FI65432C - Foerfarande foer framstaellning av antibakteriella 7beta-arylmalonamido-7alfa-metoxi-3-tiadiazolyltiometyl-1-detia-1-oxa-3-cefem-4-karbonsyror eller derivat daerav - Google Patents

Foerfarande foer framstaellning av antibakteriella 7beta-arylmalonamido-7alfa-metoxi-3-tiadiazolyltiometyl-1-detia-1-oxa-3-cefem-4-karbonsyror eller derivat daerav Download PDF

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Publication number
FI65432C
FI65432C FI782586A FI782586A FI65432C FI 65432 C FI65432 C FI 65432C FI 782586 A FI782586 A FI 782586A FI 782586 A FI782586 A FI 782586A FI 65432 C FI65432 C FI 65432C
Authority
FI
Finland
Prior art keywords
methoxy
oxa
detia
acid
compound
Prior art date
Application number
FI782586A
Other languages
English (en)
Finnish (fi)
Other versions
FI65432B (fi
FI782586A (fi
Inventor
Masayuki Narisada
Wataru Nagata
Original Assignee
Shionogi & Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Shionogi & Co filed Critical Shionogi & Co
Publication of FI782586A publication Critical patent/FI782586A/fi
Publication of FI65432B publication Critical patent/FI65432B/fi
Application granted granted Critical
Publication of FI65432C publication Critical patent/FI65432C/fi

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D505/00—Heterocyclic compounds containing 5-oxa-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. oxacephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
FI782586A 1977-08-25 1978-08-24 Foerfarande foer framstaellning av antibakteriella 7beta-arylmalonamido-7alfa-metoxi-3-tiadiazolyltiometyl-1-detia-1-oxa-3-cefem-4-karbonsyror eller derivat daerav FI65432C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP52102261A JPS609718B2 (ja) 1977-08-25 1977-08-25 チアジアゾリルチオセフアロスポリン類縁抗生物質
JP10226177 1977-08-25

Publications (3)

Publication Number Publication Date
FI782586A FI782586A (fi) 1979-02-26
FI65432B FI65432B (fi) 1984-01-31
FI65432C true FI65432C (fi) 1984-05-10

Family

ID=14322642

Family Applications (1)

Application Number Title Priority Date Filing Date
FI782586A FI65432C (fi) 1977-08-25 1978-08-24 Foerfarande foer framstaellning av antibakteriella 7beta-arylmalonamido-7alfa-metoxi-3-tiadiazolyltiometyl-1-detia-1-oxa-3-cefem-4-karbonsyror eller derivat daerav

Country Status (34)

