FI782250A - Nya antagonistiska angiotensin ii-analoger med en alfa-aminooxisyra i 1-staellningen - Google Patents

Nya antagonistiska angiotensin ii-analoger med en alfa-aminooxisyra i 1-staellningen

Info

Publication number
FI782250A
FI782250A FI782250A FI782250A FI782250A FI 782250 A FI782250 A FI 782250A FI 782250 A FI782250 A FI 782250A FI 782250 A FI782250 A FI 782250A FI 782250 A FI782250 A FI 782250A
Authority
FI
Finland
Prior art keywords
staellningen
aminoxisyra
analoger
nya
angiotensin
Prior art date
Application number
FI782250A
Other languages
English (en)
Other versions
FI64140B (fi
FI64140C (fi
Inventor
Lajos Kisfaludy
Gyoergy Nyeki
Laszlo Szirmai
Egon Karpati
Katalin Gidai
Laszlo Szporny
Original Assignee
Richter Gedeon Vegyeszet
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Richter Gedeon Vegyeszet filed Critical Richter Gedeon Vegyeszet
Publication of FI782250A publication Critical patent/FI782250A/fi
Publication of FI64140B publication Critical patent/FI64140B/fi
Application granted granted Critical
Publication of FI64140C publication Critical patent/FI64140C/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04Linear peptides containing only normal peptide links
    • C07K7/14Angiotensins: Related peptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Vascular Medicine (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
FI782250A 1977-07-18 1978-07-14 Foerfarande foer framstaellning av nya terapeutiskt anvaendbara peptider FI64140C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
HU77RI640A HU177133B (en) 1977-07-18 1977-07-18 Process for preparing angiotensin ii analogues containing alpha- amino-oxy-acid in position 1 with angiotensin ii antagonist activity
HURI000640 1977-07-18

Publications (3)

Publication Number Publication Date
FI782250A true FI782250A (fi) 1979-01-19
FI64140B FI64140B (fi) 1983-06-30
FI64140C FI64140C (fi) 1983-10-10

Family

ID=11001037

Family Applications (1)

Application Number Title Priority Date Filing Date
FI782250A FI64140C (fi) 1977-07-18 1978-07-14 Foerfarande foer framstaellning av nya terapeutiskt anvaendbara peptider

Country Status (24)

Country Link
US (1) US4179433A (fi)
JP (1) JPS5835504B2 (fi)
AT (1) AT361143B (fi)
AU (1) AU518229B2 (fi)
BE (1) BE869077A (fi)
CA (1) CA1108124A (fi)
CH (1) CH637915A5 (fi)
CS (1) CS201014B2 (fi)
DD (1) DD137220A5 (fi)
DE (1) DE2831534C2 (fi)
DK (1) DK319478A (fi)
ES (1) ES471793A1 (fi)
FI (1) FI64140C (fi)
FR (1) FR2398050A1 (fi)
GB (1) GB2001653B (fi)
HU (1) HU177133B (fi)
IL (1) IL55121A (fi)
IN (1) IN149489B (fi)
NL (1) NL7807676A (fi)
NO (1) NO148031C (fi)
PL (1) PL111979B1 (fi)
SE (1) SE443790B (fi)
SU (1) SU845773A3 (fi)
YU (1) YU41431B (fi)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU181009B (en) * 1980-01-18 1983-05-30 Richter Gedeon Vegyeszet Process for preparing angiotensin-ii analogues with antagonictic activity containing in position 1 sarcosyl,hydroxyacetyl or l-alpha-aminoxy-propionyl group and in positiona 8 esteric group
HU181008B (en) * 1980-01-18 1983-05-30 Richter Gedeon Vegyeszet Process for producing angiotenzin-ii analogues of antagonistic activity containing sarcosyl-group at the 1-positon,and an alpha-hydroxy-carboxylic acid at the 8-position
HU191961B (en) * 1984-08-02 1987-04-28 Richter Gedeon Vegyeszet Process for producing 1,5 and 8 substituted peptides of angiotenzin-ii antagonistic activity
US5182264A (en) * 1986-03-07 1993-01-26 Schering Corporation Angiotensin II receptor blockers as antiglaucoma agents
US5036048A (en) * 1986-03-07 1991-07-30 Schering Corporation Angiotensin II receptor blockers as antiglaucoma agents
US4772684A (en) * 1987-01-20 1988-09-20 Triton Biosciences, Inc. Peptides affecting blood pressure regulation
TWI268138B (en) * 2000-05-11 2006-12-11 Kanebo Seiyaku Ltd Composition containing peptide and electrolyte excretion enhancing substance, and food containing the same
AT508569A1 (de) * 2009-07-23 2011-02-15 Affiris Ag Pharmaceutical compound

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3886134A (en) * 1970-03-09 1975-05-27 Morton Norwich Products Inc Analogues of angiotensin II
GB1320104A (en) * 1971-05-20 1973-06-13 Norwich Pharma Co Hepta-and octapeptides
US3907762A (en) * 1971-12-27 1975-09-23 Univ Sherbrooke Angiotensin{hd II {B position 8 analogs
HU167360B (fi) * 1972-08-25 1975-09-27
US3975365A (en) * 1975-01-27 1976-08-17 G. D. Searle & Co. Inhibitory octapeptides angiotensin II
US3976770A (en) * 1975-02-10 1976-08-24 Francis Merlin Bumpus Sar'-(OMe)Thr8 Angiotensin II as an angiotensin II antagonist

Also Published As

Publication number Publication date
BE869077A (fr) 1979-01-18
IL55121A0 (en) 1978-09-29
CS201014B2 (en) 1980-10-31
PL111979B1 (en) 1980-09-30
DK319478A (da) 1979-01-19
CA1108124A (en) 1981-09-01
HU177133B (en) 1981-07-28
PL208496A1 (pl) 1979-07-02
YU171378A (en) 1983-01-21
YU41431B (en) 1987-06-30
SE7807823L (sv) 1979-01-19
SU845773A3 (ru) 1981-07-07
GB2001653B (en) 1982-02-10
AU3800878A (en) 1980-01-17
DE2831534C2 (de) 1982-02-18
IN149489B (fi) 1981-12-26
NO148031B (no) 1983-04-18
DE2831534A1 (de) 1979-02-01
AT361143B (de) 1981-02-25
ES471793A1 (es) 1979-02-01
FI64140B (fi) 1983-06-30
FI64140C (fi) 1983-10-10
ATA518478A (de) 1980-07-15
FR2398050B1 (fi) 1983-09-09
NO782463L (no) 1979-01-19
DD137220A5 (de) 1979-08-22
IL55121A (en) 1981-09-13
SE443790B (sv) 1986-03-10
JPS54119463A (en) 1979-09-17
NL7807676A (nl) 1979-01-22
CH637915A5 (de) 1983-08-31
JPS5835504B2 (ja) 1983-08-03
GB2001653A (en) 1979-02-07
FR2398050A1 (fr) 1979-02-16
NO148031C (no) 1983-07-27
US4179433A (en) 1979-12-18
AU518229B2 (en) 1981-09-17

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Legal Events

Date Code Title Description
MM Patent lapsed

Owner name: RICHTER GEDEON VEGYESZETI GYOER R.T.