FI68836C - Foerfarande foer framstaellning av antibakteriella 5,8-dihydro-8-oxofuro(3,2-b)-1,8-naftyridiner - Google Patents

Foerfarande foer framstaellning av antibakteriella 5,8-dihydro-8-oxofuro(3,2-b)-1,8-naftyridiner Download PDF

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Publication number
FI68836C
FI68836C FI791839A FI791839A FI68836C FI 68836 C FI68836 C FI 68836C FI 791839 A FI791839 A FI 791839A FI 791839 A FI791839 A FI 791839A FI 68836 C FI68836 C FI 68836C
Authority
FI
Finland
Prior art keywords
formula
naphthyridine
dihydro
compound
alkyl
Prior art date
Application number
FI791839A
Other languages
English (en)
Finnish (fi)
Other versions
FI68836B (fi
FI791839A (fi
Inventor
Yoshiaki Tanaka
Isao Hayakawa
Original Assignee
Daiichi Seiyaku Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Daiichi Seiyaku Co filed Critical Daiichi Seiyaku Co
Publication of FI791839A publication Critical patent/FI791839A/fi
Publication of FI68836B publication Critical patent/FI68836B/fi
Application granted granted Critical
Publication of FI68836C publication Critical patent/FI68836C/fi

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/73—Unsubstituted amino or imino radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
    • C07D213/63—One oxygen atom
    • C07D213/65—One oxygen atom attached in position 3 or 5
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/74—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/12—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
    • C07D491/14—Ortho-condensed systems
FI791839A 1978-06-09 1979-06-08 Foerfarande foer framstaellning av antibakteriella 5,8-dihydro-8-oxofuro(3,2-b)-1,8-naftyridiner FI68836C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP6968578A JPS54163596A (en) 1978-06-09 1978-06-09 Flonaphlizine derivative
JP6968578 1978-06-09

Publications (3)

Publication Number Publication Date
FI791839A FI791839A (fi) 1979-12-10
FI68836B FI68836B (fi) 1985-07-31
FI68836C true FI68836C (fi) 1985-11-11

Family

ID=13409962

Family Applications (1)

Application Number Title Priority Date Filing Date
FI791839A FI68836C (fi) 1978-06-09 1979-06-08 Foerfarande foer framstaellning av antibakteriella 5,8-dihydro-8-oxofuro(3,2-b)-1,8-naftyridiner

Country Status (23)

Country Link
US (1) US4293695A (ja)
EP (1) EP0008610B1 (ja)
JP (1) JPS54163596A (ja)
AR (1) AR220561A1 (ja)
AT (1) AT373257B (ja)
AU (1) AU520081B2 (ja)
CA (1) CA1114822A (ja)
DD (1) DD144263A5 (ja)
DE (1) DE2906253C2 (ja)
DK (1) DK156773C (ja)
ES (1) ES481418A1 (ja)
FI (1) FI68836C (ja)
GR (1) GR68369B (ja)
IL (1) IL57423A (ja)
IN (1) IN150235B (ja)
IT (1) IT1117221B (ja)
MX (1) MX5725E (ja)
NZ (1) NZ190675A (ja)
PH (1) PH15905A (ja)
PL (1) PL116341B1 (ja)
SU (1) SU982544A3 (ja)
YU (1) YU41639B (ja)
ZA (1) ZA792467B (ja)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2666219C (en) 2006-10-16 2017-02-07 Bionomics Limited Novel anxiolytic compounds
US10954231B2 (en) 2006-10-16 2021-03-23 Bionomics Limited Anxiolytic compounds
WO2012116415A1 (en) 2011-03-02 2012-09-07 Bionomics Limited Novel small-molecules as therapeutics
CA2835450C (en) 2011-05-12 2020-05-12 Bionomics Limited Methods for preparing naphthyridines

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3149104A (en) * 1961-01-03 1964-09-15 Sterling Drug Inc 4-hydroxy-7-styryl-1, 8-naphthyridine-3-carboxylic acids and esters
US3663559A (en) * 1969-12-03 1972-05-16 Union Carbide Corp Preparation of oxo-furo-pyridines from furylvinyl isocyanates
DE2030899A1 (de) * 1970-06-18 1971-12-23 Schering Ag, 1000 Berlin Und 4619 Bergkamen Chinolincarbonsäurederivate
JPS5035194A (ja) * 1973-07-19 1975-04-03
US4079058A (en) * 1973-08-29 1978-03-14 Dynamit Nobel Ag Process of performing cyclization reactions using benzyl or pyridylamino malonic acid derivatives

Also Published As

Publication number Publication date
AU4736379A (en) 1979-12-13
IL57423A (en) 1982-02-28
IL57423A0 (en) 1979-09-30
FI68836B (fi) 1985-07-31
CA1114822A (en) 1981-12-22
AT373257B (de) 1984-01-10
DK156773B (da) 1989-10-02
DD144263A5 (de) 1980-10-08
GR68369B (ja) 1981-12-23
IT1117221B (it) 1986-02-17
ATA405879A (de) 1983-05-15
DE2906253C2 (de) 1983-06-09
JPS54163596A (en) 1979-12-26
PL116341B1 (en) 1981-06-30
YU134779A (en) 1983-06-30
DE2906253A1 (de) 1979-12-13
US4293695A (en) 1981-10-06
YU41639B (en) 1987-12-31
IT7949343A0 (it) 1979-06-07
ZA792467B (en) 1980-07-30
DK156773C (da) 1990-03-19
EP0008610A1 (en) 1980-03-19
SU982544A3 (ru) 1982-12-15
AR220561A1 (es) 1980-11-14
FI791839A (fi) 1979-12-10
DK240179A (da) 1979-12-10
MX5725E (es) 1983-12-28
NZ190675A (en) 1981-03-16
PL216219A1 (ja) 1980-03-24
PH15905A (en) 1983-04-15
IN150235B (ja) 1982-08-21
ES481418A1 (es) 1980-10-01
AU520081B2 (en) 1982-01-14
EP0008610B1 (en) 1981-10-14
JPS6216955B2 (ja) 1987-04-15

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