265A FI 880265 A FI880265 A FI 880265A
- Authority
- FI
- Finland
- Prior art keywords
- substituted
- aminomethylpyrrolidines
- stereostructured
- synthesis
- efficient
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
- C07D207/09—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pyrrole Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Peptides Or Proteins (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| SE8602339 | 1986-05-22 | ||
| SE8602339A SE8602339D0 (sv) | 1986-05-22 | 1986-05-22 | An efficient stereoconservative synthesis of 1-substituted (s)- and (r)-2-aminomethylpyrrolidines |
| PCT/SE1987/000246 WO1987007271A1 (en) | 1986-05-22 | 1987-05-19 | A stereoconservative synthesis of 1-substituted (s)- and (r)-2-aminomethylpyrrolidines and intermediates thereto |
| SE8700246 | 1987-05-19 |
Publications (4)
| Publication Number | Publication Date |
|---|---|
| FI880265A0 FI880265A0 (fi) | 1988-01-21 |
| FI880265A true FI880265A (fi) | 1988-01-21 |
| FI95028B FI95028B (fi) | 1995-08-31 |
| FI95028C FI95028C (fi) | 1995-12-11 |
Family
ID=20364616
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FI880265A FI95028C (fi) | 1986-05-22 | 1988-01-21 | 1-substituoitujen (S)- ja (R)-2-aminometyylipyrrolidiinien tehokas, stereorakenteen säilyttävä synteesi sekä synteesin välituotteet |
Country Status (12)
| Country | Link |
|---|---|
| EP (2) | EP0253785B1 (fi) |
| JP (1) | JPH07103098B2 (fi) |
| KR (1) | KR950011407B1 (fi) |
| AT (1) | ATE82259T1 (fi) |
| DE (2) | DE270596T1 (fi) |
| DK (1) | DK11788A (fi) |
| ES (1) | ES2044974T3 (fi) |
| FI (1) | FI95028C (fi) |
| GR (1) | GR3006609T3 (fi) |
| IE (1) | IE59896B1 (fi) |
| SE (1) | SE8602339D0 (fi) |
| WO (1) | WO1987007271A1 (fi) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE4425070A1 (de) * | 1994-07-15 | 1996-01-18 | Degussa | Verfahren zur Herstellung optisch aktiver l-substituierter 2-(Aminomethyl)pyrrolidine |
| CN1298702C (zh) * | 2005-03-15 | 2007-02-07 | 江苏省原子医学研究所 | 一种(s)－1－烯丙基－2－胺甲基四氢吡咯的制备方法 |
| JP6359365B2 (ja) * | 2014-07-09 | 2018-07-18 | 国立研究開発法人産業技術総合研究所 | アミノ酸のアミノ基及びカルボキシル基を対象としたプレカラム誘導体化ｌｃ−ｍｓ分析法 |
| CN107641092A (zh) * | 2017-10-30 | 2018-01-30 | 广东肇庆星湖生物科技股份有限公司 | 一种l‑脯氨酰胺的合成方法 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3718688A (en) * | 1967-10-18 | 1973-02-27 | Radio Carbon Lab | Alkylidine and arylidine amino acid esters, and alkyl and aryl amino acid esters |
| US3947408A (en) * | 1974-08-05 | 1976-03-30 | American Cyanamid Company | Pyrrolo-benzodiazepines, method of preparation and method of use |
| IL52645A (en) * | 1976-08-05 | 1980-02-29 | Synthelabo | Optically active 1 substituted 2 aminomethyl pyrrolidines stereospecifics synthesis thereof and process for the preparation of optically active 2 methoxy n pyrrolidylmethyl benzamides |
| IT1095415B (it) * | 1978-02-16 | 1985-08-10 | Ravizza Spa | Processo per la produzione di una benzamide otticamente attiva,benzamide otticamente attiva cosi'ottenuta e composizioni |
| FR2452482A1 (fr) * | 1979-03-28 | 1980-10-24 | Synthelabo | Derives de benzamides et leur application en therapeutique |
| US4525473A (en) * | 1983-03-30 | 1985-06-25 | Bristol-Myers Company | Cephalosporins |
| US4698336A (en) * | 1985-01-30 | 1987-10-06 | Eisai Co., Ltd. | 3-(pyrrolidinio)methyl-3-cephem derivatives |
-
1986
- 1986-05-22 SE SE8602339A patent/SE8602339D0/xx unknown
-
1987
- 1987-05-19 WO PCT/SE1987/000246 patent/WO1987007271A1/en active IP Right Grant
- 1987-05-19 KR KR1019880700061A patent/KR950011407B1/ko not_active IP Right Cessation
- 1987-05-19 DE DE198787903468T patent/DE270596T1/de active Pending
- 1987-05-19 EP EP87850165A patent/EP0253785B1/en not_active Expired - Lifetime
- 1987-05-19 DE DE8787850165T patent/DE3782566T2/de not_active Expired - Fee Related
- 1987-05-19 JP JP62503384A patent/JPH07103098B2/ja not_active Expired - Lifetime
- 1987-05-19 AT AT87850165T patent/ATE82259T1/de not_active IP Right Cessation
- 1987-05-19 EP EP87903468A patent/EP0270596A1/en active Pending
- 1987-05-19 ES ES87850165T patent/ES2044974T3/es not_active Expired - Lifetime
- 1987-05-20 IE IE132087A patent/IE59896B1/en not_active IP Right Cessation
-
1988
- 1988-01-12 DK DK011788A patent/DK11788A/da not_active Application Discontinuation
- 1988-01-21 FI FI880265A patent/FI95028C/fi not_active IP Right Cessation
-
1992
- 1992-12-21 GR GR920403017T patent/GR3006609T3/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| KR880701226A (ko) | 1988-07-26 |
| ATE82259T1 (de) | 1992-11-15 |
| FI95028B (fi) | 1995-08-31 |
| FI880265A0 (fi) | 1988-01-21 |
| EP0253785A1 (en) | 1988-01-20 |
| IE59896B1 (en) | 1994-04-20 |
| EP0270596A1 (en) | 1988-06-15 |
| WO1987007271A1 (en) | 1987-12-03 |
| JPS63503384A (ja) | 1988-12-08 |
| ES2044974T3 (es) | 1994-01-16 |
| SE8602339D0 (sv) | 1986-05-22 |
| JPH07103098B2 (ja) | 1995-11-08 |
| IE871320L (en) | 1987-11-22 |
| GR3006609T3 (fi) | 1993-06-30 |
| FI95028C (fi) | 1995-12-11 |
| EP0253785B1 (en) | 1992-11-11 |
| DK11788D0 (da) | 1988-01-12 |
| DE3782566T2 (de) | 1993-03-25 |
| DE3782566D1 (de) | 1992-12-17 |
| DE270596T1 (de) | 1988-10-13 |
| DK11788A (da) | 1988-01-12 |
| KR950011407B1 (ko) | 1995-10-04 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| BB | Publication of examined application | ||
| MM | Patent lapsed | ||
| MM | Patent lapsed |
Owner name: ASTRA LAEKEMEDEL AKTIEBOLAG |