Country Link
US (1) US4201782A (it)
JP (1) JPS609718B2 (it)
AR (1) AR220539A1 (it)
AT (1) AT361121B (it)
AU (1) AU517618B2 (it)
BE (1) BE869955A (it)
BG (1) BG34338A3 (it)
CA (1) CA1101417A (it)
CH (1) CH637396A5 (it)
CS (1) CS203927B2 (it)
DD (1) DD137230A5 (it)
DE (1) DE2837264A1 (it)
DK (1) DK372878A (it)
ES (1) ES472817A1 (it)
FI (1) FI65432C (it)
FR (1) FR2401165A1 (it)
GB (1) GB1576796A (it)
GR (1) GR70260B (it)
HU (1) HU177900B (it)
IE (1) IE47630B1 (it)
IL (1) IL55429A0 (it)
IT (1) IT1118098B (it)
MX (1) MX5328E (it)
NL (1) NL190554C (it)
NO (1) NO782866L (it)
NZ (1) NZ188173A (it)
PH (1) PH17508A (it)
PL (1) PL110656B1 (it)
PT (1) PT68434A (it)
RO (1) RO75070A (it)
SE (1) SE452010B (it)
SU (1) SU812182A3 (it)
YU (1) YU43999B (it)
ZA (1) ZA784753B (it)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4259485A (en) * 1979-04-24 1981-03-31 Eli Lilly And Company Crystallization process
FR2494279A1 (fr) * 1980-11-20 1982-05-21 Rhone Poulenc Ind Nouvelles oxacephalosporines, leur preparation et les medicaments qui les contiennent
EP0112049B1 (en) * 1982-12-14 1987-09-09 Beecham Group Plc Process for the preparation of beta-lactam compounds
JPS60123490A (ja) * 1983-12-07 1985-07-02 Shionogi & Co Ltd マロニルオキサセフェムカルボン酸誘導体
US6013835A (en) * 1995-06-07 2000-01-11 Hfm International, Inc. Method and apparatus for preparing purified terephthalic acid
US6197794B1 (en) 1998-01-08 2001-03-06 Celltech Therapeutics Limited Phenylalanine derivatives
US6329372B1 (en) 1998-01-27 2001-12-11 Celltech Therapeutics Limited Phenylalanine derivatives
US6555562B1 (en) 1998-02-26 2003-04-29 Celltech R&D Limited Phenylalanine derivatives
GB9805655D0 (en) 1998-03-16 1998-05-13 Celltech Therapeutics Ltd Chemical compounds
US6521626B1 (en) 1998-03-24 2003-02-18 Celltech R&D Limited Thiocarboxamide derivatives
GB9811159D0 (en) 1998-05-22 1998-07-22 Celltech Therapeutics Ltd Chemical compounds
GB9811969D0 (en) 1998-06-03 1998-07-29 Celltech Therapeutics Ltd Chemical compounds
GB9812088D0 (en) 1998-06-05 1998-08-05 Celltech Therapeutics Ltd Chemical compounds
GB9814414D0 (en) 1998-07-03 1998-09-02 Celltech Therapeutics Ltd Chemical compounds
GB9821061D0 (en) 1998-09-28 1998-11-18 Celltech Therapeutics Ltd Chemical compounds
GB9821222D0 (en) 1998-09-30 1998-11-25 Celltech Therapeutics Ltd Chemical compounds
GB9821406D0 (en) * 1998-10-01 1998-11-25 Celltech Therapeutics Ltd Chemical compounds
GB9825652D0 (en) 1998-11-23 1999-01-13 Celltech Therapeutics Ltd Chemical compounds
US6518283B1 (en) 1999-05-28 2003-02-11 Celltech R&D Limited Squaric acid derivatives
US6534513B1 (en) 1999-09-29 2003-03-18 Celltech R&D Limited Phenylalkanoic acid derivatives
US6455539B2 (en) 1999-12-23 2002-09-24 Celltech R&D Limited Squaric acid derivates
WO2001079173A2 (en) 2000-04-17 2001-10-25 Celltech R & D Limited Enamine derivatives as cell adhesion molecules
US6403608B1 (en) 2000-05-30 2002-06-11 Celltech R&D, Ltd. 3-Substituted isoquinolin-1-yl derivatives
US6545013B2 (en) 2000-05-30 2003-04-08 Celltech R&D Limited 2,7-naphthyridine derivatives
EP1301488A1 (en) 2000-07-07 2003-04-16 Celltech R&D Limited Squaric acid derivatives containing a bicyclic heteroaromatic ring as integrin antagonists
US6649756B2 (en) * 2000-07-13 2003-11-18 Wyeth, Five Giralda Farms Process improvement in the preparation of (4r, 5s, 6s)-3-[[(2r,3r)-2-[[[(s)-2-amino-3-methyl-1-oxobutyl]amino]methyl]tetrahydro-3-furanyl]thio]-6-[(r)-1-hydroxyethyl]-4-methyl-7-oxo-1-azabicyclo[3.2.0]hept-2-ene-2-carboxylic acid
CA2417059A1 (en) 2000-08-02 2002-02-07 Celltech R&D Limited 3-substituted isoquinolin-1-yl derivatives
CN102827191B (zh) * 2012-09-24 2015-03-11 浙江东邦药业有限公司 一种氧头孢类化合物的制备方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL178005C (nl) * 1972-11-06 1986-01-02 Merck & Co Inc Werkwijze voor het bereiden van een farmaceutisch preparaat met antibacteriele werking, alsmede werkwijze ter bereiding van een cefalosporine-antibioticum.
US4031083A (en) * 1975-10-24 1977-06-21 Yeda Research And Development Co., Ltd. Cephalosporin antibiotics
US4045438A (en) * 1975-10-24 1977-08-30 Yeda Research And Development Co. Ltd. Cephalosporin antibiotics
CA1070688A (en) * 1975-11-12 1980-01-29 Mitsuru Yoshioka Cephalosporin analogues
CA1085392A (en) * 1976-03-25 1980-09-09 Masayuki Narisada Arylmalonamido-1-oxadethiacephalosporins

Also Published As

Publication number Publication date
IE781703L (en) 1979-02-25
YU202878A (en) 1982-10-31
FR2401165A1 (fr) 1979-03-23
FR2401165B1 (it) 1982-06-25
AT361121B (de) 1981-02-25
CH637396A5 (de) 1983-07-29
NO782866L (no) 1979-02-27
IE47630B1 (en) 1984-05-16
DE2837264A1 (de) 1979-03-01
DD137230A5 (de) 1979-08-22
NL7808802A (nl) 1979-02-27
ES472817A1 (es) 1979-02-16
NL190554B (nl) 1993-11-16
BG34338A3 (en) 1983-08-15
GR70260B (it) 1982-09-02
PL110656B1 (en) 1980-07-31
DK372878A (da) 1979-02-26
SE452010B (sv) 1987-11-09
RO75070A (ro) 1980-10-30
US4201782A (en) 1980-05-06
PL209215A1 (pl) 1979-06-04
AU517618B2 (en) 1981-08-13
BE869955A (fr) 1978-12-18
GB1576796A (en) 1980-10-15
AU3923878A (en) 1980-02-28
PH17508A (en) 1984-09-07
JPS609718B2 (ja) 1985-03-12
IT1118098B (it) 1986-02-24
YU43999B (en) 1990-02-28
IL55429A0 (en) 1978-10-31
HU177900B (en) 1982-01-28
NL190554C (nl) 1994-04-18
CS203927B2 (en) 1981-03-31
SE7808950L (sv) 1979-02-26
SU812182A3 (ru) 1981-03-07
ATA620378A (de) 1980-07-15
IT7868975A0 (it) 1978-08-24
AR220539A1 (es) 1980-11-14
JPS5436288A (en) 1979-03-16
NZ188173A (en) 1981-05-15
DE2837264C2 (it) 1991-06-13
PT68434A (en) 1978-09-01
FI65432B (fi) 1984-01-31
FI782586A (fi) 1979-02-26
ZA784753B (en) 1979-08-29
MX5328E (es) 1983-06-22
CA1101417A (en) 1981-05-19

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Owner name: SHIONOGI & CO LTD